First Exam Semester 2 Flashcards
Selective Serotonin Reuptake Inhibitors (SSRIs)
Fluoxetine (Prozac)
Paroxetine (Paxil)
Sertraline (Zoloft)
Fluvoxamine (Luvox)
Citalopram (Celexa)
Escitalopram (Lexapro)
Selective Serotonin Reuptake Inhibitors (SSRIs) and 5-HTReceptor Modulators
Vilazodone (Viibryd)
Vortioxetine (Trintellix)
Trazodone
Nefazodone
Mirtazipine
Serotonin (5-HT) and Norepinephrine (NE) Reuptake Inhibitors (SNRIs)
Venlafaxine (Effexor)
Desvenlafaxine (Pristiq)
Duloxetine (Cymbalta)
Levomilnacipran (Fetzima)
Buproprion (Wellbutrin)
(not a SNRI Dopa and NE reuptake inhibitor)
TCAs
Im/Clom/Des-ipramine
Ami/Nor-tryptyline
Other Antidepressants
Selegiline/EMSAM Patch
Ketamine
SSRI’s ADRs
ADR-s all except SD gone within a few weeks
5HT4- Diarrhea
5HT3- NV
5HT2- Solmnolence and Sexual Dysfunction
5HT1-Headache
SSRI other negative Effects.
Weight gain due to 5-HTc antagonism - Paroxetine
Triptans
Sumatriptan
Naratriptan
Razatriptam
Zolmitriptan
Almotriptan
Eletriptan
Frovatriptan
What are the GABA A subtypes?
a 1-6
b 1-3
d
e
g 1-3
q
p
p 1-3 (GABA C)
What are the GABA B subtypes?
1
2
GABA receptor subtypes and effects
GABA A
a1 - (Z drug Target) Sedative / Hypnotic, reinforcing
a2 and 3 - Anxiolytic, anticonvulsant (a2)
a5 - Leaning and memory (Psuedoalzhiemers with extended use)
b3 - Respiratory Drive, hypnotic
GABA B
Muscle relaxant
Z drugs
GABA A a1 subunit
Zolpidem
Zaleplon
Eszoplicone (Least Specific)
Benzodiazepines (BZD)
Triazolam
Clonazepam
Alprazolam
Lorazepam
Diazepam
Oxazepam
Chlordiazepoxide
The Clear And Least Desirable Option, Chlordiazepoxide
Typical Anti-Psychotics
Droperidol
Pimozide
Loxapine
Molindone
Thiothixene
Chlorpromazine
Fluphenazine
Haloperidol
Damnit People Let Me Thoroughly Cry For Help
Atypical Anti-Psychotics
Latuda
Vraylar
Quetiapine
Paliperidone
Risperidone
Olanzapine
Fanapt
Clozapine
Ziprasidone
Aripiprazole
Rexulti
Saphris
_L_eave _V_ery _Q_uickly _PROF CZARS_
Fatty Acid LAI Anti-Psychotics
Fluphenazine Decanoate
Olanzapine Pamoate
Paliperidone Palmitate
Aripiprazole Lauroxil
Haloperidol Decanoate
_F_uck _OPAH_
Other LAIs
Risperidone (Consta - 2 weeks)
Aripiprazole (Maintena - 4 weeks)
Risperidone (Perseris - 4 weeks)
ARR!
Morphine-like Agonists
Hydromorphone
Morphine
Codeine
Hydrocodone
Oxymorphone
Levorphanol
Oxycodone
HM CHOLO
Meperidine-Like agonists
Fentanyl
Meperidine
_F_uck _M_e
Methadone-Like agents
Methadone
Partial Agonists and mixed agonist - antagonist
Partial Mu agonist / Kappa antagonist
Buprenorphine
Kappa agonist / Mu antagonist
Pentazocine
Butorphanol
Nalbuphine
Delta agonist / Mu antagonist
Dezocine
_B_urp, _P_lease _B_e _N_ot _D_umb
Antagonists
Naloxone
Naltrexone (Opioid and ETOH)
Nalmefene (ETOH only)
Methylnaltrexone
Alvimopan
_N_ever, _N_ever, _N_ever, _M_eet _Anyone_
Atypical Opioids
Tramadol
Tapentadol
Trama-pentadol
First Gen Anti-Epileptics
Phenytoin
Carbamazepine
Valporic Acid
Phenny Can Vape
New-Gen Anti-Epileptics
Gabapentin
Pregabalin
Lamotrigine
Oxcarbazepine
Topiramate
G** rated **PLOT
Spasmolytic (stops spasm) Muscle Relaxants
Baclofen
Tizanidine
Dantrolene
Benzodiazepines
Botulinum Toxin
_B_en _T_ells _D_an _B_uy _B_ ig
Anti-Spasmodic (lower duration / extent of spasm) Muscle Relaxants
Benzodiazepines
Cyclobenzaprine
Carisoprodol
Metaxalone
Chlorzoxazone
Methocarbamol
Tizanidine
Orphenadrine
_B_e _C_alm, _C_arry _M_e _C_arefully, Methodically _T_o _O_ hio
General Inhaled Anesthetics
Nitrous Oxide (Gas)
Desflurane (Volatile)
Sevoflurane (Volatile)
Enflurane (Volatile)
Isoflurane (Volatile)
Halothane (Volatile)
-th/rane
General IV Anesthetics
Ketamine
Etomidate
Propofol
Thiopental
KEPT
Local Ester-Linked Anesthetics
Procaine
Benzocaine
Tetracaine
Topical cocaine
Chloroprocaine
_P_lease _B_e _T_erribly _T_erribly _C_areful
Local Amide-Linked Anesthetics
Lidocaine *
Dibucaine
Mepivacaine
Bupivacaine *
Prilocaine
Ropivacaine
Articaine
_L_ets _D_rink _M_ore _B_ooze _P_lease, _R_um _A_lways