CYP450 for Schizo, Insomnia, Anxiety, ADHD Flashcards
Aripiprazole
CYP3A4 & CYP2D6 substrate
Brexipiprazole
CYP3A4 & CYP2D6 substrate
Cariprazine
CYP3A4 substrate
Asenapine
CYP1A2 & UGT substrate
- fluvoxamine
Clozapine
CYP1A2 substrate
Olanzapine
CYP1A2 substrate
Quetiapine
CYP3A4 substrate
Iloperidone
CYP2D6 substrate
Lurasidone
CYP3A4 substrate
Ziprasidone
CYP3A4 substrate (1/3) & aldehyde oxidase (2/3)
Risperidone
CYP2D6 substrate
Lumateperone
CYP3A4 substrate
Pimavanserin
CYP3A4 substrate
Valbenazine
CYP3A4 & CYP2D6 substrate
Deutetrabenazine
CYP2D6 substrate
Zolpidem
CYP3A4 substrate
Zaleplon
CYP3A4 substrate
Eszopiclone
CYP3A4 substrate
Ramelteon
CYP1A2 substrate
Tasimelteon
CYP1A2 substrate
Suvorexant
CYP3A4 substrate
Lemborexant
CYP3A4 substrate
Daridorexant
CYP3A4 substrate
Melatonin
CYP1A2 substrate
Pitolisant
CYP3A4 & CYP2D6 substrate
CYP3A4 inducer
Buspirone
CYP3A4 substrate
Guanfacine ER
CYP3A4 substrate
Atomoxetine
CYP2D6 substrate
Viloxazine
CYP2D6 & UGT substrate
CYP1A2 inhibitor
Bupropion
CYP2B6 substrate
CYP2D6 inhibitor