Adrenoceptor agonist Flashcards
Adrenoceptor agonist
drugs that binds with adrenoceprtor receptors and causes physiological changes
adrenoceptor receptors are
alpha and Beta
alpha1 and 2
beta 1 and 2
alpha 1
contraction of smooth muscle/exocrine gland/neuronal excitation
alpha 2
inhibits NE release
CNS effect
Beta 1
increase renin secretion
increase HR
increase contractility and conduction
Beta 2
bronchodialation
relaxation of smooth muscle
glycogenolysis
3 types of adrenoceptor agonist
Direct Catecholamine
Direct noncatecholamine
indirect
mixed
Direct Catecholamine 1
Dobutamine
Dobutamine
B1,B2
Direct catecholamine 2
Dopamine
Dopamine
A2
Direct catecholamine 3
Epinephrine
Epinephrine
b1,b2,a1,D1
Direct catecholamine 4
Noepinephrine
norepinephrine
a1
Direct catecholamine 5
isoproterenol
isoproterenol
b1,b2
Direct noncatecholamine 1
albuterol
Albuterol
b2
direct noncatecholamine 2
clonidine
Clonidine
a2
direct noncatecholamine 3
midodrine
midodrine
a1
Direct catecholamine 4
oxymetazoine
oxymetazoine
a1
direct noncatecholamine 5
phenylephrine
phenylephrine
a1
direct noncatecholamine 6
terbutaline
Terbutaline
B2
Indirect acting adrenceptror agonist
amphetamine/cocaine
amphetamine
increase NE release
cocaine
Inhibits NE uptake
mixed acting adrenoceptor agonist
Ephedrine/pseudoephedrine
Ephedrine
A1 receptor/increase synaptic release of NE
Pseudoephedrine
A1 receptor/increase synaptic release of NE