Pharm Exam 1 Flashcards

1
Q

epinephrine

A

Catecholamine (agonist): alpha1, alpha2, beta1, beta2, beta3

Positive inotropic; positive chronotropic; increased automaticity; increased conduction rate of AV

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2
Q

norepinephrine

A

Catecholamine (agonist): alpha1, alpha2, beta1, weak beta2

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3
Q

isoproterenol

A

Catecholamine (agonist): beta1, beta2, beta3

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4
Q

dopamine

A

Catecholamine (agonist): alpha1, beta1, dopamine1

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5
Q

dobutamine

A

catecholamine (agonist): beta1

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6
Q

midodrine

A

non-catecholamine alpha1 (agonist)

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7
Q

phenylephrine

A

non-catecholamine alpha1 (agonist)

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8
Q

albuterol

A

non-catecholamine beta2 (agonist) short acting

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9
Q

levalbuterol inhaled

A

non-catecholamine beta2 (agonist) short acting

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10
Q

salmeterol inhaled

A

non-catecholamine beta2 (agonist) long acting

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11
Q

Brovana

A

non-catecholamine beta2 (agonist) long acting

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12
Q

formoterol inhaled

A

non-catecholamine beta2 (agonist) long acting

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13
Q

terbutaline

A

non-catecholamine beta2 (agonist) oral/inj

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14
Q

metaproterenol

A

non-catecholamine beta2 (agonist) oral

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15
Q

tyramine

A

non-catecholamine (agonist) indirect acting

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16
Q

amphetamines

A

non-catecholamine (agonist) indirect acting

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17
Q

methylphenidate

A

non-catecholamine (agonist) indirect acting

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18
Q

methylphenidate transdermal

A

non-catecholamine beta2 (agonist) indirect acting

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19
Q

ephedrine

A

non-catecholamine beta2 (agonist) mixed acting mostly alpha1 and beta1

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20
Q

pseudoephedrine

A

non-catecholamine beta2 (agonist) mixed acting

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21
Q

naphazoline ophthalmic

A

non-catecholamine alpha agonist topical vasoconstrictor

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22
Q

tetrahydrozoline ophthalmic

A

non-catecholamine alpha1 agonist topical vasoconstrictor

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23
Q

oxymetazoline nasal

A

non-catecholamine alpha agonist topical vasoconstrictor

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24
Q

oxymetazoline topical

A

non-catecholamine alpha agonist topical vasoconstrictor

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25
cocaine
norepinephrine reuptake inhibitor
26
clonidine
non-catecholamine alpha 2 agonist central-acting
27
clonidine transdermal
non-catecholamine alpha 2 agonist central-acting
28
-sin suffix
alpha antagonist
29
-olol suffix
beta antagonist
30
phenoxybenzamine
non-selective alpha blocker (alpha1 and alpha2)
31
phentolamine
non-selective alpha blocker (alpha1 and alpha2)
32
prazosin
selective alpha1 blocker
33
terazosin
selective alpha1 blocker
34
doxazosin
selective alpha1 blocker
35
alfuzosin
selective alpha1A blocker
36
tamsulosin
selective alpha1A blocker
37
yohimbine
selective alpha2 blocker
38
propanolol HCL
non-selective beta blocker (beta1 and beta2)
39
nadolol
non-selective beta blocker (beta1 and beta2)
40
penbutalol
non-selective beta blocker (beta1 and beta2)
41
sotalol
non-selective beta blocker (beta1 and beta2)
42
sotalol AF
non-selective beta blocker (beta1 and beta2)
43
timolol
