DRUGS Flashcards
galantamine
AChE inhibitor
memantine
noncompetitive NMDA antagonist
l-dopa
dopamine precursor
carbidopa
peripheral decarboxylase inhibitor
selegiline
MAO-B inhibitor
bromocriptine, pergolide, pramipexole
dopamine agonists
epinephrine
used to treat hypotension, irregular heartbeat, and bronchoconstriction associated with anaphylactic shock
cromolyn sodium
histamine release inhibitor
diphenhydramine
H1 antagonist
loratadine
H1 antagonist
cimetidine
H2 antagonist
omeprazole
proton pump inhibitor
acetylsalicylate
NSAID - apirin - acetylates COX-1 and COX-2
acetaminophen
NSAID
ibuprofen
NSAID
celecoxib
cox-2 inhibitor NSAID
phenytoin
class IB antiarrhythmics +antieplieptic
lidocaine
class IB antiarrhythmics + local anesthetic + ionized
propanolol
class II antiarrhythmic + B-blocker
sotalol
class III antiarrhythmic
verapamil
class IV antiarrhythmic - calcium channel blocker
digoxin
cardiac glycoside
nitroglycerin
organic nitrate
loop diuretics
inhibit Na+/K+/2Cl- symport by blocking reabsorption of Na+/K+/2Cl- in Loop of Henle
thiazide diuretics
inhibit Na+Cl- symport in endothelial cells that line distal convoluted tubule
B-blockers
block E = decrease blood pressure
doxazosin
a1 antagonists = decrease blood pressure
clonidine
a2 agonists - increase blood pressure
minoxidil
potassium channel activator
captopril
ACE inhibitor
losartan
angiotensin II receptor antagonist
epoprostenol
vasodilator
ambrisentan
vasodilator - competitive ET-1a receptor antagonist
sildenafil
vasodilator - phosphodiesterase V inhibitor
aspirin
antiplatelet drug
clopidogrel
antiplatelet drug
statins
cholesterol-lowering drugs - HMG CoA reductase inhibitor
clofibrate
fibrate
bile acid binding resins
Cholesterol absorption inhibitor
ezetimibe
Cholesterol absorption inhibitor
niacin
treats hypercholesterolemia
omega-3 fatty acids
reduce plasma triglycerides
recombinate
hemophilia a - factor 8
benefix
hemophilia b - factor 9
heparin
intravenous anticoagulants
warfarin
oral anticoagulants
Hydroxyurea + aspirin; alpha interferon
treat Thrombocytosis
corticosteroids or Platelet rich plasma
treat Thrombocytopenia
steptokinase
fibrinolytic drugs
pilocarpine
muscarinic agonist
bethanechol
muscarinic agonist
BUTYLRYLCHOLINESTERASE
cholinesterase
physostigmine
AChE Substrate Inhibitor - glaucoma
neostigmine
AChE Substrate Inhibitor urinary retention
ecothiophate
Irreversible AChE Inhibitor - glaucoma
pralidoxime
reversible organophosphate poisoning
scopolamine
muscarinic antagonist
atropine
muscarinic antagonist
darifenacin
M3 antagonist
isoproterenol
weakly selective adrenergic agonist
phenylephrine
a1 selective agonist
clonidine
a2 agonist
dobutamine
b1 agonist
albuterol
b2 agonist
amphetamine
stimulate NE release
a-methyl tyrosine
tyrosine-hydroxylase inhibitors
prazosin
treat hypertension
metoprolol
treat hypertension/angina
succinylcholine chloride
depolarising agent
atracurium
non-depolarising agent - competitive antagonist of ACh
botox
noncompetitive ACh antagonist
edrophonium
competitive AChE inhibitor
pyridostigmine
AChE substrate inhibitor
prilocaine
LA
articaine
LA - rapid onset / short duration
benzocaine
LA - unionized