Pharma Final Drug Names Flashcards
Direct Parasympathomimetics
ACh Carbachol Pilocarpine Bethanacol (Hu) Methacoline (Hu)
Indirect Parasympathomimetics
Physostigmine Neostigmine Pyridostigmine Edrophonium (Tensilon) Organophosphates: Diazinon (ectoparasiticide) and Echothiophate
Parasympatholytics
Atropine! Tropicamide Homatropine Ipratropium Glycopyrrolate Benzethimide Butyl scopalamine
Non-specific sympathomimetics
Adrenaline/ Epinephrine
Noradrenaline/ Norepinephrine
Dopamine
Specific Sympathomimetics: Beta1 Adrenoreceptor agonists
Dobutamine
Specific Sympathomimetics: Beta2 Adrenoreceptor Agonists
Clenbutarole Salbutamole Terbutarole Salmeterole Isoxsuprine
Specific Sympathomimetics: Alpha1 Adrenoreceptor Agonists
Phenylephrine
Xylometazoline, Oxymetazoline, Naphazoline, Tetrazoline
Phenylpropanolamine
Ephedrine
Specific Sympathomimetics: Alpha2 Adrenoreceptor Agonists
Xylazine
Detomidine
Medetomidine
Sympatholytics: Alpha
Phenoxybenzamine (non-specific)
Prazosine, Doxasosine (specific alpha1)
Atipamezole, Yohimbine (specific alpha2)
Sympatholytics: Beta
Propanole, Timolol (non-specific)
Atenolole, Metapronole (specific beta1)
Tranquilizer Sedatives
Phenothiazine and Butyrophenone derivatives
Phenothiazine Derivatives
Chlorpromazine Propionyl-promazine Acepromazine Promethazine Trifluorperazine Proquamezine
Butyrophenone Derivatives
Azaperone
Droperidol
Haloperidol
Fluanison
Alpha-2-agonists
Xylazine Detomidine Medetomidine Dexmedetomidine Romifidine
Alpha-2-Antagonists
Atipamezole
Yohimbine
Benzodiazepines
Diazepam
Midazolam
Clonazepam
Barbiturates
Long: Phenobarbital
Short: Pentobarbital
Ultra-short: Thiopental, Thiomylal, Methohexital
Proprandiol derivatives
Meprobamate
The sedato-hypnotics
Alpha-2-agonists
Benzodiazepines
Proprandiol derivs
Barbiturates
Endogenous Opioids:
Opiopeptins!
Encephalins
Endorphins
Semisynth Opioids
Azidomorphine Ethylmorphine Etorphine Heroin Burenorphine Hydro- and Oxycodone Hydro- and Oxymorphone
Synth Opioids
Morphinanes: Butorphanol Diphenyl heptanes: Methadone Phenylpiperidines: Pethidine, Fentanyl, Diphenoxylate, Loperamide Benzomorphanes: Pentazocine Cyclohexanols: Tramadol
Opioid Active substances:
Morphine Fentanyl Sulfetanyl and Remifentanyl Tramadol Buprenorphine Butorphanol
Neuroleptanalgesia
Tranquilizer and opiate
Ataranalgesia
BZD and opiate
Inhalational Anaesthetics
Halothane Isoflurane Sevoflurane Desflurane N2O
Injectable Anaesthetics
Barbiturates Propofol Imidazoles Dissociative Anaesthetics Steroid Anaesthetics
Imidazoles
Etomidate
Metomidate
Dissociative Anaesthetics
Ketamine
Tiletamine
Steroid Anaesthetics
Alfaxlon
Alfadolon
Anticonvulsants: Barbiturates
Phenobarbital
Pentobarbital
Primidone
Anticonvulsants: Benzodiazepines
Diazepam
Clonazepam
Carbamazepin
Anticonvulsants: Others
Phenytoin
Valproic acid
Treatment of status epilepticus
Diazepam
Phenobarbital (pentobarbital)
