Cholinergic and Adrenergic Drugs Flashcards
Phenylephrine
Selective Alpha-1 Agonist
Oxymetazoline
Selective Alpha-1 Agonist
Naphazoline
Selective Alpha-1 Agonist
Clonidine
Selective Alpha-2 Agonist (sympatholytic)
Guanfacine
Selective Alpha-2 Agonist (sympatholytic)
Fenoldopam
Selective DA-1 Agonist
Methyldopa
Partial Agonist of Adrenergic Receptors
Phenoxybenzamine
Irreversible Non-selective Alpha Antagonist
Phentolamine
Reversible non-selective Alpha Antagonist
Prazosin
Selective Alpha-1 Antagonist
Terazosin
Selective Alpha-1 Antagonist
Ephedrine
Stimulate α & β receptors AND release stored NE from nerve terminals
Pseudoephedrine
Stimulate α & β receptors AND release stored NE from nerve terminals
Isoproterenol
Nonselective Beta-1/2 Agonist
Dobutamine
Selective Beta-1 Agonist (B1>B2,A)
Albuterol
Selective Beta-2 Agonist (B2>B1)
Metaproterenol
Selective Beta-2 Agonist
Terbutaline
Selective Beta-2 Agonist
Ritodrine
Selective Beta-2 Agonist
Propranolol
Nonselective Beta-1/2 Antagonist
Carteolol
Nonselective Beta-1/2 Antagonist
Nadolol
Nonselective Beta-1/2 Antagonist
Pindolol
Nonselective Beta-1/2 Partial Antagonist
Atenolol
Selective Beta-1 Antagonist
Metoprolol
Selective Beta-1 Antagonist
Beta-arrestin signaling pathway agonist
Bisoprolol
Selective Beta-1 Antagonist
Beta-arrestin signaling pathway agonist
Esmolol
Short-acting Beta-1 Antagonist
Carvedilol
Beta-1/2, Alpha-1 Antagonist
Beta-arrestin signaling pathway agonist
Labetalol
Beta-1/2, Alpha-1 Antagonist
Entacapone
Catechol-O-methyltransferase Inhibitor
Isocarboxazid
Monoamine Oxidase Inhibitor
Selegiline
Monoamine Oxidase Inhibitor
Carbidopa
Dopa-decarboxylase Inhibitor
Benserazide
Dopa-decarboxylase Inhibitor
Norepinephrine
Alpha-1/2; Beta-1 agonist (A1 > A2 > B1)
Epinephrine
Alpha-1/2, Beta-1/2 agonist (B>A)
Bethanechol
Cholinergic agonist
Carbachol
Cholinergic agonist
Methacholine
Muscarinic agonist
Pilocarpine
Cholinergic agonist
Galantamine
AChE inhibitor
Donepezil
AChE inhibitor
Rivastigmine
AChE inhibitor
Edroponium
AChE inhibitor
Neostigmine
AChE inhibitor
Physostigmine
AChE inhibitor (BBB penetration)
Pyridostigmine
AChE inhibitor
Atropine
Muscarinic antagonist
homatropine
Muscarinic antagonist
tropicamide
Muscarinic antagonist
Benztropine
Muscarinic antagonist
trihexyphenidyl
Muscarinic antagonist
glycopyrrolate
Muscarinic antagonist
hyoscyamine
Muscarinic antagonist
dicyclomine
Muscarinic antagonist
ipratropium
Muscarinic antagonist
tiotropium
Muscarinic antagonist
oxybutynin
Muscarinic antagonist
solifenacin
Muscarinic antagonist
tolterodine
Muscarinic antagonist
scopolamine
Muscarinic antagonist
Fendolapam
D1 agonist
isoproterenol
Beta agonist (B1=B2)
midrodrine
alpha-1 agonist
Mirabegron
B3 agonist
mirtazapine
Alpha 2 Antagonist
acebutolol
B1 selective partial agonist
nebivolol
B1 antagonist, B3 agonist