Final Exam Drugs Flashcards
Cefazolin
1st Gen Cephalosporins
I.M. I.V.
Cephalexin
1st Gen Cephalosporins
Oral
Cefaclor
2nd Gen Cephalosporins
Oral
Cefuroxime
2nd Gen Cephalosporins
I.M. I.V.
Cefprozil
2nd Gen Cephalosporins
Oral
Ceftriaxone
3rd Gen Cephalosporins
I.M. I.V.
Cefixime
3rd Gen Cephalosporins
Oral
Cefepime
4th Gen Cephalosporins
I.V.
Ceftaroline
5th Gen Cephalosporins
I.V.
Aztreonam
Monobactam
I.M.
Vancomycin
Monobactam
I.M.
“romycin’s”
Macrolides
Oral, I.V.
“other mycins”
Aminoglycosides
IV/IM, topical
“cycline’s”
Broad Spectrum
Oral
Doxy- antimalarialsd
Chloramphenicol
Broad Spectrum
I.M.
Chloroquine
Anti-Malarial, DOC for all forms
Quinine sulfate/gluconate
Anti-Malarial, schizonticidal, DOC for Chloroquine resistant
Mefloquine
Anti-Malarial, DOC for prophylaxis, another 1st-line for Chloroquine resistant
Pyrimethamine + Sulfadoxine
Anti-Malarial, inhibition of folate metabolism, PRESUMPTIVE treatment
Atovaquonen + Proguanil (Malarone)
Anti-Malarial, mitochondrial inhibitor
Artemether + Lumefantrine (Coartem)
Anti-malarial, schizonticide
Primaquine
Anti-Malarial, exoerythrocytic AND gametocytic
Amantadine
Anti-viral, inhbits viral uncoating, influenza A (parkinson’s)
Oseltamivir
Anti-viral, Inhibits viral neuraminidase (prevents release of particles from infected cells), inluenza A+B (H5N1 bird flu)
Acyclovir
Anti-viral, inhibits DNA synthesis, herpes/varicella, alteration of viral thymidine kinase (resistance)
Ganciclovir
Anti-viral, Inhibits DNA synthesis (requires phosphorylation), causes myelosupression
HAART - Highly Active Anti-retroviral Therapy
Treatment of HIV
Zidovudine
HIV drug, NRTI- Nucleoside reverse transcriptase inhibitor, can cause myelosuppression.
Nevirapine
HIV drug, NNRTI- NonNucleoside Reverse Transcriptase Inhibitor, high SJS
Interferon Alfa-2a
Anti-viral, Immunomodulatory protein, Hep B/C, suppress proliferation and inhibit replication, Severe flu symptoms/ psychiatric effects
Ribavirin
Anti-viral, inhibits viral RNA/DNA synthesis, RSV/influenza/Hep C
Meclorethamine
Anti-cancer
Cyclophosphamide
Anti-cancer
Cisplatin
Anti-cancer
Methotrexate
Anti-cancer
Doxorubicin
Anti-cancer
Vincristine
Anti-cancer
Vinblastine
Anti-cancer
Paclitaxel
Anti-cancer
Etoposide
Anti-cancer
Topotecan
Anti-cancer
Ciprofloxacin
Fluoroquinolones
Levofloxacin
Fluoroquinolones
Nitrofurantoin
UTI drug
Methanamine
UTI drug
Metronidazole
UTI drug
Daptomycin
Against Gram +
Mupiricin
Against Gram +
Polymixin
Against Gram -