Propofol
Prevention of seizures: Maintenance
Phenobarbital Phenytoin Valproic acid Bromide salts (Na, K) Clonazepam Clorazepate Felbamate Gabapentin Primidone
Active sunstances: Anticonvulsants
Phenobarbital Diazepam Clonazepam Sodium potassium bromide Phenytoin Carbamazepine Sodium Valproate Gabapentin
Antidepressants
Tricyclic Antidepressants (TCA’s)
Serotonin Reuptake Inhibitors (SRI’s)
Monoamine Oxidase Inhibitors (MAOI’s)
Lithium
Tricyclic Antidepressants (TCA’s)
Amitryptiline
Clomipramine
Doxepin
Imipramine
Serotonin Reuptake Inhibitors (SRI’s)
Fluoxetine
Fluvoxamine
Sertraline
Monoamine Oxidase Inhibitors (MAOI’s)
Selegiline
Behaviour Modifying Drugs
Sedatives: Neuroleptics, BZD
Beta-adrenoceptor antagonists: Propranolol
Antiepileptics:Carbamezipine, Phenobarbital
Opioid antagonists: Naloxone, Naltrexone
CNS stimulants: Dexamphetamine
Antihistamines: Chlorphenamine, Diphenhydramine
Hormones: Megastrol, Cabergoline, Dalmadinon
Cerebral VasoD: Nicergoline, Propenfophylline
Artificial Pheromones: Feliway, Felifriend, DAP
Feed supplements: Alpha casozepine, Tryptophan
Depolarizing NM Blocking Agents:
Succinylcholine/ Succinylcholine Chloride/ Suxamethonium
Non-depolarizing/ Competitive NM Blocking Agents class acc to structure
Benzylisoquinolin group
Aminosteroid group
Others (Gallamine)
Non-depolarizing/ Competitive NM Blocking Agents class acc to duration of action
Ultra-short: Gentacurium
Short: Mivacurium, Chandonium
Intermediate: Atracurium, Cistracurium, Rocuronium, Vecuronium
Long….
Benzyl Isoqiunolin group NM blocking agents
d- Tobobcurarine
Atracurium
Cisatracurium
Mivacurium
Aminosteroid group NM Blocking agents
Pancuronium
Vecuronium
Rocuronium
Non-depolarizing/ Competitive NM Blocking Agents to discuss in the exam
d- Tobocurarine Gallamine Atracurium Cisatracurium Vecuronium Rocuronium Mivacurium
Local Anaesthetics: Esters
Procaine
Tetracaine
Benzocaine
Cocaine
Local Anaesthetics: Amides
Prilocaine
Lignocaine
Mepivacaine/ Ropivacaine
Bupivacaine
Cardiac Rhythm Drugs
Antiarrhythmic drugs
Cardiac Contractility
Cardiac Glycosides
Beta-adrenergic receptor Agonists
PDE Inhibitors
Calcium-sensitizing Agents
Volume Regulators (caridac)
Inhibs of RAS
B-type Natriuretic Peptide
ADH antagonists
Agents that decrease Na reabs
Agents that modify vasc tone (cardiac)
Vasoldilators
Inhibs of RAS
ACE inhibs
Angiotensin Receptor Antagonists
ACE Inhibitors
Captopril Enalopril Lisinopril Benazepril Ramipril
Angiotensin Receptor Antagonists
Valsartan
Losartan
Tilmisartan
Vasodilators: Organic Nitrates
Nitroglycerine (NO)
Nitroprusside Na
Vasodilators: Ca Channel Blockers
Dihydropyridines
Non-dihydropyridines
Dihydropyridines
Amlodipine
Nifedipine
Non-dihydropyridines
Verpamil
Diltiazem
I A Class Antiarrhythmic Drugs
Quinidine
Procainamide
I B Class Antiarrhythmic Drugs
Lidocaine
Mexiletine
II Class Antiarrhythmic Drugs
Beta Blockers!!
