Block 2 all drugs Flashcards
Q
Pyrimethamine
Sulfonamide
Dapsone
Sulfonamide.
Mafenide
topical sulfonamide
Phenazopyridine
Urinary Tract Analgesic NOT a sulfa
nitrofurantoin
urinary anti-infective
Fosfomycin
urinary anti-infective (phosphonic acid) NOT aminoglycoside
methenamine
Urinary Anti-infective ..
-floxacin
Fluoroquinolones
gentamicin
Aminoglycoside.
tobramycin
Aminoglycoside
amikacin
Aminoglycoside..
kanamycin
Aminoglycoside …
neomycin
Aminoglycoside ….
streptomycin
Aminoglycoside -
Penicillin G or V
1st generation PCNs
nafcillin
Penicillinase-Resistant Penicillin
oxacillin
Penicillinase-Resistant Penicillin .
cloxacillin
Penicillinase-Resistant Penicillin …
dicloxacillin
Penicillinase-Resistant Penicillin -
amoxicillin
Aminopenicillin (PO)
Ampicillin
Aminopenicillin (IV)
piperacillin
antipseudomonal penicillin
Ticarcillin
antipseudomonal penicillin -
amoxicillin/clavulanic acid
beta lactamase inhibitor antibiotic (PO)
Ampicillin/Sulbactam
beta lactamase inhibitor (restores activity)
piperacillin/tazobactam
antipseudomonal + beta lactamase inhibitor
Ticarcillin/Clavulanate
antipseudomonal + beta lactamase inhibitor -
cephradine
1st generation cephalosporin
cefadroxil
1st gen cephalosporin
cephalexin
first generation cephalosporin
cefazolin
1st Gen Cephalosporin (IV)
cefprozil
2nd gen cephalosporin, PO
loracarbef
2nd generation cephalosporin
cefaclor
Second Generation Cephalosporin PO
cefuroxime
2nd gen cephalosporin PO/IV
cefoxitin
2nd gen cephalosp IM/IV
cefotetan
2nd generation cephalosporin IM & IV
Ceftazidime ceftazidime/avibactam
3rd generation cephalosporin antipseudomonal
Cefotaxime
3rd gen cephalosporin NON-antipseudomonal
Ceftizoxime
3rd generation cephalosporin NON-antipseudomonal
Ceftriaxone
3rd generation cephalosporin NON-antipseudomonal IV or IM
cefdinir
Oral 3rd gen cephalosporin
cefixime
Oral 3rd generation cephalosporins NOT able to cross the BBB
cefpodoxime
PO - 3rd generation cephalosporin
ceftibuten
PO 3rd gen cephalosporin
cefditoren
3rd generation cephalosporin PO
Cefepime
4th generation cephalosporin
ceftaroline
5th generation cephalosporin
ceftolozane/tazobactam
new cephalosporins (5th)
aztreonam
monobactams
-penem
carbapenems
-cycline
tetracyclines
tigecycline
glycylcyclines
-thromycin
erythromycins
fidaxomicin
Macrolide
telithromycin
ketolide
clindamycin
lincosamides
vancomycin
glycopeptide IV & PO
dalbavancin
Glycopeptide
oritavancin
Glycopeptide IV
televancin
IV glycopeptide
daptomycin
lipoglycopeptide
colistin
Polymyxin IV
polymixin B
topical polymixin
-zolid
oxalodinones
Quinupristin/Dalfopristin
Streptogramins
chloramphenicol
“other”
bacitracin
topical antibiotic
gramicidin
topical ABX
mupirocin
topical - S. aureaus
-quine
anti-malarial
atovaquone/proguanil
Antimalarial
dapsone
antimalarial PO
doxycycline
PO antimalarial
metronidazole
anti-protazoal C. diff diarrhea
tinidazole
anti-protozoal
pyrantel pamoate
Antihelminthic .
Mebendazole
Antihelminthic ..
albendazole
Anthelmintic …
Ivermectin
Antihelminthic -
pentamidine
leishmaniasis & african trypanosomiasis
miltefosine
Leishmaniasis
Sodium stibogluconate
Leishmaniasis -
permethrin
scabies and lice
malathion
pediculicide 2nd line after permethrin
Benzyl alcohol lotion
lice (children)
Ivermectin lotion
lice (6 mo or older)
spinosad
lice treatment (4 yr and older)
lindane
pubic lice only use after all others fail
rifampin
anti-mycobacterial agent prophylaxis for meningitis
rifapentine
anti-TB
rifabutin
Anti-TB .
pyrazinamide
initial phase of active TB
ethambutol
first line active TB
isoniazid
DOC for both active and latent TB
streptomycin IV
Anti-TB, aminoglycoside
amphotericin B
polyenes DOC for cryptococcal meningitis
nystatin
topical antifungal
Ketoconazole
azole antifungals last line option
-conazole
antifungals
clotrimazole
antifungal PO candidia
terbinafine
allylamines PO & topical
naftifine
allylamines
butenafine
Allylamine ring worm
-fungin
echinocandins IV
griseofulvin
antifungal PO
selenium sulfide
tinea versicolor - antifungal
tolnaftate
antifungal ring worm, athletes foot, jock itch
Ciclopirox
nail lacquer antifungal
flucytosine
antifungal - PO
Clinical Use:
• Treatment of cryptococcal meningitis • Systemic fungal infections (e.g. septicemia, endocarditis, UTI, meningitis, or pulmonary) • Candidiasis in combination with Amphotericin B or fluconazole
acyclovir
anti-viral herpes
valacyclovir
suppression/treat HSV
gancyclovir
CMV IV
valgancyclovir
CMV - better bioavailability PO
foscarnet
last line CMV IV
trifluridine
anti-viral opth
cidofovir
agressive CMV - give fluids
penciclovir
HCV topical
Famciclovir
HSV - PO
docosanol
HSV topical
oseltamivir
anti-viral PO
zanamivir
influenza - inhalation
peramivir
influenza - IV - 18 and older
amantidine
anti-viral PO not for 2015-2016 flu virus
palivizumab
prophylaxis of immunocompromised infants with RSV
zidovudine
anti-viral (HIV) NRTI
efavirenz
anti-viral (HIV) NNRTI PO
lamuvidine
HIV (NRTI) & Hep. B
emtricitabine
HIV (NRTI)
tenofovir
(NRTI) HIV anti-viral Hep B
ritonavir
HIV (PI)
raltegravir
HIV integrase inhibitor
Dolutegravir
integrase inhibitor, HIV
Enfuvirtide
fusion inhibitor only for experienced patients
Darunavir
Protease Inhibitor (HIV)
Cobicistat
PK Booster (HIV)
Bictegravir (BIC)
integrase inhibitor (HIV)
Abacavir
NRTI (HIV)
Dolutegravir + abacavir + lamuvidine (Triumeq)
preferred regimen for naive HIV pt (HLA-B5701 negative)
Bictegravir/emtricitabine/tenofovir (Bicktarvy)
preferred regimen for naive HIV pt