Table 4 - Anti-Arrhythmics Flashcards
Naturally occurring nucleoside
Adenosine
Decreases myocardial excitability and conduction velocity; may depress contractility (by increasing electrical threshold)
Procainamide
For life-threatening ventricular arrhythmias
Procainamide
Electrolyte
MgSO4 (IV)
Inhibits adrenergic alpha and beta stimulation affecting Na, K, and Ca channels; prolongs AP and refractory period; decreases AV conduction and sinus node function
Amiodarone
Class 3 repolarization delay via K channels
Amiodarone
Slows conduction in cardiac tissue (by altering transport of ions across cell membranes), causes slightly prolonged refractory periods, increases threshold
Flecainide
Adrenergic B1 and B2 receptor inhibitor; reduces O2 demand, HR, contractility, BP
Propranolol
Class 1C Na channel blocker
Flecainide
Class 4 calcium channel: CCB NDHP
Verapamil, Cardizem
Dilates coronary arteries and decreases O2 demands
Verapamil, Cardizem
PSVT: Slows conduction time through AV node by interrupting reentry pathways in AV node and restoring NSR
Stress testing: Causes coronary vasodilation and increases blood flow in normal coronary arteries with little to no increase in stenotic coronary arteries
Adenosine
Inhibits Na/K pump causing increased Ca influx causing increased contractility; decreases ventricular rate (by suppressing AV node)
Digoxin
Selective B1 adrenergic receptor inhibitor
Metoprolol and Atenolol
Class 1A Na channel blocker
Procainamide
Class 2 beta blockers - nonselective
Propranolol
ONLY life-threatening recurrent VF, unstable VT, off-label for A-fib, PSVT, adjunct to ICD to suppress ventricular tachyarrhythmias in HF
Amiodarone
Digitalis-induced arrhythmias with low Mg, low Mg-induced arrhythmias (VF, VT)
OFF LABEL: Torsades de pointes, severe asthma in children
Mg SO4 (IV)
Class 1B Na channel blocker
Lidocaine
Suppressing existing ventricular arrhythmias
Lidocaine
Prevention of ventricular arrhythmias; PSVT; Paroxysmal Afib/Aflutter
Flecainide
PSVT, Pharmacologic stress testing
Adenosine
Mild to moderate HF, Afib
Digoxin
Blocks initiation and conduction of nerve impulses (by decrease permeability of Na), suppresses automaticity of conduction tissue (by increasing threshold during diastole)
Lidocaine
Class 2 Beta blockers: Cardioselective B1
Metoprolol tartrate/succinate and atenolol
Cardiac glycoside
Digoxin