First gen Beta blocker
Propranolol
2nd gen beta blocker
Metoprolol
Atenolol
Esmolol
3rd gen beta blocker
Carvedilol
III Class Antiarrhythmic Drugs
Sotalol
Amiodarone
IV Class Atiarrhythmic Drugs
Dihydropyridine: Amlodipine, Nifedipine
Non-Dihdropyridine: Verapamil, Diltiazem
Emetics
Apomorfin
Xylazine
Peripheral: Syrup of Ipecacuanha, 3-4% H2O2
Antiemetics: Local
Local anaesthetics- Lidocaine, Vit B6
Antiemetics: Systemic
Phenothiazines Dopamine antagonists Antihistamines Serotonin antagonists NK-1 receptor antagonists Parasympathomimetics
Antiemetics: Phenothiazines
Tiethylperazine
Acepromazine
Chlorpromazine
Promethazine
Antiemetics: Dopamine antagonists
Metoclopramide
Domperidone
Antiemetics: Serotonin Antagonists
Ondansetron
Dolasetron
Antiemetics: Antihistamines
Dimenhydrinate
Diphenhydramine
Antiemetics: Neurokinin-1-Antagonists
Maropitant Citrate
Prokinetics/ Propulsive/ Modulators of gastric motility
Metoclopramide, Domperidone Cisapride Ranitidine, Nizatidine Parasympathomimetics: Neostigmin, Piridostigmin, Bethanecol Erythromycin
Laxatives
Stimulant
Osmotic
Colloidal
Coating agents
Stimulant Laxatives
Phenophtalein Bisacodyl Emodin Aloe Docusate Atrakinone Derivs Castor Oil
Osmotic Laxatives
Na2SO4
MgSO4
Na- Citrate
Lactulose
Colloidal Laxatives
Psyllium, cornmeal, pumpkin
Coating agents
Liquid parrafin
Antidiarrheals
Adsorbents
Adstringents
Motility Modifiers
Treatment of chronic colitis
Antidiarrheals : Adsorbents
Activated charcoal
Kaolin
Montomorillonit
Antidiarrheals: Adstringents
Bismuth Salts (subsalicylate, subgallate, subnitrate, carbonate) Tannic acid
Antidiarrheals: Motility Modifiers
Parasympatholytics (atropine)
Morphine Derivs: Diphenoxylate, Loperamide
Treatment of Chronic Colitis
Sulfasalazine: Sulfapyridin and Amino-salicylic acid
Mesalazine
Olsalazine
Appetite Stimulants
B-Vits Anabolic steroids: Nandrolone, Stanozolone BZD: Diazepam, oxazepam Cyproheptidine Propofol
Antiulcer Drugs
Acid Neutralizers (Antacids)
Acid Secretion Inhibitors: H2 antagonists and PPI’s
Drugs increasing mucosal resistance: PGE analogues, coating agents
Antiulcer: Acid Neutralizers/ Antacids
Systemic: NaHCO3
Non-systemic: Mg(OH)2 and Al(OH)3 combo, Al-Mg carbonate
Antiulcer: H2 antagonists
Cimetidine
Ranitidine
Famotidine
Antiulcer: Proton Pump Inhibitirs (PPI’s)
Omeprazole
Antiulcer: Drugs increasing mucosal resistance: PGE analogues
Misoprostole
Antiulcer: Drugs increasing mucosal resistance: Coating agents
Sucralfate: Sucrose Octasulfate and Al(OH)3
Hepatoprotectives
Cholagogues: Cholekinetics and Cholerectics
Hepatoprotectants
Lipotopic Agents
Hepatoprotectives: Cholagogues: Cholekinetics
UDCA: ursodeoxycholic acid
Menbuton
Clanobutin
Hepatoprotectants
Silymarin D-Penicillamin Glucose, fructose NAC: N-acetyl-Cysteine Vit E Vit C Selenium
Hepatoprotectives: Lipotropic Agents
Choline
SAMe (S-Adenosyl Methionine)
Methionine
Diuretics
Cardiac Diuretics
Osmotic diuretics
Natriuretics
Cardiac Diuretics
Digoxin
Xanthine derivs: Caffeine, Theophylline, Theobromine
ACE inhibs
Osmotic Diuretics
Mannitol
Glycerine
Natriuretics
PCT: Carboanhydrase Inhibs
LOOP: Furosemide
DCT: Thiazides
CT: Potassium sparing diuretics
Natriuretics: Carboanhydrase inhibs
Acetazolamide
Dorsalamide
Brinzolamide
Natriuretics : Loop diuretics
Furosemide
Turosemide
Natriuretics : Thiazides
Hydrochlorothiazide
Chlorothiazide
Natriuretics: Potassium Sparing diuretics
Spironolactone
Combined treatment of CHF in dogs
