GABA, glycine drugs Flashcards
1
Q
Muscimol
A
GABA-A orthosteric agonist
2
Q
Isoguvacine
A
GABA-A orthosteric agonist
3
Q
Bicuculline
A
GABA-A orthosteric antagonist
4
Q
Flumazenil
A
Benzodiazepine antagonist on GABA-A receptors
5
Q
Beta carboline (CCE)
A
Negative allosteric modulator of benzodiazepine site on GABA-A receptors
6
Q
Alphaxalone
A
Positive allosteric modulator at neurosteroid site on GABA-A receptors
7
Q
Picrotoxin
A
Agonist at channels site on GABA-A receptors
8
Q
Baclofen
A
Agonist at GABA-B receptors
9
Q
Phaclofen
A
Antagonist at GABA-B receptors
10
Q
Vigabatrin
A
GABA transaminase inhibitor
11
Q
Valproate
A
GABA transaminase inhibitor
12
Q
Tiagabine
A
GAT-1 inhibitor
13
Q
DABA
A
GAT-1 inhibitor
14
Q
Beta-alanine
A
GAT2,3 inhibitor
15
Q
Strychnine
A
Glycine receptor antagonist
