Autonomic Drug Classifications Flashcards
Oxymetazoline
Nonselective Alpha agonist
Mecamylamine
Ganglionic blocker
Guanethidine
Sympathetic Modulator 1. Prevention of transmitter release
Atenolol
Beta 2 antagonist
Physostingmine
ACE Inhibitor
Triazolam
Skeletal muscle relaxant 1. Benzodiazepine
Dantrolene
Skeletal muscle relaxant 1. Treat malignant hyerthermia 2. Ryanodine receptor antagonist
Mivacurium
Competitive NMJ blocker 1. Short lasting
Epinephrine
Alpha 1, Alpha 2, Beta 1, Beta 2
Metoprolol
Beta 2 antagonist
Atracurium
Competitive NMJ blocker 1. Long lasting
Botulinum Toxin
ACh Release inhibitor 1. Treats dystonia, wrinkles, sweating
Succinylcholine
Depolarizing NMJ blocker 1. Fast onset, fast offset
Baclofen
Skeletal muscle relaxant 1. GABA agonist
Scopolamine
Mucarinic antagonist
Midazolam
Skeletal muscle relaxant 1. Benzodiazempine
Prazosin
Alpha 1 antagonist
Salmeterol
Beta 2 agonist
Pentolamine
Nonselective Alpha antagonist
Norepinephrine
Alpha 1, Alpha 2, Beta 1
Isoproterenol
Nonselective Beta agonist
Edrophonium
ACE Inhibitor
Doxazosin
Alpha 1 antagonist
Organophosphates
ACE Inhibitor 1. Toxicities seen with farm workers 2. Treat with atropine/2-PAM
Acetylcholine
Neurotransmitter
Albuterol
Beta 2 agonist
Acebutolol
Beta 2 antagonist (ISA)
Atropine
Mucarinic antagonist
Ipratropium
Mucarinic antagonist
Donepezil
ACE Inhibitor 1. Used for Alzheimer’s
2-PAM
ACE Reactivator
Bethanechol
Muscarinic agonist
Terbutaline
Beta 2 agonist
Dopamine
- Vasoconstriction to renal/splanctic 2. High levels = Norepinephrine
Tyramine
Sympathetic Modulator 1. Stimulant for release of NT from axon terminal
Clonidine
Alpha 1 agonist
Propranolol
Nonselective Beta antagonist
Pilocarpine
Muscarinic agonist
Tiotropium
Mucarinic antagonist
Ephedrine
Sympathetic Modulator 1. Stimulant for release of NT from axon terminal
Phenylephrine
Alpha 1 agonist
Labetalol
Nonselective Beta antagonist (mixed beta/alpha)
Metaproterenol
Beta 2 agonist
Diazepam
Skeletal muscle relaxant 1. Benzodiazepine
Tubocurarine
Competitive NMJ blocker
Reserpine
Sympathetic Modulator 1. Destruction of NE by MAO and depletion from nerve ending
Pindolol
Nonselective Beta antagonist (ISA)
Neostingmine
ACE Inhibitor
Phenoxybenzamine
Nonselective Alpha antagonist
Vecuronium
Competitive NMJ blocker 1. Long lasting