Pimobendan and Furosemide and Spironolactone or
ACE Inhibs and Furosemide and Spironolactone
Combined treatment of CHF in cats
Furosemide and Spironolactone
Treating Hypertension
Amlodipine
AT-II-Antag
ACE inhibitor
Gandotropin releasing hormones (GnRH)
Buserelin
Gonadorelin
Fertilin
Dezlorelin
Hormones of the Anterior pituitary/ Adenohypophysis
GH TSH ACTH PRL FSH and LH
Hormones of the posterior pituitary/ Neurohypophysis
Oxytocin
Vasopressin/ ADH
Growth hormones
Pure hST (human)
Bovine bST
Porcine pST
But all are banned in the EU
Corticotropin, ACTH
Tetracosactrin
The ergolides/ PRL antagonists
Bromocriptidine
Cabergoline
What are the analogues of FSH and LH? i.e the non-pituitary gonadotropins
hCG= human corionic gonadrotropin (LH activity)
PMSG/eCG (FSH activity)
Insulin formualtions
Regular crystalline zinc insulin
Isophane insulin
Lente insulin
Protamine Zinc Insulin (PZI)
Drugs influencing glucose metab i.e oral antidiabetics
Acarbose
Sulphonylurea substances
Biguanides
The sulphonylurea substances
Tolbutamide Chlorpropramide Metahexamide Glipizide/ Glibenclamide Glinides e.g Nateglinide Glitazones e.g pioglitazone
Biguanides
Fenformine
Buformine
Methformine
Short acting GC drugs
Cortisol
Cortisone
Middle acting GC drugs
Prednisolone
Prednisone
Methylprednisolone
Triamcinolone
Long acting GC drugs
Dexamethasone
Betamethasone
Flumethasone
Treatment of Hypoadrenocorticism/ Addison’s
Aldosterone Deoxycorticosterone Pivalat (DOCP) Fludrocortisone Acetate
Treatment of Hyperadrenocorticism/ Cushing’s
Pituitary dependent: Bromocriptidine, Cyproheptidine HCl
Pituitary and or adrenal dependent: Ketoconazole, Mitotane, Trilostane
Preparations for Hypothyroidism
Crude thyroid products
Iodine containing products: Iodised salt, Lugol’s soln
Synth preps: Levothyroxine, Levothyroxine Na, L-triiodothyronine, Liothyronine
Preparations for Hyperthyroidism
Thiouracil
Methimazol/ Tiamazol
Propylthiouracil
Iodine
Prostaglandin systemic analogues
Cloprostenol
Dinoprost
Luprostiol
Etiproston
Anticoccidials
Ionophores Triazines Sulphonamides Pyridine deriv: Clopidol Pyrimidine deriv: Amprolium Quinazolin deriv: Halofuginon Carbanilide deriv: Nicarbazin Guanidine deriv: Robenidine Quinoline deriv: Decoquinate Purine deriv: Aprinocid
Ionophore antibiotics:
Monensin Narasin Salinomycin Lasalocid Maduramycin Semduramycin
Sulphonamide anticoccidials
Sulphaquinoxaline
Sulphachlorpyrazine
Triazines anticoccidials
Toltrazuril
Diclazuril
Drugs for extraintestinal coccidia:
Toxoplasmosis and canine neosporosis
Clindamycin
Sulfadiazine and Pyrimethamin
Drugs for extraintestinal coccidia:
Only toxoplasmosis
Doxycycline
Decoquinate
Classes of benzimidazoles
Thiazolil benzimidazoles
Benzimidazole carbamates
Probenzimidazoles
Thiazolil benzimidazoles
Thiabendazole
Cambendazole
Benzimidazole Carbamates
Albendazole Flubendazole Fenbendazole Mebendazole Oxfendazole Oxibendazole Ricobendazole Luxabendazole Triclabendazole
Probenzimidazoles= Prodrugs
Febantel- fenbendazole- oxfendazole
Netobimin- albendazole- ricobendazole
Thiophanate- lobendazole
Imidazothiazoles
Tetramisole
Levamisole
Tetrahydopyrimidines
Pyrantel
Morantel
Oxantel
Salicylanilides
Closantel Oxyclozanide Rafoxanide Brotianide Clioxanide Niclosamide
Substituted Phenols
Nitroxinil Bithionol Disophenol Dichlorophene Diamphenethide Nitroscanate
Isoquinolin and Benzazepin Derivs
Praziquantel
Epsiprantel
Macrocyclic Lactones
Avermectins
Milbemycins
Avermectins
