Drugs Flashcards
Opioids
Mu agonists:
Morphine
Hydromorphone
Fentanyl
Methadone
Partial mu agonists:
Buprenorphine
Mu antagonist/ kappa agonist:
Butorphanol
Alpha 2s
Xylazine
Dexmedatomidine
Medetomidine
Romifidine
Detomidine
NMDA receptor antagonists
Ketamine
Amantadine
Dextromethorphan
NSAIDS
Non-steroidal anti-inflammatory drugs
COX 1 (aspirin) vs. COX 2
COX 2 drugs:
Carprofen
Meloxicam
Firocoxib
Robenacoxib
Deracoxib
Phenylbutazone
Benzodiazepines
Diazepam
Midazolam
What are benzodiazepines reversible with?
Flumazenil
Anticholinergics
Atropin
Glycopyrrolate (glyco)
Phenothiazines
Acepromazine (ACE)
Pain pathways
Transduction
Transmission
Modulation
Perception
Multimodal analgesia
Use of multiple analgesic drugs (often different classes) to target different points along the pain pathway
GOAL: to max pain relief w minimal side effects
Pre-emptive analgesia
Administration of pain meds prior to a painful procedure or event to prevent the establishment of pain
What drugs act at transduction
(Sensory cells - superficial)
Corticosteroids
Opioids
Local anes
NSAIDS
What drugs act at transmission
(Along nerves)
Alpha 2s
Local anesthetics
What drugs act at modulation
(Spinal cord - windup)
Local anesthetics
Opioids
NSAIDS
NMDA
Alpha 2
What drugs act at the level of perception
(Brain)
Benzodiazepines
Alpha 2s
Anesthetic agents
Opioids