non-selective beta blocker (beta1 and beta2)
44
timolol ophthalmic
non-selective beta blocker (beta1 and beta2)
45
acebutolol
selective (cardio) beta1 blocker
46
atenolol
selective (cardio) beta1 blocker
47
bisoprolol
selective (cardio) beta1 blocker
48
esmolol
selective (cardio) beta1 blocker
49
metoprolol tartrate
selective (cardio) beta1 blocker
50
metoprolol succinate
selective (cardio) beta1 blocker
51
labetalol
combined alpha and beta blocker
52
carvedilol
combined alpha and beta blocker
53
acetylcholine
Cholinocepter agonist ester
54
bethanechol
Cholinocepter agonist ester
55
cevimeline
Cholinocepter agonist ester
56
methacholine inhaled
Cholinocepter agonist ester
57
pilocarpine
Cholinocepter agonist alkaloid
58
muscarine
Cholinocepter agonist alkaloid
59
physostigimine
reversible anticholinesterase (carbamates)
60
neostigimine
reversible anticholinesterase (carbamates) (for MG)
61
pyridostigmine
reversible anticholinesterase (carbamates) (for MG)
62
edrophonium
reversible anticholinesterase (carbamates) (for MG)
63
donepezel
reversible anticholinesterase (carbamates) (for Alzheimer's)
64
galantamine
reversible anticholinesterase (carbamates) (for Alzheimer's)
65
rivastigmine
reversible anticholinesterase (carbamates) (for Alzheimer's/Parkinson's)
66
malathion topical
irreversible anticholinesterases (organophosphates)
67
echothiophate ophthalmic
irreversible anticholinesterases (organophosphates)
68
soman
irreversible anticholinesterases (organophosphates)
69
nerve gases
irreversible anticholinesterases (organophosphates)
70
pralidoxime (2-PAM)
cholinesterase reactivator)
71
atropine
muscarinic cholinoceptor antagonist (alkaloid) M1, M2, M3, M4, M5 antagonist
72
scopolamine transdermal
muscarinic cholinoceptor antagonist (alkaloid)
73
hyoscyamine
muscarinic cholinoceptor antagonist (alkaloid)
74
dicyclomine
muscarinic cholinoceptor antagonist (alkaloid)
75
benztropine
muscarinic cholinoceptor antagonist (alkaloid)
76
ipratropium inhaled; nasal
muscarinic cholinoceptor antagonist (synthetic/semisynthetic quaternary)
77
tiotropium inhaled
muscarinic cholinoceptor antagonist (synthetic/semisynthetic quaternary)
78
glycopyrrolate inhaled/ glycopyrrolate
muscarinic cholinoceptor antagonist (synthetic/semisynthetic quaternary)
79
oxybutynin
muscarinic cholinoceptor antagonist (synthetic/semisynthetic non-quaternary)
80
tolterodine
muscarinic cholinoceptor antagonist (synthetic/semisynthetic non-quaternary)
81
tropicamide ophthalmic
muscarinic cholinoceptor antagonist (synthetic/semisynthetic ocular)
82
Succinylcholine
Neruomuscular-blocking depolarizing
83
d-Tubocurarine
Neuromuscular-blocking non-depolarizing
84
pancuronium
Neuromuscular-blocking non-depolarizing
85
vecuronium
Neuromuscular-blocking non-depolarizing
86
botulinum toxin
Neuromuscular-blocking (blocks release of acetylcholine)
87
dantrolene
Other; used to treat malignant hyperthermia by decreasing intracellular calcium in skeletal muscles causing muscle relaxation
88
fluoxetine (Prozac)
SSRI; also used as an anxiolytic
89
fluoxetine (Prozac Weekly)
SSRI; also used as an anxiolytic
90
fluoxetine (Sarafem)
SSRI; also used as an anxiolytic
91
sertraline
SSRI; also used as an anxiolytic
92
paroxetine
SSRI; also used as an anxiolytic
93
citalopram
SSRI; also used as an anxiolytic
94
escitalopram
SSRI
95
fluvoxamine
SSRI; also used as an anxiolytic
96
olanzapine/fluoxetine
Combo antipsychotic+SSRI
97
duloxetine
SNRI
98
Fetzima
SNRI
99
milnacipran
SNRI
100
venlafaxine
Serotonin, Norepinephrine, Dopamine reuptake inhibitor (also considered an SNRI); also used as an anxiolytic
101
desvenlafaxine
Serotonin, Norepinephrine, Dopamine reuptake inhibitor (also considered an SNRI)
102
trazodone
Serotonin modulator; 5HT2A/C antagonist and alpha 1 adrenergic antagonist; inhibits serotonin re-uptake
103
nefazodone
Serotonin modulator; inhibits NE and serotonin reuptake; 5HT2 antagonist
104
Viibryd
Serotonin modulator; selective inhibitor of serotonin reuptake and partial 5-HT1A agonist
105
Trintellix
Serotonin modulator; selective inhibitor of serotonin reuptake 5-HT3 antagonist and 5-HT1A agonist
106