Abamectin Ivermectin Doramectin Eprinomectin Selamectin
Milbemycins
Milbemycin oxime
Moxidectin
Chemical classes of ectoparasiticides
Organophosphates Carbamates Pyrethroids Formamidines Macrocyclic lactones Phenylpyrazoles Indoxacarb Neonicotinoids Isoxazolines IGR's
Organophosphates
Diazinon
Coumaphos
Phoxim
Fenthion
Carbamates
Propoxur
Pyrethroids
Tetramethrin
Permethrin
Deltamethrin
Flumethrin
Formamidines
Amitraz
Neonicotinoids
Imidacloprid
Nitenpyramin
Dinotefuran
Phenylpyrazoles
Fipronil
Pyriprol
Juvenile hormone analogues
Pyriproxyfen
Methoprene
Chitin inhibitors
Lufenuron
Novaluron
Progestagens/ Gestagens (synth)
Fluorogestone acetate Norgestomet Proligestone Medroxyprogesterone acetate Altrenogest Megestrol acetate
Progesterone antagonists
Aglepriston
Bromocriptidine and Cabergoline
Oestrogens (synth)
Estradiol benzoate
Estradiol cypionate
Estradiol valerate
Estradiol incurin
Androgens (synth)
Testosterone undecanoate
Testosterone phenylpropionate
Methyltestosterone and etinyl-estradiol
Anabolic steroid
Stanazolole
Metandienone
Nandrolone
Anti-Androgens
Cyproterone
Delmadinon
Uterine Stimulants
Oxytocin
Ergot alkaloids
Prostaglandins
Oxytocin deriv
Carbetocin
Ergot alkaloids
Ergotoxin
Ergotamine
Erogometrine (maleate salt and methyl ergometrine)
Prostaglandins
Etiproston
Luprostiol
Dinoprost
Uterine relaxing agents
Antispasmodics
Beta adrenoceptor agonists
Antispasmodics (uterine)
Danaverin
Vetrabutin/ Dimophebumine
Proquamezine, Aminopromazin
Beta adrenoceptor agonists (uterine)
Clenbutarol
Terbutaline
Isoxsuprine lactate
Isoxazolines
Fluralaner
Afoxolaner
Sarolaner
Lotilaner
Antifungal drugs
Poliene AB’s
Azoles (imidazoles and triazoles)
Allylamines
Inhibitor of fungal mitosis (griseofulvin)
Inhibitor of fungal nucleic acid (flucytosine)
Lufenuron
Echinocandins
Poliene AB’s
Natamycin
Nystatin
Amphotericin B
Azoles
Imidazoles: Thiabendazole Clotrimazole Enilconazole Miconazole Bifoconazole Ketoconazole
Triazoles: Posaconazole Itraconazole Fluconazole Voriconazole
Allylamines
Terbinafin
Naftidine
Echinocandins
Caspofungin
Micafungin
Anidulafungin
Drugs acting on the respiratory system
Bronchodilators
Resp anti-inflamm drugs
Antitussives
Mucolytics, expectorants
The groups of bronchodilators
Sympathomimetics
Parasympatholytics
Methylxanthine derivatives
Non-specific sympathomimetics
Adrenaline
Ephedrin
Isoproterenol
Specific Sympathomimetics (acting on beta2)
Short-acting:
Salbutamol
Long-acting:
Terbutaline
Clenbutarole
Salmeterole
Parasympatholytics (resp)
Ipratropium
Atropine
Glycopyrrolate
Methylxanthine derivatives
Caffeine
Theophylline
Theobromine
The respiratory anti-inflammatories
Inhalational Glucocorticoids
Chromones
Leukotriene antagonists
Inhalational glucocorticoids
Inhalosol dosage form
Beclomethasone
Fluticasone
Chromones
Na-chromoglycate
Nedocromil
Leukotriene synthesis inhibitors
Zileuton
Fenleuton
Leukotriene antagonists
Zafirlukast
Montelukast
Central antitussives
Codeine (vs morphine) Dihydrocodeine, hydrocodon Butorphanol Tramadol Dextrometorphen
Mucolytics
N-acetylcysteine
Carbocysteine
Expectorants
Bromhexin
Ambroxol
Dembrexine
Guaifenesin
Anaemia: Erythropoietin as a drug
Epoetin alpha (rhEPO-alpha) Darbepoetin-alpha
Iron deficiency anaemia: oral
Iron fumarate
iron glutamate
Fe2+
Iron deficiency anaemia: IM
Iron dextran Fe3+ 100mg elemental iron/kg
Classes of 1st generation antihistamines
Ethylenediamines
Ethanolamines
Phenothiazines
Piperidines
AH: Ethylenediamines
Chloropyramine
