DRUGS NAME Flashcards

1
Q

LIST TYPICAL DRUGS OF SCHIZOPHENIA

A

HALOPERIDOL
ZUCLOPENTHIXOL
SULPIRIDE
PROCHLOROPERAZINE
CHLOROPROMAZINE

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2
Q

WHAT IS MOA OF PROCHLOROPERAZINE

A

-BLOCK DOPAMINE REUPTAKE
- EFFECTIVE TOWARDS POSITIVE SYMPTOMS

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3
Q

WHY ZUCLOPENTHIXOL DIDNT RECOMMEND AS A FIRST LINE TREATMENT IN SCHIZOPHENIA

A

GIVING EXTRAPRAMYDAL SIDE EFFECT

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4
Q

WHY QUETIAPINE WAS RECOMMENDED AS FIRST LINE TREATMENT IN SCHIZOPHENIA

A

ITS GIVING METABOLIC CHANGES SUCH AS HYPERGLYCEMIA , HYPERLIPIDEA AND EXCESSIVE WEIGHT GAIN

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5
Q

WHAT IS MOA OF OLAZAPINE

A

-BLOCK DOPAMINE AND SEROTONIN IN SOME EXTENT
- EFFECTIVE TOWARDS POSITIVE AND NEGATIVE SYMPTOMS IN SOME EXTENT

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6
Q

NAME DRUG THAT WAS GIVING AFTER 2 ANTIPSYCHOTICS DRUGS FAILED TO RESPOND IN PATIENT AND WHY

A
  • CLOZAPINE
  • AS A ;LAST RESORT OF TREATMENT
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7
Q

LIST ATYPICAL ANTIPSYCHOTICS DRUGS

A
  • OLAZAPINE
    -CLOZAPINE
  • AMISULPRIDE
  • ARIPIPRAZOLE
  • QUETIAPINE
    -RISPERIDONE
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8
Q

LIST NAME ANTI DEPRESSANT DRUGS IN TRYCLIC ANTI DEPRESSANT (TCA)

A
  • NORTRIPTYLINE
  • AMITRIPTYLINE
    -CLOMIPRAMINE
    -DOTHIEPIN HCL
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9
Q

WHAT IS MOA OF AMITRIPTYLINE

A

BLOCK SEROTONIN AND NORADRENALINE REUPTAKE TRANSPORTER

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10
Q

WHAT IS PHARMACOLOGICAL CLASS OF PHENELZINE

A

MONOAMINE OXIDASE INHIBITOR ANTI DEPRESSANT

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11
Q

EXPLAIN WHAT SHOULD PATIENT BE AWARE WHEN PRESCRIBED WITH PHENELZINE

A

-HIGH TYRAMINE FOOD
-SINCE THERE IS NOT MONOAMINE OXIDASE ENZYME MORE TYRAMINE AVAILABLE IN OUR BODY
- HENCE IT CAN LEAD TO HYPERTENSION

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12
Q

EXPLAIN MOA OF PHENELZINE

A
  • INHIBIT MONOAMINE OXIDASE ENZYME THAT DEGRADE SEROTONIN AND NORADRENALINE
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13
Q

WHAT IS PHARMACOLOGICAL CLASSIFICATION OF ESCITALOPRAM

A

SELECTIVE SEROTONIN REUPTAKE INHIBTOR ANTI DEPRESSANT

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14
Q

WHAT IS MOA OF CITALOPRAM

A

-SELECTIVELY INHIBIT SEROTONIN REUPTAKE
-HENCE MORE SEROTONIN AVAILABLE

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15
Q

WHY DID PATIENT CONDITION STILL NO PROGRESSION AFTER 1-2 WEEKS OF PRESCRIBED DRUG

A
  • WHEN TAKING ANTI DEPRESSANT DRUG IN EARLY TREATENT, IT ACTIVATED THE AUTO RECEPTOR OF SEROTONIN.
    -IT GIVING NEGATIVE FEEDBACK
  • HENCE MORE SEROTONIN AVAILABLE
  • HOWEVER AFTER 4- 6 WEEKS. AUTORECEPTOR WILL BE DECREASED
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16
Q

WHAT IS SEROTONIN SYNDROME

A
  • LIFE THREATENING CONDITION DUE OF EXCESSIVE LEVEL OF SEROTONIN
    -LEADS TO SYMPTOMS SUCH AS HIGH FEVER AND INDUCE SEIZURE
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17
Q

