Drugs Related to Hypothalamic and Pituitary Hormones Flashcards
Somatrem or somatropin MOA?
GH analog
Octreotide MOA?
somatostatin analog
Cosyntropin MOA?
ACTH analog
Urofollitropin MOA?
FSH analog
Placental HCG MOA?
LH analog
Menotropins MOA?
FSH and LH analogs
Cabergoline MOA?
PIH (prolactin inhibiting hormone) (DA) analog
Oxytocin indications?
labor induction
Desmopressin MOA?
vasopressin analog
Indications for somatropin?
pituitary dwarfism, osteoporosis
Indications for octreotide?
acromegaly, carcinoid and secretory- GI tumors
Indictions Cosyntropin
Infantile spasms
Indications nafarelin?
endometriosis, prostate carcinoma (repository form)
Indication Cabergoline?
hyperprolactinemia
Indications Desmopressin (V2 selective)?
- neurogenic (pituitary) DI
- Hemophilia A (inc. factor VIII from liver)
- von Willebrand disease (inc. vW factor from endothelium)
- Primary nocturnal enuresis
What are the indications for leuprolide use?
endometriosis, prostate carcinoma (repository form)
What is the use for placental HCG?
hypogonadal states
Indications for menotropins?
hypogonadal states
Indications for urofollitropin?
hypogonadal states
What are some drugs used to treat SIADH?
demeclocyline, tolvaptan, loop diuretics
MOA demeclocyline which makes it useful in treating SIADH?
V2 receptor blockers in collecting duct