Tertiary Amine TCAs Flashcards by Sean Mlodzinski | Brainscape

Q

imipramine (Tofranil)

A

Tertiary amine TCA

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Q

amitryptyline (Elavil)

A

Tertiary amine TCA

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Q

doxepin (Sinequan)

A

Tertiary amine TCA

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Q

trimipramine (Surmontil)

A

Tertiary amine TCA

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Q

clominipramine (Anafrantil)

A

-approved for child OCD but very anticholinergic so SSRIs used first

Tertiary amine TCA

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Q

All tertiary amine TCAs

A

5HT
downregulate NE and 5HT2A receptors
inhibit reuptake via NET and SERT transporters

SE: antiarrhythmatic, lethal in overdose, sedation, weight gain, hypertension

H1 block, M1, alpha1, alpha2, 5HT2, 5HT3

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