LIST SSRI DRUGS

A

-CITALOPRAM
-ESCITALOPRAM
-FLUOXETINE
-SETRALINE
-FLUROXAMINE
-PAROXETINE

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18
Q

WHAT IS PHARMACOLOGICAL CLASSIFICATION OF VENLAFAXINE

A

SEROTONIN NORADRENALINE REUPTAKE INHIBITOR

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19
Q

WHAT IS MOA OF DESVENLAFAXINE

A

BLOCK SEROTONIN AND NORADRENALINE REUPTAKE TRANSPORTER

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20
Q

LIST SNRI DRUGS

A

DULOXETINE
VENLAFAXINE
DESVENLAFAXINE

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21
Q

LIST ANTI EPILEPTIC DRUGS

A

PHENYTOIN
CARBAMAZEPINE
SODIUM VALPORATE
LAMOTRIGINE
LEVETIRACETAM

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22
Q

WHAT IS PHENYTOIN SIDE EFFECTS

A

HIRSUTISM
GINGIVAL HYPERPLASIA
CLEFT PALATE

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23
Q

WHAT IS CARBAMAZEPINE SIDE EFFECTS

A

DIPLOPIA
JAUNDICE
BRUISING

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24
Q

WHAT DRUGS IS TOXICITY TO PREGNANT WOMAN AND WHY

A

SODIUM VALPORATE
IT DISRUPT FOLATE METABOLISM LEAD TO NEURAL TUBE DEFECT

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25
WHAT DRUGS IS SAFE FOR PREGNANCY AND ANY ADVICE TO PATIENT
CARBAMAZEPINE LAMOTRIGINE PATIENT SHOULD TAKE ACID FOLID SUPPLEMENT AND VITAMIN K INJECTION
26
WHAT IS PHARMACOLOGICAL CLASSIFICATION OF ALPRAZOLAM
BENZODIAPINE
27
WHAT IS MOA OF DIAZEPAM
ENHANCE GABA EFFECTS HENCE REDUCE OVEREACT IN NERVOUS SYSTEM
28
WHAT IS POSSIBLE EFFECTS PATIENT WILL HAVE WHEN PRESCRIBES WITH LORAZEPAM
FALLS SEDATION DEPENDENCE
29
LIST BENZODIAPINES DRUGS
ALPRAZOLAM LORAZEPAM DIAZEPAM MIDAZOLAM CHLODIAZEPOXIDE
29
WHAT IS MIDAZOLAM INDICATION FOR
ANXIETY AND INSOMNIA
30
LIST DRUGS IN Z DRUGS PHARMACOLOGICAL CLASS
ZALEPION ZOLPIDEM ZOPICLONE
31
WHAT IS MOA OF ZALEPION
ENHANCE GABA EFFECTS BY BINDING TO ANOTHER SIDE OF RECEPTOR
32
WHAT INDICATION ARE WHEN PATIENT WAS PRESCRIBED WITH BUSPIRONE
ANXIETY
33
WHAT MOA OF BUSPIRONE
INCREASED SEROTONIN LEVEL
34
LIST GENERAL ANESTHETIC THAT WAS AVAILABLE AS IV DRIPS
PRPOFOL THIOPENTAL SODIUM ETOMIDATE KETAMINE
35
WHAT IS GENERAL ANESTHETIC THAT AVAILABLE AS INHALED GAS
ISOFLURANE SEROFLURANE DESFLURANE NITROUS OXIDE
36
LIST LOCAL ANESTHETIC
LIDOCAINE NOVOCAINE BENZOCAINE TETRACAINE BUPIVACAINE
37
WHAT IS PHARMACOLOGICAL CLASSIFICATION OF DONEPEZIL
ANTI CHOLINESTERASE IN ALZHEIMER'S
38
WHAT IS MOA OF GALANTAMINE
INHIBIT CHOLINESTERASE ENZYME MORE ACETYLCHOLLINE AVAILABLE
39
WHAT IS RIVASTAGMINE POSSIBLE SIDE EFFECTS
