hypertension drugs Flashcards
Amlodipide brand name and class
Norvasc
CCB
Atenolol brand name and class
Tenormin
Beta blocker
Clonidine brand name and class
Catapres
alpha agonist
Enalapril brand name and class
Vasotec
ACE inhibitor
HCTZ brand name and class
Microzide
thiazide diuretic
Labetalol brand name and class
Trandate
beta blocker
Lisinopril brand name and class
Zestril
ACE inhibitor
Losartan brand name and class
Cozaar
ARB
Metoprolol succinate brand name and class
Toprol XL
Beta blocker
Metoprolol tartrate brand name and class
Lopressor
beta blocker
Nifedipine brand name and class
Procardia
CCB
Valsartan brand name and class
Diovan
ARB
Amlodipine dosing
Start: 2.5-5 mg/day
Next: 5 mg/day
Max: 10 mg/day
Atenolol dosing
Start: 25 mg/day
Next: 50 mg/day
Max: 100 mg/day
Clonidine dosing
PO: 0.1 mg BID
Max: 2.4 mg/day
usual 0.1 - 0.2 mg BID
Transdermal: 0.1 mg/24 hr patch applied q7days, increase by 0.1 at 1 week intervals if necessary (available as 0.1, 0.2 and 0.3 mg/24 hr patch)
Enalapril dosing
Start: 2.5 mg BID
Next: 10 mg/day or 5 mg BID
Max: 40 mg/day or 20 mg BID
HCTZ dosing
Start: 12.5 mg/day
Next: 25 mg/day
Max: 50 mg/day
Labetalol dosing
Start: 100 mg BID
Next: 200 mg BID
Max: 400 mg BID
Lisinopril dosing
Start: 10 mg/day
Next: 20 mg/day
Max: 40 mg/day
Losartan dosing
Start: 25 mg/day
Next: 50 mg/day in 1-2 doses
Max: 100 mg/day in 1-2 doses
Metoprolol succinate dosing
Start: 25 mg/day
Next: 50 mg/day
Max: 400 mg/day
Metoprolol tartrate dosing
Start: 25 mg BID
Next: 50 mg BID
Max: 200 mg BID
Nifedipine dosing
Start: 30 mg/day
Next: 60 mg/day
Max: 90 mg/day (120 according to Lexicomp)
Valsartan dosing
Start: 80 mg/day
Next: 160 mg/day
Max: 320 mg/day
Amlodipine side effects
Amlodipine specific: dose related palpitations
All CCBs: tachycardia, dizziness, HA, flushing, peripheral edema, gingival hyperplasia
Atenolol side effects
Atenolol specific: impotence, nightmares, insomnia
All beta blockers: bronchospasm, bradycardia, masked hypoglycemia, impaired peripheral circulation, fatigue, decreased exercise tolerance, depression, withdrawal syndrome
Clonidine side effects
Dry mouth, sedation, depression, withdrawal syndrome
Enalapril side effects
Enalapril specific: hypotension, dizziness, HA
All ACE inhibitors: cough, angioedema, hyperkalemia, loss of taste, acute renal failure, glomerulonephritis, neutropenia, agranulocytosis, proteinuria
HCTZ side effects
HCTZ specific: hypotension, nausea, diarrhea
All thiazide diuretics: hypokalemia, hypomagnesemia, hypercalcemia, hyperuricemia, hyperglycemia, hyperlipidemia, sexual dysfunction, lithium toxicity w/ concurrent administration
Labetalol side effects
Labetalol specific: nausea, increased BUN
all beta blockers: bronchospasm, bradycardia, masked hypoglycemia, impaired peripheral circulation, fatigue, decreased exercise tolerance, depression, withdrawal syndrome
Lisinopril side effects
Lisinopril specific: hypotension, dizziness, syncope, increased BUN, increased SCr (often transient)
all ACE inhibitors: Cough, Angioedema, Hyperkalemia, Loss of Taste, Acute Renal Failure, Glomerulonephritis, Neutropenia, Agranulocytosis, Proteinuria
Losartan side effects
Losartan specific: Diarrhea, Chest Pain, Hypoglycemia, Cough
all ARBs: Orthostatic Hypotension, Renal Insufficiency, Hyperkalemia
Metoprolol side effects
Metoprolol specific: Hypotension, Dizziness, Pruritus, Rash, Diarrhea
all beta blockers: Bronchospasm, Bradycardia, Masked hypoglycemia, Impaired peripheral circulation,Fatigue, Decreased Exercise Tolerance, Depression, Withdrawal syndrome
Nifedipine side effects
Nifedipine specific: Nausea, Heart Burn
all CCBs: Tachycardia, Dizziness, Headaches, Flushing, Peripheral Edema, Gingival Hyperplasia
Valsartan side effects
valsartan specific: Dizziness, Increased BUN
all ARBs: Orthostatic Hypotension, Renal Insufficiency, Hyperkalemia
amlodipine monitoring
Heart rate, blood pressure
atenolol monitoring
ECG, blood pressure
clonidine monitoring
Blood pressure, standing and sitting/supine, mental status, heart rate
enalapril monitoring
Blood pressure, serum creatinine, serum potassium, renal function within 1-2 weeks of initiations
HCTZ monitoring
Assess weight, ins & outs reports daily to determine fluid loss, blood pressure, serum electrolytes, BUN, creatinine
Labetalol monitoring
Blood pressure, standing and sitting/supine, pulse
lisinopril monitoring
BUN, serum creatinine, renal function, WBC, and potassium
Hypotensive effects within 1 to 3 hours of initial dose or with increased dosages
Consider baseline hepatic function tests (if pre-existing hepatic impairment)
losartan monitoring
Supine blood pressure, electrolytes, serum creatinine, BUN, urinalysis, symptomatic hypotension and tachycardia, CBC
metoprolol monitoring
Heart rate, blood pressure
nifedipine monitoring
Heart rate, blood pressure, signs and symptoms of CHF, peripheral edema
valsartan monitoring
Baseline and periodic electrolyte panels, renal function, BP
In HF, serum potassium during dose escalation and periodically thereafter
Hyzaar
losartan + HCTZ
Lotrel
amlodipine + benazepril
Maxide
HCTZ + triamterine
Zestoretic
lisinopril + HCTZ