Antidiabetics Class Flashcards
chlorpropamide
first gen sulfonylurea
chlorpropamide
first gen sulfonylureas
tolazamide
first gen sulfonylureas
tolbutamide
first gen sulfonylureas
glyburide
2nd gen sulfonylureas
glimepiride
2nd gen sulfonylureas
glipizide
2nd gen sulfonylureas
sulfonylureas
stimulate release of insulin from pancreas, increase cell sensitivity to insulin
do sulfonylureas cause hypoglycemia
yes
metformin
buganide
Buganide
decrease hepatic production of glucose, decrease intestinal reabsorption of glucose, increase cell uptake of glucose
do buganides cause hypoglycemia
no
repaglinide
meglitinide
nateglinide
meglitinide
Meglitinide
stimulate release of insulin from pancreas
do meglitinides cause hypoglycemia
yes
rosiglintazone
thiazolidinedione
pioglintazone
thiazolidinedione
Thiazolidinediones
increase cell sensivity to insulin and decrease hepatic production of glucose, take 3-4mo
albiglutide
incretin mimetic agonist
dulaglutide
incretin mimetic agonist
exeratide
incretin mimetic agonist
liraglutide
incretin mimetic agonist
lixisenatide
incretin mimetic agonist
incretin mimetic agonist
activate GLP-1, increase insulin secretion, decrease glucagon secretion, delay gastric emptying, slow glucose aborption, increase statiety
alogliptin
incretin enhancer
linagliptin
incretin enhancer
saxagliptin
incretin enhancer
sitagliptin
incretin enhancer
incretin enchancer
prevent breakdown of incretin/GLP-1, increase insulin secretion, decrease glucagon secretion, delay gastric emptying, slow glucose absortption, increase statiety
do incretin mimetic agonists cause hypoglycemia
no
do incretin enhancers cause hypoglycemia
no
acarbose
alpha glucosidase inhibitor
miglitol
alpha glucosidase inhibitor
do alpha glucosidase inhibitors cause hypoglycemia
no
bromocriptine
dopamine receptor antagonist
does bromocriptine cause hypoglycemia
no
canagliflozin
sodium-glucose cotransporter inhibitor
dapagliflozin
sodium-glucose cotransporter inhibitor
empagliflozin
sodium-glucose cotransporter inhibitor
sodium-glucose cotransporter inhibitor MoA
inhibit SGCI in kidney, lose glucose in urine