Inhalers and related drugs Flashcards
MDI general information and instructions?
metered dose inhalers contain a hydrofluoroalkane propellant
• To use: shake 10 seconds → exhale fully → place inhaler one or two fingers from mouth → start inhaling as the button is pressed → finish inhalation → hold breath 10 seconds → exhale via nose → rinse mouth
DPI general info and instructions?
dry powder inhalers
• To use: exhale fully → make tight seal around inhaler → quick, deep inhale → hold breath 10 seconds → exhale via nose → rinse mouth
asthma definition?
inflammatory condition of the lungs caused by inflammatory mediators
inflammatory mediators?
histamine, leukotrienes, prostaglandins
bronchodilators vs. steroids:
- Use bronchodilator first, then steroid to treat underlying cause
- Inhaled bronchodilators; only treat symptoms
Beta-2 agonists details:
sympathomimetics
stimulate beta-2 receptors in the lungs → bronchodilaton
rescue inhaler details
- Onset of 5 minutes
* Metered dose inhalers; used QID
rescue inhaler generics?
albuterol, levalbuterol, pirbuterol class of all is beta-2 agonists
albuterol Trades?
Proventil HFA, Ventolin HFA, ProAir HFA
albuterol details?
beta-2 agonist
• Racemeic
• May have more side effects
levalbuterol Trade and details?
Xopenex HFA (quick relief, beta-2 agonist)
• R-isomer
• May have fewer side effects than albuterol
Xopenex generic?
levalbuterol
beta-2 agonist
Maxair generic and details?
pirbuterol (quick relief, beta-2 agonist)
Autohaler - breath activated MDI
pirbuterol Trade?
Maxair Autohaler
quick relief beta-2 agonist
long term control inhalers info?
beta-2 agonists (sympathomimetics)
• Indicated for asthma prophylaxis → will not relieve acute attack
• Dry powder inhalers
• BBW: increases risk of asthma related deaths in patients who use this alone instead of in combination with a steroid
long-term control Beta-2 generics?
salmeterol, indacaterol, formoterol
Serevent generic?
salmeterol
long acting beta-2 agonist
salmeterol Trade and details?
Serevent Diskus (long acting beta-2 agonist) • BID - DPI • Number on the top of the diskus means the number of doses remaining
Foradil generic?
formoterol
sympathomimetic - long acting
formoterol Trade and details?
Foradil Aerolizer (long acting b-2 agonist)
• BID - DPI
• Refrigerate in the pharmacy
• Can be kept at room temperature for 4 months by the patient
indacaterol Trade and details?
Arcapta NeoHaler (long acting b-2 agonist) qday -- DPI
Arcapta generic?
indacaterol
long acting b-2 agonist
anticholinergic bronchodilator details?
o Block cholinergic receptors in the lungs → blocks ACh → bronchodilation
o Indicated for asthma prophylaxis
o Side effect: xerostomia
anticholinergic bronchodilator generics?
ipratropium, tiotropium, aclidinium
ipratropium bromide + albuterol
ipratropium Trade and details?
Atrovent HFA (anticholinergic)
• QID
• MDI
tiotropium Trade and details?
Spiriva Handihaler (anticholinergic) • qday - long acting • DPI
aclidinium Trade and details?
Tudorza Pressair (anticholinergic) • BID - long acting • DPI
combination anticholinergic brochodilator generics?
albuterol, ipratropium bromide
combination bronchodilator Trade and details?
Combivent Respimat (albuterol, ipratropium bromide)
• MDI
• Rescue inhaler
• Contains soya lecithin; do not use if allergic to soy or peanuts
bronchodilators for nebulization details?
o Used in an updraft machine; drug diluted with normal saline
• Put solution for nebulization in machine → machine nebulizes liquid into a mist and patient breathes in with a mask for about 15 minutes
generics available for nebulization?
albuterol, levalbuterol, ipratropium, arformoterol, combo of albuterol and ipratropium
AccuNeb generic?
albuterol (nebulization)
QID
albuterol Trade for nebulization?
AccuNeb QID
Xopenex generic nebulization?
levalbuterol
QID
no Trade generic for nebulization?
ipratropium
QID
levalbuerol Trade for nebulization?
Xopenex solution for nebulization
arformoterol Trade?
Brovana
nebulization
Brovana generic and details?
arformoterol for nebulization • BID • R-isomer of formoterol • Long-acting • Refrigerate in the pharmacy
combination nebulization product Trade?
DuoNeb
DuoNeb generic and details?
albuterol, ipratropium for nebulization
QID
Inhaled corticosteroid details?
• Treat underlying cause of asthma by decreasing inflammation in the airways
• Indicated for asthma prophylaxis; will not relieve acute attack - Maintenance drugs
• Side effect: oral candidiasis
o Rinse mouth with water 15 minutes after using inhaler
QVAR generic and details?
beclomethasone
inhaled corticosteroid
MDI - BID
beclomethasone Trade?
