HIV Meds Flashcards
Abacavir
NRTI
Nausea, hypersensitivity rxn
Didanosine
NRTI
Pancreatitis, peripheral neuropathy, nausea, diarrhea, xerostomia
Emtricitabine
NRTI
Minimal side effects
Nausea, rare CNS effects and lactic acidosis
Lamivudine
NRTI
Minimal side effects
Nausea, rare CNS effects and lactic acidosis
Stavudine
NRTI
Peripheral neuropathy, lactic acidosis
Tenofovir
NRTI
Abd pain, diarrhea, n/v, gas, rare neutropenia, elevated LFTs, hypermylasemia
Zidovudine
NRTI
Anemia, neutropenia, headache, fatigue, anorexia, lactic acidosis, nausea
Delavirdine
NNRTI
Rash, nausea
Efavirenz
NNRTI
Nightmares, nausea, dizziness, rash, CNS changes
induce CYP450 and 3A4
Etravirine
NNRTI
Rash, hypersensitivity rxn, nausea
Nevirapine
NNRTI
Rash, hepatitis, nausea, hypersensitivity Rxn
induce CYP450 and 3A4
Rilpivirine
NNRTI
HA, rash, depression, insomnia
Amprenavir
PI
Nausea, HA, diarrhea
Atazanavir
PI
indirect hyperbili, prolonged PR
Darunavir
PI
Skin rash, SJS
Fosamprenavir
PI
Skin rash, diarrhea, n, HA
Indinavir
PI
nephrolithiasis, abd pain, diarrhea, elevated LFTs, HA, rash, dizziness, altered taste, n, thrombocytopenia
Lipinavir/ritonavir
PI
nausea, diarrhea, rash
Nelfinavir
PI
Diarrhea, nausea
Ritonavir
Booster to other PIs
Nausea, HA, diarrhea, circumoral paresthesia, elevated LFTs
saquinavir
PI
elevated LFTs, HA, nausea, diarrhea, CNS changes
Raltegravir, dolutegravir, Elvitegravir
Integrase inhibitors
nausea, HA, diarrhea, CPK elevation
Enfuvirtide
Fusion inhibitor
Rxn at injection site, bacterial PNA
Maraviroc
CCR5 antagonist
Abd pain, cough, dizziness, rash, hepatotox, MSK sx