side effect neurotransmitters Flashcards
constipation, blurred vision and dry mouth in TCAs
M1, M3
hypersalivation in clozapine
M4
hypertension in venlafaxine
noradrenergic receptiors
TD in Antipsychotics
dopamine supersensitivity
parkinsonism and dystonia in antipsychotics
dopamine receptor blockade in substantia nigra
hypotension in olanzapine and quetiapine
alpha adrenergic receptor blocking- post synaptic alpha 1
sexual dysfunction in SSRIs
5HT2C
Anxiety in SSRIs
5HT1A
nausea in SSRIs
5HT3
hyperprolactinaemia in antipsychotics
D2 in tuberoinfundibular system
weight gain and sedation in mirtazapine
5HT2C, H1
weight gain in antipsychotics
H1, 5HT2C
better EPSEs in atypical antipsychotics
5HT2 antagonism and increased dopamine in SN with D2 antagonism in mesolimbic system
increased anxiety with salbutamol
beta adrenergic
better anxiety with propanolol
beta adrenergic
memantine
NMDA receptor antagonist
tolerance to halluconogens
5-HT 2A receptor desenstitisation
Benzo withdrawal
decreased Brain GABA
trazadone
5HT-2 receptor binding, blocks serotonninreuptake
trazodone sedation
H1 antagonism, alpha blocking
irregular periods with antipsychotics
D2 antagonism
NMS
D2 blockade
priapism
5HT2A/5HT2C, alpha 1 antagonism
weight gain and sedation
H1 antagonism
obsessive compulsive symptoms in antipsychotic use
5HT1D
sedative action in trazodone
H1 antagonism
smooth muscle
M3 blockade
CNS
M4
Heart
M2
priapism
Alpha 1
initial energy boost with SSRIs
5HT2C antagonism
morning drowsiness on atypical antipsychotics
H1 antagonism
constipation on TCA
M1
hypnotic effect of zopiclone
GABA agonism