Drugs acting on Common receptors Flashcards
Alpha agonists
Alpha-1: Decongestants (e.g. phenylephrine/oxymetazoline)
Alpha-2: Glaucoma (e.g. topical brimonidine)
alpha antgonists
Benign prostatic hyperplasia (e.g. tamsulosin)
Hypertension (e.g. doxazosin)
Beta-1agonist
Inotropes (e.g. dobutamine)
Beta-1 antagonist
Non-selective & selective beta-blockers (e.g. atenolol, bisoprolol)
Beta-2 agonist
Bronchodilators (e.g. salbutamol)
beta-2 antagonist
Non-selective beta-blockers (e.g. propranolol, labetalol)
dopamine agonist
Parkinson’s disease (e.g. ropinirole)
Prolactinoma
dopamine antagonist
Schizophrenia (antipsychotics e.g. haloperidol)
Anti-emetics (e.g. metoclopramide/domperidone)
GABA agonist
Benzodiazepines
Baclofen
GABA antagonist
Flumazenil
Histamine-1 antagonist
Antihistamines (e.g. loratadine)
Histamine-2 antagonist
Antacids (e.g. ranitidine)
muscarinic agonist
Glaucoma (e.g. pilocarpine)
muscarinic antagonist
Atropine (e.g. for bradycardia)
Bronchodilator (e.g. ipratropium bromide, tiotropium)
Urge incontinence (e.g. oxybutynin)
Nicotinic agonist
Nicotine
Varenicline (used for smoking cessation)
Depolarising muscle relaxant (e.g. suxamethonium)
nicotinic antagonist
Non-depolarising muscle relaxants (e.g. atracurium)
oxytocin agonist
Inducing labour (e.g. Syntocinon)
oxytocin antagonist
Tocolysis (e.g. atosiban)
Serotonin agonist
Triptans (for acute migraine, e.g. zolmitriptan)
Serotonin antagonist
Anti-emetics (e.g. ondansetron)