Pharma retake Flashcards

1
Q

Topic 51: Anticoccidial drugs

A

Ionophore antibiotics:

  • Monensin
  • Narasin
  • Maduramicin
  • Semiduramycin
  • Salinomycin
  • Laslocid

Troazine derivates:

  • Toltrazuril
  • Clazuril
  • Declazuril
  • Ponazuril

Sulphamies:

  • Sulphacholoropyrazine
  • Sulphaquinoxaline

Amprolium

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2
Q

Topic 52: Anti-protozoal drugs (Except cocciosis)

A

Histomonas & Trichomonas
Nitroimidazoles: Metronidazole, Ronidazole, Tinidazole
Nitrofurans: Nitrofurantoin, Furazolidone
(H. Megleangridis): Flubendazole or Fenbendazole

Giardia:
Metronidazole & Fenbendazole

Leishmania:
Paromomycin

Babesia:
Diamidine derivates, Imidocarb, Amicarbalide, Phenamide, Tetracyclines (Preventive)

Trypanosoma:
Homidium bromide/chloride, Isometamidium, Quinapyramine chloride/sulphate, Suramin

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3
Q

Topic 53: Anthelmintics (Benzimidazoles, Imidazothiazoles, Tetrahydropyrimidines)

A

Benzimidazoles:

  • Thiabendazole
  • Mibendazole
  • Oxibendazole
  • Triclabendazole
  • Flubendazole
  • Luxabendazole
  • Albendazole
  • Fenbendazole
  • Ricobendazole
  • Oxfendazole
  • Netobimin
  • Febantel

Imidazothiazoles:
- Levamisole

Piperazine:

  • Piperazine
  • Diethylcarbamazine

Tetrahydropyrimidines

  • Pyrantel
  • Morantel
  • Oxantel
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4
Q

Topic 54: Anthelmintics (Salicylanilides, Substituted phenols, isoquinolines, clorsulon, monepantel)

A

Salicylanilides:

  • Niclosamide
  • Oxyclozanide

Substituted phenols:

  • Diamphenetide
  • Dichlorophene
  • Disophenol

Isoquinolones

  • Praziquantel
  • Epsiprantel

Clorsulon
Monepantel

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5
Q

Topic 55: Endectocides Macrocyclic lactones

A

Avermectins and milbemycin:

  • Ivermectin
  • Doramectin
  • Selamectin
  • Eprinomectin
  • Moxidectin
  • Milbemycin oxime
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6
Q

Topic 56: Drugs for external parasites (Except endectocides)

A

Organophosphates:

  • Diazinon
  • Phoxim
  • Coumaphos
  • Antidote: Pralidoxime

Carbamates:
- Propoxur

Pyrethroids:

  • Permethrin
  • Deltamethrin
  • Tetramethrin

Formamides
- Amitraz

Neonicotinoids

  • Imidacloprid
  • Nitenpyram
  • Dinotefuran

Others:

  • Fipronil
  • Pyriprole
  • Indoxacarp

Isoxazolines:

  • Fluralaner
  • Sarolaner
  • Afloxolaner
  • Lotilaner

Insect regulators:

  • Methoprene
  • Fibronil
  • Pyriproxyfen
  • Lufenuron
  • Navaluron
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7
Q

Topic 57: Antifungal drugs

A

Allyamines:

  • Terbinafine
  • Naftifine

Imidazoles:

  • Thiabendazole
  • Clotrimazole
  • Enilconazole
  • Miconazole
  • Bifonazole
  • Ketoconazole

Triazoles

  • Posaconazole
  • Voriconazole
  • Fluconazole
  • Itraconazole

Griseofluvin

Poliene antibiotics:

  • Natamycin
  • Nystatin
  • Amphotericin B

Flucytocine

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8
Q

Topic 58: Antiviral drugs

A

Pyrimidine analogues:

  • Idoxuridine
  • Trifluridine
  • Zidovudine

Purine analogues:

  • Acyclovir
  • Ribavirin
  • Ganciclovir
  • Vidarabine
  • Cytarabine

Amantadine
Interferons

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9
Q

Topic 59: Antineoplastic agents

A

Methotrexate

Alkylating agents:

  • Cyclophosphamide
  • Chlorambucil
  • Lomustine

Platinum compound:
- Carboplatin

Topoisomerase inhibitors:

  • Doxorubicin
  • Mitoxantrone
  • Epipodophyllin toxin

Microtubule inhibitors:

  • Vinblastine
  • Vincristine

Other:

  • Toceranib
  • Masitinib
  • Asparaginase

COX:

  • Firocoxib
  • Deracoxib
  • Carprofen
  • Piroxicam
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10
Q

Topic 9 Parasympathomimetics and Parasympatholytics

A

Direct mimetics:

  • Acetylcholine
  • Carbechol
  • Pilocarpine
  • Betanechol
  • Metacholine

Indirect mimetics:

  • Physostigmine
  • Neostigmine
  • Pyridostigmine
  • Edrophonium
  • Organophosphates
  • Droperidol
  • Domperidone
  • Propanolol
  • Atenolol

Lytics:

  • Atropine
  • Homatropine
  • Tropicamide
  • Glycopyrrolate
  • Ipatropium
  • Scopolamine
  • Levodopa
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11
Q

Topic 48: Polypeptides and other antibiotics (Glycopeptides, Rifamycin)

A

Glycopeptides:

  • Vancomycin
  • Teicoplanin
  • Oritavancin
  • Dalbavancin
  • Telavancin

Rifamycin:

  • Rifamycin B
  • Rifampin
  • Rifabutin

Mupirocin

Polymyxin:

  • Polymyxin B, Polymyxin E = Colistin
  • Polymyxin M = Mattacin
  • Colistimethate

Bacitracin-Zn

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12
Q

Topic 49: Sulphonamides and Diaminopyrimidines

A

Sulphonamides:

  • Sulfaguandine
  • Sulfacetamide
  • Sulfadiamidine
  • Sulfachlorpyridazine
  • Sulfadoxine
  • Sulfadiazine
  • Sulfamethoxasole
  • Sulfaquinoxaline
  • Sulfachlorpyrazine
  • Sulfasalazine
  • Sulfadimethoxine
  • Sulfamethoxypyrazine

Diaminopyrimidine:

  • Trimethoprim
  • Diaveridine
  • Primimethamin
  • Ormethoprim
  • Aditoprim
  • Baquiloprim
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13
Q

Topic 50: Fluroquinolones

A

1st:
- Nalidixic acid

2nd:

  • Flumequine
  • Norfloxacin
  • Ciprofloxacin
  • Enrofloxacin
  • Danofloxacin
  • Difloxacin
  • Marbofloxacin

3rd:

  • Levofloxacin
  • Sparfloxacin

4th:

  • Moxifloxacin
  • Pradofloxacin
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14
Q

Topic 10: Sympathomimetics and sympatholytics

A

Non-specific:

  • Adrenaline
  • Noradrenaline
  • Dopamine

B1 agonists:

  • Dobutamine
  • Isoproterenol

B2 agonists:

  • Clenbuterole
  • Salbutamole
  • Terbutaline
  • Salmeterole

A1 agonist:

  • Phenylephrine
  • Xylometazoline
  • Oxymetazoline
  • Naphazoline
  • Tertryzoline
  • Phenylpropanollamine
  • Ephedrine

A2 agonist:

  • Xylazine
  • Detomidine
  • Medetomidine
  • Dexmedetomidine

A antagonists:

  • Phenoxybenzamine
  • Phentolamine
  • Tolazoline

A1 antagonists:

  • Prazosine
  • Doxasozine

A2 antagonists:

  • Yohimbine
  • Atipamezole

B antagonists

  • Propanolol
  • Timolol
  • Metoprolol
  • Atenolol
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15
Q

Topic 11: Tranquilizers

A

Phenothiazines:

  • Chlorpromazine
  • Propionylpromazine
  • Acepromazine
  • Thiethylperazine
  • Promethazine

Butyrophenones:

  • Azeperone
  • Droperidol
  • Fluanison
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16
Q

Topic 12: Sedato-hypnotics

A

Alpha 2:

  • Xylazine
  • Detomidine
  • Medetomidine
  • Dexmedetomidine
  • Romifidine

Benzodiazepines:

  • Diazepam
  • Zolacepam
  • Midazolam
  • Alprazolam
  • Loracepam

Barbiturates

  • Phenobarbital
  • Pentobarbital
  • Thiopental
  • Methohexital
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17
Q

Topic 45: Tetracyclines

A
Chlortetracycline
Tetracycline
Oxytetracycline
Doxycyline
Minocycline
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18
Q

Topic 46: Macrolides

A
Erythromycin
Azithromycin
Clarithromycin
Spiramycin
Tylosin
Tylvalosin
Tilmicosin
Gamithromycin
Tulathromycin
Tildipirosin
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19
Q

Topic 47: Phenicols, Lincosamides and Pleuromutilins

A

Phenicols:

  • Chloramphenicol
  • Florfenicol
  • Thiamphenicol

Lincosamides:

  • Lincomycin
  • Clindamycin

Pleuromutilins:

  • Tiamulin
  • Valnemulin
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20
Q

Topic 13: Opioids

A
Morphine
Codeine
Methadone
Fentanyl
Sufentanyl
Alfentanyl
Remifentanyl
Tremadol
Hydrocodone
Oxycodone
Butorphanol
Buprenorphine
21
Q

Topic 14: Inhalation anaethetics

A
N2O
Halothane
Isoflurane
Desflurane
Sevoflurane
Enflurane
Methoxyflurane
22
Q

Topic 15: Injectable anaesthetics

A

Barbiturates:

  • Pentobarbital
  • Thiopental
  • Thiamylal
  • Methohexital

Propofol
Propanidid

Imadazoles:

  • Etomidate
  • Metomidate

Dissociative anaesthetics:

  • Ketamine
  • Tiletamine

Benzodiazepines:

    • Diazepam
  • Zolacepam
  • Midazolam
  • Alprazolam
  • Loracepam

Phenothiazines:

  • Chlorpromazine
  • Propionylpromazine
  • Acepromazine
  • Thiethylperazine
  • Promethazine

Steroid anaesthetics:

  • Alfaxolone
  • Alfadonolone
23
Q

Topic 42: Penicillins and Beta-lactamase inhibitors

A

Narrow spectrum penicillins:

  • Procaine penicillin
  • Benzylpenicillin
  • Phenoxymethyl penicillin
  • K and Na

Beta-lactamase stable penicillin:

  • Oxacillin
  • Cloxacillin
  • Dicloxacillin
  • Flucloxacillin
  • Meticillin

Broad spectrum penicillin:

  • Ampicillin
  • Amoxicillin
  • Bacampicillin
  • Pivampicillin

Penicillin acting acainst Pseudomonas

  • Piperacillin
  • Ticaricillin

Beta-lactamase inhibitors:

  • Clavulanic acid
  • Sulbactam
  • Tazobactam
24
Q

Topic 43: Cephalosporins, monobactams and carbapenems

A

1st generation:

  • Cefazolin
  • Cefapirin
  • Cefadroxil
  • Cefalexin

2nd generation:
- Cefuroxime

3rd generation:

  • Ceftiofur
  • Cefovecin
  • Ceftriaxone
  • Cefotaxime
  • Ceftazidim
  • Cefoperazone
  • Cefixime

4th generation:
- Cefquinome

Monobactams:

  • Axtreonam
  • Tigemonan

Carbapenems:

  • Imipenem
  • Metropenem
  • (Cilastatin = Dihydropeptidase inhibitor)
25
Topic 44: Aminoglycosides
``` Streptomycin Neomycin Kanamycin Gentamycin Tobramycin Amikacin Apramycin Spectinomycin ```
26
Topic 16: Anticonvulsants
Phenobarbital Primidone Midazolam Lorazepam Diazepam Alprazolam Phenytoin Sodium/Potassium bromide Imepitoin Levetriacetam Isoflurane Sevoflurane ``` Big NO-NO: Tranquilizers Opioids Ketamine Alpha 2 agonists Methylxanthines ```
27
Topic 17: Antidepressant and behaviour modifying drugs
TCA: - Amitriptyline - Clomipramine SRI: - Fluoxetine - Fluvoxamine - Sertraline MAOIs: - Selegiline Benzodiazepines
28
Topic 18: Peripheral muscle relaxants, spasmolytics
Non-depolarising neuromuscular blocking agents: - Gentacurium - Mivacurium - Vecuronium - Atracurium - Rocuronium - Gallamine Depolarising neuromuscular blocking agents: - Succinylcholine - Suxamethonium Spasmolytics: - Papaverine - Drotaverine
29
Topic 19: Local anaesthetics
Esters: - Procaine - Chloroprocaine - Tetracaine - Cocaine - Benzocaine Amides: - Lidocaine - Prilocaine - Bupivacaine - Mepivacaine - Ropivacaine
30
Topic 20: Digital Glycosides, Phosphodiesterase inhibitors
Adrenaline Dobutamine Dopamine Nitroglycerine Digitalis glycosides Digitoxin Digoxin Pimobendan (+ Furosemide)
31
Topic 21: ACE-inhibitors, angiotensin-receptor antagonists, vasodilators
ACE inhibitors: - Captopril - Enalapril - Ramipril - Benazepril - Lisinopril Angiotensin II receptor antagonists: - Losartan - Valsartan - Telmisartan Vasodilators: - Nitroglycerine Ca- channel blockers: - Amlodipine - Nifedipine - Verapamil - Diltiazem Others: - Prazosin - Doxazosin - Hydralazine
32
Topic 39: Pharmacology of immunosuppression
Antimetabolites: - Azathiprine - Mycophenolic acid - Methotrexate - Leflunomide Alkylating agents: - Cyclophosphamide Glucocorticoids Cytokine gene expression inhibitors: - Cyclosporin - Tacrolimus - Pimecrolimus
33
Topic 38: Glucocorticoids
``` Cortisole Prednisolone Methylprednisolon Triamcinolone Betamethasone Dexamethasone Beclomethasone Fluticasone Budesonide ```
34
Topic 36: Antihistamines, Leukotriene-antagonists, Janus kinase inhibitors, monoclonal antibodies in the veterinary medicine
Etylenediamines: - Chloropyramine - Chlorophenramine Ethanoleamines: - Diphenhydramine - Dimenhydrinate Phenotiazine: - Promethazine Piperazines: - Hydroxyzine - Cyproheptadine 2nd Generation: - Cetrizine - Loratidine - Levecetrizine JAK inhibitors: - Oclacitinib - Lokivetmab Leukotriene inhibitors: - Zileuton - Fenleuton - Montelukast - Zafirlukast Monoclonal antibodies: - Lokivetmab
35
Topic 37: Non-steroid anti-inflammatory agents (NSAID's)
- Acetylsalicyclic acid - Sodium salicylate - Sulfasalazine - Mesalazine - Olsalazine - Ketoprofen - Carprofen - Vedaprofen - Flunizin meglumine - Tolfenamic acid - Phenylbutazone - Etodolac - Meloxicam - Piroxicam - Metamizole sodium - Paracetamol - Nimesulide - Firocoxib - Robenacoxib - Deracoxib - Cimicoxib - Mavacoxib
36
Topic 33: Pharmacology of sexual function 2 (Progestagens, Oestrogens, Androgens)
Progestagens: - Flurogeston - Norgestomet - Altrenogest - Medroxyprogesteron acetate - Proligeston - Megestrol acetate - Aglepriston (Antagonist) Estrogens: - Estriol - Estradiol benzoate - Estradiol valerate Anti-estrongens - Tamoxifen - Raloxifen Androgens: - Testosterone - Androstenedione - Dihydrotestosterone - Testosterone undercanoate - Testosterone phenylpropionate
37
Topic 34: Uterus muscle stimulants and relaxants
``` Stimulants: Prostaglandins - Cloprostenol - Dinoprost - Etiproston - Luprostiol Oxytocin Carbetocin Parasympathomimetics: - Carbachol Ergot alkaloids: - Ergometrine - Methylergometrine ``` ``` Uterus relaxants: Antispasmodics: - Denaverine - Papaverine - Drotaverine B2 agonists: - Terbutaline - Clenbuterol ```
38
Topic 35: Pharmacology of Anaemia (Iron, Erythropoietin and derivates)
Iron: - Apoferretin - Ferretin - Iron – fumarate - iron – gluconate - Fe-dextrane - Deferoxamine If overdose: - Deferoxamine - Hepcidin - Pyrodoxine - B6, 9 and 12 Erythropoietin: - Epoetin-alpha - Darbepoetin Immunomodulatory therapy: - Levamisole
39
Topic 22: Antiarrhytmic drugs