LOSS APETITE NAUSEA VOMITTING
40
WHAT IS PHARMACOLOGICAL CLASSIFICATION OF MEMANTINE
NMDA RECEPTOR ANTAGONIST
41
WHAT IS MOA OF MEMANTINE
INHIBIT NMDA RECEPTOR DECREASED LECEL OF GLUTAMATE HENCE REDUCE EXCITOTOXICITY AND NEURON DEATH
42
WHAT IS MOA OF LEVODOPA
ENSURING DOPAMINE CAN PASS THORUGH BLOOD BRAIN BARRIER
43
WHAT IS PHARMACOLOGICAL CLASS OF LEVODOPA
DOPAMINE PRECUSOR ANTI PARKINSON
44
WHY DID LEVODOPA WAS USED AS LAST TREATMENT OF PARKINSON
IT GIVING DYSKINESIA,WEARING OFF AND ON-OFF SIDE EFFECTS
45
WHAT DRUGS THAT WAS USED SYNERGERSTICALLY WITH LEVODOPA AND STATE THEIR PHARMACOLOGICAL CLASS
CARBIDOPA BENSERAZIDE -DECARBOXYLASE INHIBITOR
46
WHAT IS MOA OF CARBIDOPA
REDUCE CONVERSION OF LEVODOPA INTO DOPAMINE TO REDUCE LEVODOPA LONG TERM SIDE EFFECT
47
WHAT DRUGS IS LISTED UNDER MAOB INHIBITOR IN ANTI PARKINSON
SELEGILINE RASAGILINE
48
WHAT IS MOA OF RASAGILINE
INHIBIT MAOB ENZYME THAT HELP IN DEGRADATION OF DOPAMINE HENCE MORE DOPAMINE AVAILABLE INSIDE BRAIN
49
WHAT IS ENTACAPONE MOA
INHIBIT COMT ENZYME THAT HELP IN DEGRADATION OF LEVODOPA MORE LEVODOPA AVAILABLE OUTSIDE BRAIN
50
WHAT IS PHARMACOLOGICAL CLASSIFICATION OF TOLCAPONE
COMT INHIBITOR ANTI PARKINSON
51
WHAT IS AMANTADINE MOA
MIMICKING DOPAMINE EFFECTS IN OUR BRAIN
52
WHAT IS PHARMACOLOGICAL CLASSIFICATION OF PIRIBEDIL
DOPAMINE AGONIST
53
WHY IS PATIENT CANT CONTROL THEIR HABIT SUCH AS SHOPPING WHEN PRESCRIBED WITH PRAMIPEXOLE
GIVING SUDDEN IMPULSE CONTROL SIDE EFFECTS
54
WHAT DRUG IN DOPAMINE AGONIST ANTI PARKINSON
BROMOCLIPTINE AMANTADINE PIRIBEDIL PRAMIPEXOLE
55
WHAT IS PROCYCLIDINE MOA
REDUCE ACETYLCHOLINE HENCE BALANCING DOPAMINE LEVEL
56
WHAT IS PHARMACOLOGICAL CLASSIFICATION OF TRIHEXYLPHENIDYL
ANTI MUSCARINIC
57
WHAT IS MOA OF METFORMIN
REDUCE GLUCOGENESIS INCREASE INSULIN SENSITIVITY REDUCE GLUCOSE ABSORPTION
58
WHAT DRUGS IS IN SULPHONYLUREAS
GLICAZIDE GLIMEPIRIDE
59
WHAT IS MOA OF GLICAZIDE
INCREASE INSULIN PRODUCTION IN PANCREAS
60
THE POSSIBLE SIDE EFFECTS OF GLIMEPIRIDE
HYPOGLYCEMIA AND WEIGHT GAIN
61
WHAT IS MOA OF ACARBOSE
DELAY CARBOHYDRATES DIGESTION SLOW DOWN GLUCOSE ABSORPTION
62
WHAT IS ADVICE SHOULD BE GIVEN TO PATIENT WHEN TAKE ACARBOSE
USE SANITARY PAD ON MORNING TAKE WITH MOUTHFUL OF LIQUID OR FOOD
63
LIST DRUG UNDER DIPEPTIDYL-PEPTIDASE 4 INHIBITOR (DPP4i)
SITAGLIPTIN VILDAGLIPTIN LINAGLIPTIN
64
VILDAGLIPTIN MOA
INHIBIT INCRETIN BREAKDOWN HELPS IN INCREASING INSULIN SECRETION SLOW DOWN GLUCOSE ABSORPTION
65
LINAGLIPTIN SIDE EFFECTS
HYPOGLYCEMIA
66
DRUGS UNDER GLUCAGON-LIKE PEPTIDE -1 RECEPTOR
LIRAGLUTIDE DULAGLUTIDE SEMAGLUTIDE EXENATIDE LIXISENATIDE