QVAR
inhaled corticosteroid
Flovent generic and details?
fluticasone
inhaled corticosteroid
MDI - BID
budesonide Trade?
Pulmicort Flexhaler and Pulmicort Respules
Pulmicort Flexhaler details?
budesonide - inhaled corticosteroid
BID - DPI
Pulmicort Respules details?
budesonide - inhaled corticosteroid
BID - suspension for nebulization
mometasone Trade?
Asmanex Twisthaler
inhaled corticosteroid
Asmanex generic and details?
mometasone - inhaled corticosteroid
qday - DPI
• 4-11 years old: 110 mcg
• 12+ years old: 220 mcg
ciclesonide Trade and details?
Alvesco - inhaled corticosteroid
MDI - BID
Alvesco generic?
cclesonide - inhaled corticosteroid
thrush details?
oral cadidiasis - candida albicans
medications indicated for thrush?
gentian violet, nystatin, clotrimazole troches
gentian violet details?
- OTC
* Topical antiseptic - thrush
nystatin details?
- Rx only
* Antifungal- thrush
clotrimazole details?
- Rx only
- Imidazole antifungal - thrush
- Dissolve 1 troche in the mouth five times daily x 14 days
combination bronchodilator/corticosteroid indication?
asthma prophylaxis
Symbicort generic and details?
budesonide, formoterol
• Combination bronchodilator/corticosteroid
MDI - BID
budesonide, formoterol Trade?
Symbicort
• Combination bronchodilator/corticosteroid
Dulera generic and details?
mometasone, fomoterol
• Combination bronchodilator/corticosteroid
MDI - BID
mometasone, formoterol Trade?
Dulera
• Combination bronchodilator/corticosteroid
Advair generic and details?
fluticasone, salmeterol
• Combination bronchodilator/corticosteroid
BID
fluticasone, salmeterol Trade?
Advair HFA (MDI - BID) Advair Diskus (DPI - BID)
inhaled antiviral agents details?
- Indicated for treatment and prevention of the flu
* Neuraminidase inhibitors: neuraminidase is the enzyme that influenza needs to replicate
antiviral agent generics?
oseltamivir and zanamivir
neuraminidase inhibitors
zanamivir Trade and details?
Relenza Diskhaler
• 5 mg powder/blister - DPI
• Treatment: 10 mg BID x 5 days
• Prevention (household): 10 mg qday x 10 days
• Prevention (community): 10 mg qday x 28 days
oseltamivir Trade and details?
Tamiflu - tablet
Beconase generic?
beclomethasone
intranasal corticosteroid
Nasacort generic?
triamcinolone
intranasal corticosteroid
Rhinocort generic?
budesonide
intranasal corticosteroid
no Trade intranasal corticosteroid?
flunisolide
Flonase generic?
fluticasone propionate
intranasal corticosteroid
Veramyst generic?
fluticasone furoate
intranasal corticosteroid
Nasonex generic?
mometasone
intranasal corticosteroid
Omnaris generic?
ciclesonide
intranasal corticosteroid
beclomethasone Trade?
nasal
Beconase AQ
intranasal corticosteroid
triamcinolone Trade?
Nasacort AQ
intranasal corticosteroid
budesonide Trade?
nasal
Rhinocort Aqau
intranasal corticosteroid
fluticasone Trades?
nasal
Flonase - propionate
Veramyst - furoate
intranasal corticosteroid
mometasone Trade?
nasal
Nasonex
intranasal corticosteroid
ciclesonide Trade (nasal)
Omnaris
intranasal corticosteroid
intranasal mast cell stabilizer
Nasalcrom - cromolyn sodium
intranasal pituitary hormone
DDAVP, Stimate - desmopressin acetate
intranasal anticholinergic?
Atrovent Nasal Spray - ipratropium bromide
intranasal antihistamine?
Astelin, Astepro - azelastine
Combination intranasal?
Dymista - azelastine, fluticasone
intranasal for osteoporosis?
Miacalcin - calcitonin
Fortical - calcitonin
Leukotriene receptor antagonist indication:
inflammatory mediator
Ind: asthma prophylaxis
Leukotriene receptor antagonists generics?
zafirlukast, montelukast, zileuton (kind of)
zafirlukast Trade and details?
Accolate
o Leukotriene receptor antagonists
take on empty stomach
montelukast Trade and details?
Singulair (leukotriene receptor antagonist)
• qday
• Indicated for prevention of exercise-induced asthma (2 hours prior), asthma prophylaxis, and allergic rhinitis
• 10 mg tablet: 15 and older
• 4 mg chewable tablet: 2-5 years old
• 5 mg chewable tablet: 6-14 years old
• 4 mg/packet granules: 6 months-5 years old; can sprinkle on food, but do not mix with liquid
• Can be taken without regard to meals
zileuton Trade and details?
Zyflo CR
• Leukotriene formation inhibitor
• ER tablet
• BID