ANS pharm Flashcards
Dobutamine
β-1 and α-1 agonist
Dopamine
α and β agonist
Norepinephrine
α and β-1 agonist
Epinephrine
low dose – β-2 agonist
high dose – hits everything, esp α-1
Isoproterenol
non-selective β agonist
Clonidine
α-2 agonist
Methyldopa
α-2 agonist
Midodrine
α-1 agonist
Carvedilol
α-1 selective and β non-selective antagonist
Labetalol
β > α-1 antagonist
Doxazosine
α-1 antagonist
Metoprolol
β-1 antagonist
Propanolol
non-selective β-antagonist
Phentolamine
non-selective α antagonist
Phenoxylbenzamine
non-selective α antagonist
Atropine
non-selective muscarinic antagonist
Pyridostigmine
reversible inhibitor of AChE
What drug would you use for:
Bradycardia?
Isoproterenol
What drug would you use for:
Chronic orthostatic hypotension due to autonomic insufficiency?
Midodrine
What drug would you use for:
Acute hypotensive states?
Phenylephrine
Norepinephrine
What drug would you use for:
Shock and heart failure
Dopamine
What drug would you use for:
Acute heart failure
Dobutamine
What drug would you use for:
reversal of vagal bradycardia?
Atropine
What drug would you use for:
Treatment of neurogenic orthostatic hypotension?
Pyridostigmine