Farma vascular Flashcards

1
Q

Sulfonilureas

A

Glibenclamida, Glicazida, Glimperida, Glipizida, Glisentida

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2
Q

Mecanismo de acción sulfonilureas

A

Antagonistas de los canales de potasio célula bata del páncreas

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3
Q

Reacciones adversas sulfonilureas

A
  • Hipoglucemia
  • Aumento de peso
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4
Q

Meglitinidas

A

Repaglinida, Nateglinida

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5
Q

Mecanismo de acción Meglitinidas

A

Antagonistas de los canales de potasio célula bata del páncreas
La diferencias con las Sulfonilureas es que la duración del efecto es muy corta

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6
Q

Biguanidas

A

METFORMINA (fármaco estrella)

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7
Q

Matfornina reacciones adversas

A

NO produce hipoglucemia

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8
Q

Tiazolidindionas

A

Pioglitazona

  • Agonista del receptor que favorece la lecturad e genes con efecto antidabéticos
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9
Q

Inhibidores de la alfa-glucosidasa

A

Acarbosa, Miglitol

Hace que no se rompan los hidratos de carbono de la dieta

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10
Q

Miméticos de GLP-1

A

Selmaglutida, exenatida

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11
Q

Inhibidores de DPP4

A

Sitagliptina…
-gliptina

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12
Q

Glifozinas (terminación)

A

-gliflozina

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13
Q

Mecanismo de acción glifozinas

A

Inhiben SGLT-2

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14
Q

Reacciones adversas glifozinas

A
  • Combinación sulfonilurea o insulna –Z hipoglucemia
  • Infecciones genitourinarias (aumento de glucosa en orina)
  • Hipotensión
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