CHOLINORECEPTOR ACTIVATING AND CHOLINESTRASE INHIBITING DRUGS Flashcards
choline esters
A
M
C
B
acetylcholine
metacholine
carbachol
betanechol
muscarinic alkaloids
M
A
P
O
muscarine
arecoline
pilocarpine
oxotremonine
nicotinic alkaloids
N
L
D
nicotine
lobeline
dmpp
reversible indirect acting cholinomimetics
Inhibits the breakdown of Ach:
N
P
P
neostigmine
physostigmine
pyridostigmine
irreversible indirect acting
E
S
S
echothiopate
parathion
sarin
_______– is a nicotinic partial agonist
it appears to reduce craving in persons addicted to nicotine by causing smaller amounts of dopamine release compared to nicotine itself
varenicline
___________ a carbamate and several others are used exclusively in alzheimer’s disease
rivastigmine
____________ used for the rapid reversal of nondepolarizing neuromuscular blockade____
endrophonium
the antidote of first choice is the antimuscarinic agent __________
atropine