Pharmacology Exam 4 Flashcards
Nadolol
Non-selective, water soluble
Pindolol
Non-selective, ISA
Propranolol
Non-selective, lipid soluble, without
Atenolol
B1-selective, water soluble, without
Esmolol
B1-selective, ultra-short acting, IV use only
Metoprolol
B1-selective, lipid soluble, without
Carvedilol
alpha 1 blocking, anti-oxidant
Labetalol
alpha 1 blocking, used for hypertension and in pregnancy
Nebivolol
Increases NO synthesis
Acetylcholine
Muscarinic Agonist
Bethanechol
Muscarinic Agonist, GI and urinary tract
Cevimeline
Muscarinic Agonist (Helps Sjogren’s Syndrome by increasing saliva and lacrimal production)
Methacholine
Muscarinic Agonist
Pilocarpine
Muscarinic Agonist, glaucoma
Donepezil
AChesterase Inhibitor (Helps Alzheimer’s)
Ecothiophate
AChesterase Inhibitor
Edrophonium
AChesterase Inhibitor
Galantamine
AChesterase Inhibitor (Helps Alzheimer’s)
Neostigmine
AChesterase Inhibitor
Pyridostigmine
AChesterase Inhibitor
Rivastigmine
AChesterase Inhibitor (Helps Alzheimer’s)
Sarin
AChesterase Inhibitor (an organophosphate)
Tacrine
AChesterase Inhibitor (Helps Alzheimer’s)
Atropine
Muscarinic ANTagonist
Darifenacin
Muscarinic ANTagonist
Homatropine
Muscarinic ANTagonist
Scopolamine
Muscarinic ANTagonist
Tropicamide
Muscarinic ANTagonist, dilate pupils
Ipratropium
Muscarinic ANTagonist, manage asthma
Tiotropium
Muscarinic ANTagonist, manage asthma
Pralidoxime
Regenerates ACh, treatment of organophosphates
Cyclopentolate
Muscarinic ANTagonist, dilate pupils
Hyoscine
Muscarinic ANTagonist, prevent motion sickness
Benzhexol
Muscarinic ANTagonist, prevent Parkinsonism
Benztropine
Muscarinic ANTagonist, prevent Parkinsonism