Na-channel blockers: - Quinidine (A) - Procainamide (A) - Lidocaine (B) - Mexiletine (B) Beta-blockers: - Propanolol - Metoprolol - Atenolol - Esmolol - Carvedilol K+-channel blockers: - Sotalol - Amiodarone Ca2+-channel blockers: - Amlodipine - Nifedipine - Verapamil - Diltiazem - Digoxin - Atropine
40
Topic 23: Pharmacology of Respiratory tract
Sympathomimetics: - Adrenaline - Ephedrine - Salbutamol - Clenbuterole - Terbutaline - Salmeterol - Formoterol Parasympatholytics: - Atropine - Glycopyrrolate - Ipratropium Xanthine derivates: - Caffeine - Theobromine - Theophylline - Aminophyllin - Propentophylline Antitussives: - Codeine - Dihydrocodeine - Butorphanol - Tramadol - Dextrometorphan Mucolytics: - Acetylcysteine - Carbocysteine Expectorants: - Bromohexine - Ambroxal - Dembrexine - Guaifenesine - Ammonium chloride - Volatile oils Respiratory anti-inflammatory: - Beclomethasone - Fluticasone - Na-chromoglcate - Nedocromil Leukotrienes antagonists: - Zileuton - Fenleuton - Zafirlukast - Montelukast
41
Topic 24: Emetics, Antiemetics, Prokinetic drugs
``` Emetics: - Apomorphine - Xylazine - H2O2 (- Carbechol - Neostigmine) ``` Antiemetics: - Lidocaine - Benzocaine - Sucralfat - Acepromazine - Chlorpromazine - Promethazine - Metoclopramide - Domperidone - Ondansetron - Dimenhydrinate - Diphenhydramine - Maropitant Prokinetic drugs: - Metoclopramide - Domperidone - Cisapride - Ranitidine - Nizatidine - Neostigmine - Pyridostigmine - Erythromycin
42
Topic 30: Adrenocortical hormones, drugs for treatment of cushing's disease and addison's disease
Adrenocortical hormones: - Mineralcorticoids (Aldosterone) - Glucocorticoids - Androgens (Estrogen, Testosterone) Cushing's disease: - Bromocriptine - Mitotane - Trilostane Addison's disease: - Deoxycortixosterone pivalate - Fludrocortisone acetate
43
Topic 31: Thyroid hormones, drugs for treatment of hypothyroidism and hyperthyroidism
Hormones: - Triiodothyronine (T3) - Thyroxine (T4) - Calcitonin Hypothryroidism: - Levothyroxine - Levothyroxine-Na Hyperthyroidism: - Methimazole - Carbimazole - Iodine
44
Topic 32: Pharmacology of sexual functions 1. (GnRH, Gonadotropins, prostaglandins)
GnRH: - Gonadorelin - Buserelin - Fertirelin - Deslorelin Gonadotropins - FSH - LH - eCG - hCG Prostaglandins: - Cloprostenol - Dinoprost - Etiproston - Luprostiol
45
Topic 25: Laxatives, antidiarrheals, appetite stimulants
Stimulant laxatives: - Phenolphtalein - Bisacodyl - Aloe - Emodin Osmotic laxatives: - Na2SO4 - MgSO4 - Lactulose Colloidal laxatives: - Corn meal - Pumpkin Emolliant laxatives: - Liquid paraffin Antidiarrheals, adsorbents: - Activated charcoal - Kaolin Antidiarrheals, adstringents: - Bismuth salts (Salicyclic acid) - Tannic acid Motility reducers: - Atropine - Butyl-scopalamine - Loperamide - Diphenpxylate Appetite stimulants: - B vitamins - Nandrolone - Stanozolole - Diazepam - Oxazepam - Cyproheptadine - Propofol
46
Topic 26: Antiulcer drugs and liver protectants
Antacids: - MgO - MgOH - AlOH H2- antagonists: - Cimetidine - Ranitidine - Famotidine Proton-pump inhibition: - Omeprazole PGE-analogues - Misoprostol Coating agents: - Sucralfate Cholagogues: - Ursodiol - Clanobutin Hepatoprotectants: - Silimarine Lipotropic drugs: - Choline - Methionine - Lecithin Others: - Glucose and Fructose - N-acetylcysteine - Vitamin E, B, K, C and Se
47
Topic 27: Diuretics
Cardiac diuretics: - Digoxin - Caffeine - Theophyllin - Theobromine ACE inhibitors: - Captopril - Enalapril - Ramipril - Benazepril - Lisinopril Osmotic diuretics: - Mannitol Carboanhydrase: - Acetazolamide - Dorzolamide Loop diuretics: - Furosemide - Torsemide Thiazides: - Hydrocholothiazide - Cholothiazide Potassium sparing diuretics: - Amiloride - Triamterene Aldosterone antagonists: - Spironolactone
48
Topic 28: Pharmacology of the hypothalamus and hypophysis hormones
Hypothalamus: - Buserelin - Fertirelin - Gonadorelin - Deslorelin Thyreotropin: - Levothyroxine Prolactin: - Bromocriptine Hormones of the pituitary gland: - eCG - hCG - Oxytocin - Carbetocin Others: - Thyroid gland: T3 & T4 - Pancreas: Insulin - Pineal gland: Melatonin Antidiuretic hormone: - Desmopressin
49
Topic 29: Insulin and other antidiabetics
Insulin: - Insulin zinc - Protamine zinc insulin - Isophane insulin Antidiabetics: - Tolbutamide - Chloropropamide - Metahexamide - Glipizide - Fenformine - Buformine - Methoformine - Troglitazone - Draglitazone - Acarbos