CNS Drugs: Classes Flashcards
What class?
Disulfiram Diazepam Chlordiazepoxide Lorazepam Phenytoin Naltrexone Acamprostate Topiramate
EtOH Abuse
Benzodiazepine Antagonist
Flumazenil
BZ that doesn’t follow the “pam” suffix…
chlordiazepoxide
Zolpidem
Zaleplon
Eszopiclone
Z-Drugs - sedative hypnotics
Melatonin Analogue
Ramelteon
Orexin Receptor Antagonist
Suvorexant
Buspirone
anxiolytic
Phenytoin
Carbamazepine
Lamotrigine
Topiramate
Levetiracetam
Anticonvulsant - Decrease Glutamate
Tigabine
Vigabatrin
Phenobarbital
Gabapentin
Pregabalin
Anticonvulsant - increase GABA
Ethosuximide
Valproic Acid
Anticonvulsant - CCB, decreased glutamate
Absence seizure drugs
Ethosuximide (Zarontin®)
Valproic acid (Depakene®)
Clonazepam (Klonopin®)
Status Epilepticus Drugs
Diazepam (Valium®)
Lorazepam (Ativan®)
What type of seizures?
Phenytoin (Dilantin®) Fosphenytoin (Cerebyx®) Carbamazepine (Tegretol®) Phenobarbital (Luminal®) Gabapentin (Neurontin®) Pregabalin (Lyrica®) Levetiracetam (Keppra®) Lamotrigine (Lamictal®) Topiramate (Topamax®) Tiagabine (Gabatril®) Vigabatrin (Sabril®)
partial seizures and generalized tonic-clonic seizures
What type of local anesthetic?
Procaine (Novocain®)
Tetracaine (Pontocaine®)
Benzocaine (Americaine®)
Cocaine
Ester
What type of local anesthetic?
Lidocaine (Xylocaine®) Prilocaine (Citanest®) Bupivacaine (Marcaine®) Mepivacaine (Carbocaine®) Ropivacaine (Naropin®) Etidocaine (Duranest®) Articaine (Septocaine®) Dibucaine (Nupercainal®)
Amide
Spinal cord or brain stem sedatives (2)
Cyclobenzaprine (Flexeril®)
Carisoprodol (Soma®)
GABA Mimetic muscle relaxant
Baclofen (Lioresal®)
Tizanidine (Zanaflex®)
Dantrolene (Dantrium®)
muscle relaxant
Amitriptyline
Imipramine
TCAs - Tertiary Amines
Nortriptyline
Desipramine
TCAs - Secondary Amines
Phenelzine
Selegiline
MAOIs
Fluoxetine Paroxetine Sertraline Citalopram Escitalopram
SSRI
Venlafaxine
Duloxetine
SNRI
DA reuptake inhibitor
Bupropion
NE Reuptake Inhibitor
Atomoxetine
5HT2A Antagonist
Trazodone
Chlorpromazine (Thorazine®)
Prochlorperazine (Compazine®)
Fluphenazine (Prolixin®)
Classic Antipsychotics
Clozapine (Clozaril®) Olanzapine (Zyprexa®) Quetiapine (Seroquel®) Aripiprazole (Abilify®) Risperidone (Risperdal®) Ziprisadone (Geodon®) Lurasidone (Latuda®)
Atypical Antipsychotics
Valproic acid (Depakene®)
Carbamazepine (Tegretol®)
Gabapentin (Neurontin®)
Lamotrigine (Lamictal®)
Mood Stabilizers
- Heroin
- Morphine
- Hydromorphone(Dilaudid)
- Methadone(Dolophine)
- Meperidine(Demerol)
- Fentanyl(Sublimaze)
Strong Opioid
Hydrocodone(Codan)
•Oxycodone(OxyContin)
Oxymorphone (Opana)
Moderate to Strong Opioid
- Codeine
* Tramadol (Ultram)
Weak Moderate opioid
Pentazocine/naloxone(Talwin NX)
•Buprenorphine(Buprenex); buprenorphine/naloxone (Suboxone)
Mixed opioid agonist-antagonist
Dextromethorphan (with guaifenesin; Robitussin DM)
•Codeine
antitussive
Hydrocodone/acetaminophen (Vicodin)
•Oxycodone/acetaminophen (Percoset)
Combination opioids
- Naloxone(Narcan)
* Naltrexone(ReVia)
opioid antagonists
The below drugs treat…
Levodopa
Carbidopa
parkinson’s
The below are what class of parkinson’s drug?
Selegiline (Deprenyl®)
Rasagiline (Azilect®)
Safinaminde (Xadago®)
MAOI
Tolcapone (Tasmar®)
Entacapone (Comtan®)
COMT Inhibitor, parkinson’s
Bromocriptine (Parlodel®)
Pramipexole (Mirapex®)
Ropinirole (Requip®) Apomorphine (Apokyn®)
DA Receptor Agonists
Amantadine (Symmetrel®)
Pimavanserin (Nuplazid®)
Benztropine (Cogentin®)
DA releasers
Anticholinergic for Parkinson’s
Benztropine (Cogentin®)
Donepezil
Rivastigmine
Galantamine
Memantine
Alzheimer’s drugs
Cocaine
Amphetamine
Methamphetamine
Nicotine
CNS Stimulants
Bupropion (Zyban®)
Varenicline (Chantix®)
nicotine addiction