67
LIXISENATIDE MOA
MIMICS INCRETIN FUNCTION SLOW DOWN GLUCOSE ABSORPTION INCREASE INSULIN SECRETION
68
SEMAGLUTIDE SIDE EFFECTS
WEIGHT LOSS
69
METFORMIN SIDE EFFECTS
WEIGHT LOSS PERIPHERAL NEUROPAHTY
70
WHAT IS PHARMACOLOGICAL CLASS OF EMPAGLIFLOZIN
SODIUM GLUCOSE 2 TRANSPORTER INHIBITOR
71
WHAT CANAGLIFLOZIN MOA
SELECTIVE INHIBIT SODIUM GLUCOSE 2 TRANSPORTER IN KIDNEY REDUCE GLUCOSE READSORPTION INTO BLOOD INCREASE INSULIN EXCRETION IN URINE
72
POSSIBLE EFFECT OF DAPAGLIFLOZIN
UTI WEIGHT LOSS DEHYDRATION
73
BENEFIT OF CANAGLIFLOZIN
CARDIOPROTECTIVE HEART FAILURE TREAMENT RENOPROTECTIVE
74
INSULIN MOA
FACILITATE GLUCOSE UPTAKE BY BODY CELL FROM BLOOD
75
INSULIN SIDE EFFECT
HYPOGLYCEMIA FAT ACCUMULATION WEIGHT GAIN
76
HYPOTHYROID DRUG
LEVOTHYROXINE THYEOXINE SODIUM LITHYROXINE SODIUM INJECTION
77
LEVOTHYROXINE MOA
REPLACE NATURAL HORMON THYROID
78
ADVICE WHEN TAKING LEVOTHYROXINE
ON MORNING ONCE DAILY 30 MINS BEFORE BREAKFAST OR CAFFIENE
79
HYPERTHYROID DRUGS
CARBIMAZOLE PROPYLTHIOURACIL
80
PROPYLTHIOURACIL MOA
REDUCE THYROID HORMONE PRODUCATION
81
WHY IS CARBIMAZOLE IS DANGER DRUG
CAUSE BIRTH DEFECT
82
LIST COMBINED ORAL CONTRACEPTIVES
YASMIN YAZ QLAIRA NORDETTE MARVELON MERECILON COTTE DIANE 35
83
DIANE 35 MOA
PREVENT OVULATION THICKEN CERVICAL MUCUS PREVENT SPERM REACHS OVUM
84
IS QLAIRA SAFE FOR PREGNANCY AND WHY
NO. INCREASED BLOOD CLOT
85
WHAT IS NORIDAY MOA
THICKEN CERVICAL MUCUS THINNING UTERINE LINE
86
IS CERAZETTE SAFE IN PREGNANCY
YES
87
EXPLAIN EMERGENCY PILLS AND EXAMPLE
POSTINOR-2 AND ESCAPELLE WILL DELAYS OVULATION WITHIN 72 HOURS ELLAONE BLOCK OVULATION WITHIN 120 HOURS
88
LIST ACUTE MIGRAINE TREATMENT
SUMATRIPTAN ALMOTRIPTAN ZOLMITRIPTAN RIZATRIPTAN ERGOTAMINE CAFFIENE
89
WHAT IS SUMATRIPTAN MOA
ACTIVATE SEROTONIN RECEPTOR HENCE LESS RELEASE NEUROPEPTIDE LESS NOCICEPTOR ACTIVATION AND VASODILATION
90
ZOMITRIPTAN SIDE EFFECTS
HOT FLUSHING SENSATION DROWSY
91
EXPLAIN HOW SHOULD WE TAKE MIGRAINE TREATMENT
WHEN MIGRAINE SYPMTOPS OCCUR TAKING NSAID OR PAIN KILLER ASAP WHEN MIGRRAINE START TO ATTACK TAKE TRIPTAN DRUGS
92
WHAT IS MOA OF CORTICOSTEROID
REDUCE INFLAMMATION AND MODULATE IMMUNE SYSTEM
93
WHAT IS BETHAMETHAOSONE SIDE EFFECTS IF USE LONG TERM
OSTEOPOROSIS CUSHING SYNDROME BETHAMETHASONE HIGH POTENCY TOPICAL CREAM.
94
STEROID FUNCTION
ENHANCE RECOVERY AND REDUCE FATIGUE MIMICS MALE SEX HORMONE AND PROMOTE TISSUE AND MUSCLE GROWTH.
95
EXAMPLE OF STEROID
TESTERONE NANDRONOLE STANOZOL METHENOLONE
96
CORTICOSTEROID EXAMPLE
HYDROCORTISONE PREDNISOLONE DEXAMETHASONE BUDESONIDE