P450 Interactions Flashcards
Phenytoin
inducer, substrate, inhibitor
induces P450
Ritonavir
inducer, substrate, inhibitor
inhibits P450
Rifampin
inducer, substrate, inhibitor
induces P450
Amiodarone
inducer, substrate, inhibitor
inhibits P450
Macrolides (except Azithromycin)
inducer, substrate, inhibitor
inhibits P450
Griseofulvin
inducer, substrate, inhibitor
induces P450
mnemonic for inducers of P450
CHRONIC ALCOHOLics STeal PHEN-PHEN and Never Refuse Greasy CARBs
St. John’s Wart
inducer, substrate, inhibitor
induces P450
Acute Alcohol Abuse
inducer, substrate, inhibitor
inhibits P450
Warfarin
inducer, substrate, inhibitor
substrate of P450
Chronic Alcohol use
inducer, substrate, inhibitor
induces P450
mnemonic for Inhibitors of P450
AAA RACKS IN GQ Magazine
Nevirapine
inducer, substrate, inhibitor
induces P450
Isoniazid (INH)
inducer, substrate, inhibitor
inhibits P450
Cimetidine/Ciprofloxacin
inducer, substrate, inhibitor
inhibits P450
mnemonic for Substrates of P450
Always Think When Outdoors
Theophylline
inducer, substrate, inhibitor
substrate of P450
Ketoconazole
inducer, substrate, inhibitor
inhibits P450
Grapefruit Juice
inducer, substrate, inhibitor
inhibits P450
Carbamazepine
inducer, substrate, inhibitor
induces P450
Phenobarbital
inducer, substrate, inhibitor
induces P450
OCP
inducer, substrate, inhibitor
substrate of P450
Anti-epileptics
inducer, substrate, inhibitor
substrate of P450
Quinidine
inducer, substrate, inhibitor
inhibits P450