Quiz1 A-C Flashcards
3MP
3-mercaptopropionic acid
Blocks GABA synthesis (anti GAD)
6-OH-DA
Kills DA and NE neurons
Allylglycine
Block GABA synthesis
Anti-pyridoxyl phosphate
Alphaxalone
Enhance GABA transmission
Via steroid site
Alprazolam
Enhances GABA-A
Benzodiazepine
Amitriptyline
Block NE and 5HT re-uptake
Amphetamine
Stimulates release of NE & DA
AMPT
Alpha-methylparatyrosine
Inhibit synthesis of NE and DA
Anti-hydroxylase
Atropine
Blocks postsynaptic mascarinic receptor
Belladonna - Galenical
Baclofen
Stimulates GABA-B receptors
Benzodiazepine
Enhance GABA-A transmission
Via BZ receptor
Benztropine
Block muscarinic receptor
Betacarbolines
Inverse BZ agonist
Bicuculline
Blocks muscarinic receptors
Black willow spider venom
Stimulates release of ACH
Botulinum Toxin
Inhibit ACh release
Bromides
Sedatives
Anti-seizure drugs of 19th century
Mechanism unknown
Buproprion
Block NE uptake?
Raise NE?
Antidepressant
Smoking cessation
Buspirone
5HT 1-A partial agonist
5HT autoreceptors - Lower 5HT
Antidepressant
Caffeine
blocks adenosine receptor
Coffee - galenical
Cannabis
Stimulates anandamide receptors (CB1 and CB2)
Galenical
Carbamazepine
Inhibit VGSC
Seizure
Neuropathic pain
Depression
Chloral hydrate
GABA-enhancer
Old sedative / hypnotic
“Mickey Finn”
Chlordiazepoxide
Enhances GABA-A transmission
Via BZ receptor
Citalopram
SSRI
Clobazam
Enhances GABA-A transmission
Via BZ receptor
Clonazepam
Enhances GABA-A transmission
Via BZ receptor
Clonidine
NE alpha2 autoreceptor Agonist
Inhibit NE release
Cocaine
Block re-uptake of NE and DA