CNS Drugs: Classes Flashcards
What class?
Disulfiram Diazepam Chlordiazepoxide Lorazepam Phenytoin Naltrexone Acamprostate Topiramate
EtOH Abuse
Benzodiazepine Antagonist
Flumazenil
BZ that doesn’t follow the “pam” suffix…
chlordiazepoxide
Zolpidem
Zaleplon
Eszopiclone
Z-Drugs - sedative hypnotics
Melatonin Analogue
Ramelteon
Orexin Receptor Antagonist
Suvorexant
Buspirone
anxiolytic
Phenytoin
Carbamazepine
Lamotrigine
Topiramate
Levetiracetam
Anticonvulsant - Decrease Glutamate
Tigabine
Vigabatrin
Phenobarbital
Gabapentin
Pregabalin
Anticonvulsant - increase GABA
Ethosuximide
Valproic Acid
Anticonvulsant - CCB, decreased glutamate
Absence seizure drugs
Ethosuximide (Zarontin®)
Valproic acid (Depakene®)
Clonazepam (Klonopin®)
Status Epilepticus Drugs
Diazepam (Valium®)
Lorazepam (Ativan®)
What type of seizures?
Phenytoin (Dilantin®) Fosphenytoin (Cerebyx®) Carbamazepine (Tegretol®) Phenobarbital (Luminal®) Gabapentin (Neurontin®) Pregabalin (Lyrica®) Levetiracetam (Keppra®) Lamotrigine (Lamictal®) Topiramate (Topamax®) Tiagabine (Gabatril®) Vigabatrin (Sabril®)
partial seizures and generalized tonic-clonic seizures
What type of local anesthetic?
Procaine (Novocain®)
Tetracaine (Pontocaine®)
Benzocaine (Americaine®)
Cocaine
Ester
What type of local anesthetic?
Lidocaine (Xylocaine®) Prilocaine (Citanest®) Bupivacaine (Marcaine®) Mepivacaine (Carbocaine®) Ropivacaine (Naropin®) Etidocaine (Duranest®) Articaine (Septocaine®) Dibucaine (Nupercainal®)
Amide
Spinal cord or brain stem sedatives (2)
Cyclobenzaprine (Flexeril®)
Carisoprodol (Soma®)
GABA Mimetic muscle relaxant
Baclofen (Lioresal®)
Tizanidine (Zanaflex®)
Dantrolene (Dantrium®)
muscle relaxant