bupropion HCL
weakly inhibits NE and dopamine reuptake
107
amitryptyline
TCA/TeCA
108
nortriptyline
TCA/TeCA
109
protriptyline
TCA/TeCA
110
doxepin
TCA/TeCA; also used as an anxiolytic
111
desipramine
TCA/TeCA
112
imipramine
TCA/TeCA; also used as an anxiolytic
113
mirtazapine
TCA/TeCA
114
phenelzine
MAOI
115
tranylcypromine
MAOI
116
Marplan
MAOI
117
Emsam
MAOI
118
lithium
drug for bipolar disorder: mood stabilizer
119
aripiprazole
Atypical Antipsychotic drug for bipolar disorder
120
olanzapine
Atypical Antipsychotic (for bipolar disorder)
121
quetiapine
Atypical Antipsychotic (for bipolar disorder)
122
asenapine
Antipsychotic (for bipolar disorder)
123
loxapine
Typical Antipsychotic (for bipolar disorder)
124
loxapine inhaled
Typical Antipsychotic (for bipolar disorder)
125
Vraylar
Antipsychotic (for bipolar disorder)
126
Latuda
Atypical Antipsychotic (for bipolar disorder)
127
risperidone
Atypical Antipsychotic (for bipolar disorder)
128
ziprasidone
Atypical Antipsychotic (for bipolar disorder)
129
carbamzepine
anti-seizures (for bipolar disorder)
130
oxcarbazepine
anti-seizures (for bipolar disorder)
131
lamotrigine
anti-seizures (for bipolar disorder)
132
valproic acid
anti-seizures (for bipolar disorder)
133
divalproex sodium
anti-seizures (for bipolar disorder)
134
valbenazine
Other neruologic inhibits VMAT2
135
haloperidol
Typical anti-psychotic 1st generation
136
chlorpromazine
Typical anti-psychotic 1st generation
137
fluphenazine
Typical anti-psychotic 1st generation
138
thiothixene
Typical anti-psychotic 1st generation
139
trifluoperazine
Typical anti-psychotic 1st generation
140
prochlorperazine maleate
Typical anti-psychotic 1st generation (Selective D2 Antagonist); used as as an anxiolytic
141
thioridazine
Typical anti-psychotic 1st generation
142
perphenazine
Typical anti-psychotic 1st generation
143
pimozide
Typical anti-psychotic 1st generation
144
loxapine
Typical anti-psychotic 1st generation
145
loxapine inhaled
Typical anti-psychotic 1st generation
146
olanzapine
Atypical anti-psychotic 2nd generation
147
quetiapine
Atypical anti-psychotic 2nd generation
148
ziprasidone
Atypical anti-psychotic 2nd generation
149
risperidone
Atypical anti-psychotic 2nd generation
150
clozapine
Atypical anti-psychotic 2nd generation
151
aripiprazole
Atypical anti-psychotic 2nd generation
152
Latuda
Atypical anti-psychotic 2nd generation
153
valproic acid
Anti-seizure
154
divalproex sodium
Anti-seizure
155
valproate sodium
Anti-seizure
156
oxcarbazepine
Anti-seizure
157
carbamazepine
Anti-seizure
158
levetiracetam
Anti-seizure
159
topiramate
Anti-seizure
160
zonisamide
Anti-seizure
161
lamotrigine
Anti-seizure
162
primidone
Anti-seizure
163
phenobarbital
Anti-seizure; barbituate
164
phenytoin
Anti-seizure
165
fosphenytoin
Anti-seizure
166
ethosuximide
Anti-seizure
167
gabapentin
Anti-seizure
168
pregabalin
Anti-seizure
169
clonazepam
Anti-seizure; Long acting benzodiazepine
170
diazepam
Anti-seizure; Long acting benzodiazepine
171
lorazepam
Anti-seizure; intermediate-acting benzodiazepine
172
Wellbutrin SR
weakly inhibits NE and dopamine reuptake
173
Wellbutrin XL
weakly inhibits NE and dopamine reuptake
174
Forfivo XL
weakly inhibits NE and dopamine reuptake
175
Zybann
weakly inhibits NE and dopamine reuptake
176
bupropion hydrobromide (Aplenzin)
weakly inhibits NE and dopamine reuptake
177
buspirone
5HT1A Partial Agonist
178
melatonin
melatonin receptor agonist
179
ramelteon
melatonin receptor agonist
180
suvorexant
Orexin receptor antagonist
181
hydroxyzine
sedating antihistamine 1st generation
182
diphenhydramine
sedating antihistamine 1st generation
183
alprazolam
short acting benzodiazepine
184
midazolam
short acting benzodiazepine
185
oxazepam
short acting benzodiazepine
186
triazolam
short acting benzodiazepine
187
estazolam
intermediate-acting benzodiazepine
188
lorazepam
intermediate-acting benzodiazepine
189
temazepam
intermediate-acting benzodiazepine
190
chloridazepoxide
Long acting benzodiazepine
191
chloridazepoxide/amitriptyline
combo: long acting benzodiazepine+TCA
192
clonazepam
Long-acting benzodiazepine
193
diazepam
