ION CHANNELS AND TOXINS Flashcards
Sodium Channel
Tetrodotoxin
Batrachotoxin (BTX)
Potassium Channel
Apamin
Charybdotoxin
Calcium Channel
Omega-conotoxin
Agatoxin
Nicotinic Ach Receptor
a-Bungarotoxin
GABAA Receptor
Pictrotoxin
Glycine Receptor
Strychnine
AMPA Receptor
Philanthotoxin
Blocks sodium channel from outside
Tetrodotoxin
Slows sodium channel inactivation; shifts activation
Batrachotoxin
Source: Puffer fish
Tetrodotoxin
Source: Colombian frog
Batrachotoxin
Blocks small Ca-activated K receptors
Apamin
Blocks big Ca-activated K receptors
Charybdotoxin
Source: Honeybee
Apamin
Source: Scorpion
Charybdotoxin
Blocks N-type calcium channel
Omega conotoxin
Blocks P-type calcium channel
Agatoxin
Source: Pacific Cone Snail
Omega conotoxin
Source: Funnel Web Spider
Agatoxin
Irreversible antagonist
a-Bungarotoxin
Source: Marine snake
a-Bungarotoxin
Blocks GABAA channel
Pictrotoxin
Source: South Pacific Plant
Pictrotoxin
Competitive glycine antagonist
Strychnine
Source: Indian plant
Strychnine
Blocks AMPA channel
Philanthotoxin
Source: Wasp
Philanthotoxin