Spring 25 - Farm - Local Anesthetics Flashcards
Max single dose
Procaine max single dose
7mg/kg
Pediatric 350 mg
Adults 600 mg
Procaine (infiltration/Spinal)
- Infiltration: 0.25–1%
- Spinal: 50–200 mg
Chloroprocaine max single dose (plain/Epi)
- 800 mg plain
- 1000 mg with epinephrine)
Chloroprocaine (Infiltration/Epidural)
- Infiltration: 1%
- Epidural/peripheral block: 2–3%
Tetracaine max single dose
20 mg
Highly potent and long-acting
Tetracaine (Spinal dose/onset/duration
- Dose: 0.5–1%
- Onset: 3–5 minutes
- Duration: 2–3 hours, extended to 4–6 hours with epinephrine
Cocaine max single dose
150 mg
Benzocaine max single dose
200 mg
Treatment of Methemoglobinemia induced by Benzocaine, after 200 - 300 mg administration
Treat with 1% methylene blue, 1–2 mg/kg IV over 20 minutes.
Lidocaine max single dose (plain/epi)
- Plain 200 mg
- With Epi 500 mg
Lidocaine (Infiltration/Spinal/Epidural dose)
- 0.5–1% for infiltration
- 100 mg Spinal/Epidural (controversial)
Lidocaine dose for Ventricular ectopy
100–200 mg bolus → 1–4 mg/min infusion
Prilocaine max single dose
600 mg
Mepivicaine (do not use in pregnancy) max single dose (plain/epi)
- Plain 400 mg
- With Epi 500 mg
Mepivicaine (Spinal/epidural/peripheral dose)
- Spinal 100 mg
- Epidural (1.5–2%): Onset in 10–15 minutes, duration 70–90 minutes
- Peripheral nerve block (1–1.5%): Duration 2–4 hours
Bupivacaine max single dose (pain/epi)
- Plain 175 mg
- With Epi 225 mg
Bupivicaine (Infiltration/spinal/epidural/peripheral doses)
- Infiltration: 0.25% into surgical wounds
- Spinal: Fast onset (<5 minutes), duration 1–4 hours
- Epidural: Ideal for labor and postoperative analgesia
o <0.25% reduces motor block; 0.1% gives sensory analgesia with minimal motor
effects - Peripheral block: Duration 4–12 hours, may extend to 24 hours
What three agents will cause vasoconstriction
- Ropivicaine
- Levobupivicaine
- Cocaine
Etidocaine max single dose (plain/epi)
- Plain 300 mg
- With Epi 400 mg
Ropivacaine max single dose
200 mg
What two agents will cause methemoglobinemia
- Prilocaine
- Benzocaine