Long-acting benzodiazepine
194
flurazepam
Long-acting benzodiazepine
195
flumazenil
Benzodiazepine antagonist
196
zolpidem
Nonbenzodiazepine benzodiazepine receptor agonist: Interacts with GABA-benzodiazepine receptor complexes
197
zaleplon
Nonbenzodiazepine benzodiazepine receptor agonist: Interacts with GABA-benzodiazepine receptor complexes
198
eszopiclone
Nonbenzodiazepine benzodiazepine receptor agonist: Interacts with GABA-benzodiazepine receptor complexes
199
secobarbital
barbituate
200
pentobarbital
barbituate
201
phenobarbital
barbituate
202
thiopental
barbituate
203
ethanol
Enchances GABA neurotransmission/ Blocks Glutamate neurotransmission
204
disulfiram
Aldehyde dehydrogenase inhibitor: treats alcohol dependace
205
cocaine
CNS stimulant; blocks NE reuptake
206
amphetamine
CNS stimulant; indirect sympathomimetic
207
methamphetamine
CNS stimulant
208
dextroamphetamine
CNS stimulant
209
dextroamphetamine/amphetamine
CNS stimulant
210
methylphenidate
CNS stimulant; indirect sympathomimetic
211
methylphenidate transdermal
CNS stimulant; indirect sympathomimetic
212
dexmethylphenidate
CNS stimulant
213
lisdexamfetamine
CNS stimulant
214
phentermine
CNS stimulant
215
atomoxetine
Selective NE reuptake inhibitor; treats ADHD and cataplexy
216
modafinil
dopamine reuptake inhibitor; used to treat narcolepsy
217
armodafanil
dopamine reuptake inhibitor; used to treat narcolepsy
218
Gabapentin
Non-opioid used for pain and antiseizure
219
Pregabalin
Non-opioid used for pain and antiseizure
220
NSAIDS
Non-opioid used for pain
221
TCAs
Non-opioid used for pain; sedative analgesic
222
morphine sulfate
High Efficacy opioid agonist
223
hydomorphone
High Efficacy opioid agonist
224
meperidine
High Efficacy opioid agonist
225
methadone
High Efficacy opioid agonist; used to treat opioid abuse in dependance programs
226
oxycodone
High Efficacy opioid agonist
227
fentanyl
High Efficacy opioid agonist
228
fentanyl transdermal
High Efficacy opioid agonist
229
heroin
High Efficacy opioid agonist
230
butorphanol
High Efficacy opioid mixed agonist/antagonist; kappa agonist
231
nalbuphine
High Efficacy opioid mixed agonist/antagonist; kappa agonist and mu antagonist
232
hydrocodone
Intermediate efficacy opioid agonist
233
Hydrocodone/acetaminophen
Intermediate efficacy opioid agonist +NSAID
234
hydrocodone/ibuprofen
Intermediate efficacy opioid agonist +NSAID
235
oxycodone
Intermediate efficacy opioid
236
oxycodone/aspirin
Intermediate efficacy opioid agonist +NSAID
237
oxycodone/acetaminophen
Intermediate efficacy opioid agonist +NSAID
238
oxycodone/ibuprofen
Intermediate efficacy opioid agonist +NSAID
239
pentazocine
Intermediate efficacy opioid mixed agonist/antagonist; kappa agonist and partial mu agonist
240
codeine
Low efficacy opioid agonist
241
buprenorphine
Low efficacy opioid mixed agonist/antagonist; used to treat opioid abuse
242
tramadol
Low efficacy opioid weak agonist/reuptake inhibitor
243
naloxone
opioid antagonist; used to treat opioid abuse
244
naltrexone
opioid antagonist; used to treat opioid abuse and alcohol abuse
245
Movantik
Peripheral opioid antagonist used to treat opioid-induced constipation
246
Relistor
Peripheral opioid antagonist used to treat opioid-induced constipation
247
Entereg
Peripheral opioid antagonist used to treat ileus and post-operatively
248
loperamide
binds gut wall opioid receptor, inhibits peristalsis
249
diphenoxylate/atropine
binds gut wall opioid receptor, inhibits peristalsis
250
difenoxin/atropine
binds gut wall opioid receptor, inhibits peristalsis
251
codeine/guaifenesin
antitussive effects; (combos of opioid combined with antihistamine, expectorant, decongestant); used to treat upper respiratory symptoms
252
chlorpheniramine/hydrocodone
antitussive effects; (combos of opioid combined with antihistamine, expectorant, decongestant); used to treat upper respiratory symptoms
253
hydrocodone/homatropine
antitussive effects; (combos of opioid combined with antihistamine, expectorant, decongestant); used to treat upper respiratory symptoms
254
Trimethaphan
nicotinic antagonist in the autonomic ganglia