Mini 1 Flashcards
Local Anastatics- esters
Procaine
Cocaine
Tetracaine
Benzocaine
Local Anesthetics - amides
Prilocaine
Lidocaine
Articaine
Bupivacaine
M-cholinergic agonists
Pilocarpine
Betanechole
Cevimeline
Nicotinic agonists
Nicotine
Lobeline
MN cholinergic agoinists (directly acting)
Carbachole
MN cholinergic agoinists (indirectly)- reversible
Galantamine Edrophonium Rivastigmine Donepezil Neostigmine Pyridostigmine
MN cholinergic agoinists (indirectly)- irreversible
Echothiophate
M-cholinergic antagoinsts- Plant alkaloids
Atropine
Scopalamine
M-chilinergic antagonists -semi,syn
Homatropine Oxubutynin Tropicamide Tolerodine Ipratropium Trihexyphenidyl Solifenacin Propantheline Pirenzepine Darifenacin
Ganglion blockers
Trimethaphan
Mecalamine
Neuromuscular blocking - dep
Suxamethonium
Neuromuscular blocking - non de
Pancuronium Rocuronium Atracurium Cisatracurium Tubocurarine Vecuronium Micacurium
Alpha beta adrenergic agoinsts (D,I,M)
D- epinephrine Norepinephrine I- amphetamine Cocaine M - ephedrine
Alpha adrenergic agonists ( 1, p2 , 2)
1- phenylephrine
Midodrine
P2 - xylometazoline
Oxymetazoline
Nafzoline
2 - clinidine
Methyldopa
Beta adrenergic agoinists (non selective b1 b2, selevctive b1 , selective b2)
Non - isoprenaline
Selective b1 - dobutamine
Selective b2 - salbutamol Salmeterol Fenoterol Orciprenaline Hexoprenaline Ritodrine
Dopamine agonists
Fenoldopam
Bromocriptine
Alpha anta ( non selective, selective a1 , a2)
Non - phenoxybenzamine
Phentolamine
A1 - prazosin Terazosin Doxazosin Tamsulosin Silodosin
A2 - yohimbine
Beta antagonists ( non , b1 ,ab antagonists)
Non - propanolol
Nadolol
Timolol
Pindolol
B1 - metoprolol Atenolol Bisoprolol Esmolol Acebutolol Nebivolol
ab - labetalol
Carvedilol
Genaral anesthetic - inhalation
Non halogenated - NO
Halogenated hydrocarbons- (HEDISM) Halothane Enflurane Desflurane Isoflurane Sevoflurane Methoxyflurane
New-
Dexmedetomidine
Fosprofol
GA - intravenous
(PETMIKE) Propofol Etomidate Thiopental Midazolam Ketamine
Hypnotic - benzodiazepam
(2 zolam 5 zepam) Triamzolam Estazolam lorazepam Flurazepam Nitrazepam Temazepam Quazepam
Hypnotic - barbiturates, MISC
B- phenobarbital
Pentobarbital
MISC - zolpidem
Diphenhydramine
Ramelteon
For alcoholism
Disulfiram
Naltrexone
Acamprosate
Opioid analgesics - agonists ( strong, weak)
Strong - morphine
Meperidine
Methadone
Fentanyl
Weak - codeine
Propoxyphene
Opioid - partial Ago-anta and pure antagonists
Partial - tramadol
Tapentadol
Pentazocine
Buprenorphine
Pure - naloxone
Naltrexone
Alvimopan
Methyl naltrexone
Non opioid analgesics
NSAIDs - aspirin Ibuprofen Ketorolac Indomethacin Diclofen
Others - paracetamol
Anti epiletic - GABA potentiation
(BBGe TV) Benzodiazepines Barbiturates Gabapentin Tigabin Vigabatrin
Antiepiletic drugs : Na+ channel blockers , Ca2+ channel blockers and glutaic acid antagonists
Na- Carbamazepine
Phenytoin
Ca - ethosuximide
Valproic acid
Glutaic acid antagonists -
Lamortigine
Felbamate
Topiramate
Anti parkinsonic
Lovadopa Bromocriptine, pergolid Selegiline Entacapone, tolcapone Amntadine Trihexyfenidyl Benztropine
Skeletal muscle relaxants
Baclofen
Tizonidine
Dontrolen
Antipsychotic- typical- phenothiazines ( aliphatic, piperazine, piperidine) i
A - chlorpromazine
P.zine - trifluoperazine
Fluphenazine
Prochlorperazine
P.dine - thioridazine
Antipsychotic- typical - other
Buterophenone - haloperidol
Trifluperidol
Droperidol
Thioxanthine - chlorprotixene
Antipsychotic- atypical
Clozapine Olanzapine Cariprazine Asenapine Quetiapine Risperidone Ziprasidone Lurasidone
Anxiolytics ( B deri, agonists of ……
Benzodiazepines derivatives -
ST - triazolam
IN - oxazepam , lorazepam, alprazolam
LT - diazepam, chlordiazepoxide, medazepam, nitrazepam
Agonists of serotonine 5HT1A -
Buspirone
Antidepressants- non selective …..
Non selective serotonin and norepinephrine reuptake inhibitors-
Nortriptyline Imipramine Protriptyline Amitriptyline Maprotiline Amoxapine
Antidepressants- selective …..and selective …..
Selective serotonin and norepinephrine reuptake inhibitors-
Venlafaxine
Duloxetine
Selective serotonin reuptake inhibitors- Fluoxetine Padoxetine Sertraline Escitalopram
Antidepressants- MOA inhibitors ( irreversible, reversible, others)
Irr- tranylcypromine
Selegiline
Re - moclobemide
Others - mirtazapine
Trazodone
Vortioxetine
Agomelatin
Normothymic ( mood stabilizing , antimanic)
Lithium carbonate
Carbamezapine
Valproic acid
Psycho stimulants
derivatives of …. X 2
Derivatives of phenylalkylamine and their analogues( groups of amphetamine) -
Amphetamine
Methylphenidate
Derivatives of methylxanthine -
Caffeine
Theophylline
Nootropic ( phychometabolic)
Pyracetam
GABA ( aminalon)
Citicoline
Drugs for Alzheimer
Glutamate NMDA agonists-
Memantine
Acetylcholine esterase inhibitors-
Donepesil
Rivastigmine
Galantamine