Sympathomimetics Flashcards
Epi
beta > alpha
NE
alpha1 > alpha2 > beta1
Isoproterenol
Beta1 = Beta2
Dopamine
Delta1 = Delta2 > Beta > Alpha
Dobutamine
Beta1 > Beta2, Alpha
Phenylephrine
Alpha1 > Alpha2
Albuterol, Salmeterol, Terbutaline
Beta2 > Beta1
Direct Sympathomimetics
Epi, NE, Isoproterenol, Dopamine, Dobutamine, Phenylephrine, Albuterol, Salmeterol, Terbutaline
Direct sympathomimetics. Alpha1 > Alpha2 > Beta1
NE
Direct sympathomimetics. Beta > Alpha
Epi
Direct sympathomimetics. Beta1 = Beta2
Isoproterenol
Direct sympathomimetics. Delta1 = Delta2 > Beta > Alpha
Dopamine
Direct sympathomimetics. Beta1 > Beta2, Alpha
Dobutamine
Direct sympathomimetics. Alpha1 > Alpha2
Phenylephrine
Direct sympathomimetics. Beta2 > Beta1
Albuterol, Salmeterol, Terbutaline
Indirect Sympathomimetics
Amphetamine, Ephedrine, Cocaine
Amphetamine
Reuptake inhibitor
Ephedrine
Release stored catecholamines
Cocaine
Reuptake inhibitor
Sympatholytics (alpha2 agonists)(2)
Clonidine, Alpha-methyldopa
Alpha blockers
Non-selective (2) Phenoxybenzamine, Phentolamine Alpha1 selective (4) Prazosin, Terazosin, Doxazosin, Tamsulosin Alpha2 selective (1) Mirtazapine
Non-selective alpha blockers (2)
Phenoxybenzamine (irr) and Phentolamine (rev)
Alpha1 selective blockers (4)
Prazosin, Terazosin, Doxazosin, Tamsulosin
Alpha2 selective (1)
Mirtazapine
Phenoxybenzamine
Non-selective alpha blocker, irreversible
Phentolamine
Non-selective alpha blocker, reversible
Prazosin
Alpha1 selective blocker
Terazosin
Alpha1 selective blocker
Doxazosin
Alpha1 selective blocker
Tamsulosin
Alpha1 selective blocker
Beta blockers
Metoprolol, Acebutolol, Betaxolol, Carvedilol, Esmolol, Atenolol, Nadolol, Timolol, Pindolol, Labetalol
Metoprolol
Beta blockers
Acebutolol
Beta blockers
Betaxolol
Beta blockers
Carvedilol
Beta blockers
Esmolol
Beta blockers
Atenolol
Beta blockers
Nadolol
Beta blockers
Timolol
Beta blockers
Pindolol
Beta blockers
Lebetalol
Beta blockers