Chlorpheniramine
AH: Ethanolamines
Diphenhydramine
Dimenhydrinate
AH: Phenothiazine
Promethazine
AH: Piperidine
Cyproheptadine
2nd generation antihistamines
Loratidine
Cetirizine
Levocetirizine
Leukotriene synth inhibitors
Zileuton
Fenleuton
Adenosine
Leukotriene receptor antagonists
Montelukast
Zafirlulast
Human JAK inhibitors
Ruxolitinib
Tofacitinib
Vet JAK inhibitors
Oclacitinib-apoquel
Monoclonal antibodies
Lokivetmab-cytopoint
NSAID’s classification
Salicylates
Acetic acid derivatives
Arilpropionic acids
Acidic substances: Heteroaryl acetic acids, butyl pyrazolidines, anthranilic acids
Non-acid substances: Anilin derivs, pyrazoles
NSAID’s acetic acid derivs
Diclofenac
Eltenac
NSAID’s arilpropionic acid deriv’s
Ketoprofen Vedaprofen Carprofen Ibuprofen Naproxen
NSAID’s acidic substances
Heteroaryl acetic acids: Diclofenac, Indomethacin, Etoldolac
Butyl pyrazolidines: Phenylbutazone
Anthranilic acids: Flunixin meglumine, Tolfenamic acid, Meloxicam
NSAID’s non-acidic substances
Anilin derivatives: paracetemol
Pyrazolones: Metrimidazole Na
NSAID’s: Selective COX= COXIBs
Deracoxib Firocoxib Robendacoxib Cimicoxib Mevacoxib
Immunosuppression: classification of drugs
Inhibitors of gene expression
Cytotoxic agents: antimetabolites and alkylating agents
Specific lymphocyte-signalling inhibitors
Cytokine inhibition: TNFalpha inhibs and IL-1 inhibs
Inhibitors of gene expression
Glucocorticoids
Cytotoxic agents: Antimetabolites
Purin analogues: Azathioprene,
Mycophenolate mofetil
Pyrimidine analogue: Leflunomide
FA antag: Methotrexate
Cytotoxic agents: Alkylating agents
Cyclophosphamide
Specific lymphocyte-signalling inhibs (calcineurin inhibs)
Cyclosporin
Tacrolimus, Pimecrolimus
Cytokine inhibs: TNFalpha inhibs
Adalimumab
Infiximab
Etanercept
Cytokine inhibs: IL-1 inhibs
Anakira
Antiviral drugs: Pyrimidine analogues
Idoxuridin
Trifluridin
Antiviral drugs
Acyclovir Gancyclovir Famciclovir Vidarabin Zidovudin Oseltamavir
Neuramidinase and ion channel inhibitors against influenza virus
Amantadine
Rimantidine
Antineoplastic agents
Antimetabolites Agents that directly modify DNA structure Topoisomerase inhibitors Microtubule inhibitors GC's-- lymphoma and mastocytoma Other
Antineoplastic: antimetabolites
Methotrexate
5-FU
Cytarabin
Antineoplastic: Agents that directly modify DNA structure
Alkylating:
Cyclophosphamide
Chlorambucil
Lomustine
Platinum compounds:
Cisplatin
Carboplatin
Antineoplastic: Topoisomerase inhibs
Anthracyclines- Topoisomerase II:
Doxorubicin
GZ
Mitoxantrone
Antineoplastic: Microtubule inhibs
Inhibit microtubule polymerization: Vinblastine Vinchristine Inhibit microtubule depolymerization: Pacltaxel
Classes of drugs with analgesic activity
Narcotic analgesics: opioids
Non-narcotic: antipyretics, NSAID’s
Antoconvulsive/ Antiepileptics: Gabapentin, Pregabalin, Iamotrigin, Carbamazepine
Anti-arrythemic: Mexileting, Lidocaine
NMDA receptor antagonists: Ketamine, Tiletamine, Dextrometorphan
Alpha-2 agonists: Xylazine, Medetomidine
Local anaesthetics
General anaesthetics
Aminoquinolines
Chloroquine
Primaquine
Hydroxy (hakogenated) FQ’s
Chlorquinaldole
Isoquinolone derivatives (FQ’s)
Papaverine
Praziquantel
1st gen 4 Quinolones
Oxolinic acid
Nalidixic acid
Pipemedic acid
1st gen Fluoroquinolones 2
Flumequin
Norfloxacin
2nd gen Fluoroquinolones 2
Enrofloxacin Marbofloxacin Ibafloxacin Danofloxacin Orbifloxacin Difloxacin Ciprofloxacin
3rd and 4th gen fluoroquinolones
Moxifloxacin
Pradofloxacin