Drugs Names Flashcards
Drugs that block H1 receptor:
Dimenhydrinate Diphenhydramine Cyclizine Loratadine Azelastine
Cyclooxygenase (COX) inhibitors
NSAIDs Aspirin
Angiotensin Receptor Antagonists (ARBs)
Losartan Valsartan Olmesartan
Beta Blocker - partial agonist
Pindolol
CystLT1 antagonist
Montelukast Zafirlukast
Neuro-sympathetic Agonists
Phenylephrine Methoxamine Norephinephrine Epinephrine Isoproterenol
Seritonin Agonists;
Buspirone Cisapride Sumatriptan
selective B1 Adrenergic Antagonists
metoprolol atenolol
Seritonin Antagonist used for Antihypertensive in Europe
Ketaserin
Nitrovasodilators
hydralazine minoxidil sodium nitroprusside (SNP)
B1-Adrenergic Antagonists
metoprolol atenolol pindolol lebetolol carvedilol
5-HT3 Antagonists
Ondansetron
5-HT4 Agonist
Cisapride
Central Agents (a2 agonists)
Clonidine Methyldopa
DHP’s
nifedipin, amlodipine
non-selective ET-1 Antagonist:
Bosentan
Second Generation Antihistaminics:
Loratadine (claratin)
Seritonin Antagonists
Clozapine Cyproheptadine Methysergide Ketaserin Ondasetron
ETa/ETb Antagonists
Bosentan
First Generation Antihistaminics:
Dimenhydrinate (gravol) Diphenhydramine (benadryl) Cyclizine (motion sickness)
5HT1A Agonist
Buspirone
Thiazide Diuretics
Hydrochlorothiazide Chlorthalidone Indapamide
5-Lipoxygenase (LOX) Inhibitor
Zileuton
Nitrates
nitroglycerin isosorbide dinitrate
a1 agonists (selective)
Phenylephrine methoxamine
5-HT1B/D Agonist
Sumatriptan
ACE - Inhibitors
captopril Enalapril Ramipril Perindopril
a1,a2,B1,B2 agonist
epinephrine
B1,B2 agonist
Isoproterenol
Phospholipase A2 (Ca2+/Calmodulin) Inhibitors
Glucocorticoids (annexins/lipocortins) Calcium Channel Antagonists
ETa1 Antagonists
Ambrisentan
selective ETa1 Antagonist:
Ambrisentan
Direct Renin Inhibitor (DRI)
Aliskiren
Endothelin (ET-1) Antagonists:
Bosentan Ambrisentan
Intranasal Antihistamines:
Azelastine
5-HT2 Antagonists
Clozapine Cyproheptadine Methysergide Ketaserin
a1,a2,B1 agonist
Norepinephrine
Beta Blockers with a-blocks
Carvedilol Lebetolol
Drugs that Block H2 receptor:
Ranitidine
Hypertensive Crisis Drug:
SNP sodium nitroprusside
Calcium channel Antagonists
Diltiazem Verapamil nifedipine Amlodipine