Exam 2 Drugs Flashcards
Glycopyrrolate
Direct muscarinic antagonist
atropine
Direct muscarinic antagonist
Tolterodine
Direct muscarinic antagonist
Ipatropium
Direct muscarinic antagonist (bronchodilator)
ACh
Direct cholinergic neurotransmitter
Methacholine
Direct muscarinic agonist (additional methyl group on ACh)
Bethanechol
Direct muscarinic agonist (NH2 and methyl substitution on ACh)
Pilocarpine
Direct muscarinic agonist
muscarine
Direct muscarinic agonist
Edrophonium
Cholinergic Indirect acting agonist (AChE inhibitor)
Physostigmine
Nicotinic Indirect acting agonist (reversible AChE Inhibitor)
Neostigmine
Nicotinic Indirect acting agonist
Malathion (insecticide)
Nicotinic Indirect acting agonist
Nerve Gas
Nicotinic Indirect acting agonist (irreversibly blocks AChE)
What do you give to someone with Nerve gas poisoning?
Atropine and 2 PAM pralidoxime
Nicotine
Nicotinic agonist/antagonist
Succinlycholine
Nicotinic agonist/antagonist
Trimethaphan
Nicotinic antagonist/ganglionic blocker (antihypertensive use)
Atracurium
Nicotinic antagonist/ND NMB
Pancuronium
Nicotinic antagonist/ND NMB
Rocuronium
Nicotinic antagonist/ND NMB
Curare
Nicotinic antagonist/ND NMB
Phenylephrine
Alpha 1 direct agonist
NE
Alpha and Beta direct agonist (greatest affinity for alpha 1)
Epi
direct agonist Alpha and Beta (B>A)
Isoproternal (used to treat bradycardia)
Beta agonist (1=2)
Dobutamine (assists in Heart contractility)
Beta agonist (1>2»>A)
Albuterol
Beta agonist (2»1»»A)
Amephetamine
Indirect Alpha/Beta agonist (releasing agent)
Ephedrine
Indirect Alpha/Beta agonist (A1 = A2; B1=B2>A1)
Reserpine
Indirect antagonist for Alpha/Beta
Cocaine
Indirect agonist for Alpha/Beta (Uptake Inhibitor)
Clonodine
Direct alpha 2 agonist
Dexmedetomidate
Direct Alpha 2 agonist (sedative w/o decreasing respiration)
Doxazosin
Indirect Alpha 1 antagonist (used to treat hypertension)
Labetalol
Beta/alpha antagonist (B1-2 > A1»_space;>A2)
will reduce HR and cause bronchoconstriction
Metoprolol (used to treat angina and hypertension)
Direct Beta antagonist (B1»_space;> B2)
Propanolol
Beta antagonist (B1=B2) beta blocker
Tetredotoxin
Indirect Antagonist for all Na+ channels
Conotoxin
Indirect Antagonist for all Ca++ channels
Botulinum toxin
Indirect nicotinic antagonist