Drugs classification Flashcards
Isocarboxazid
MAOI (AD)
Phenelzine
MAOI (AD)
Tranylcypromine
MAOI (AD)
Selegiline
MAOI (AD)
Cyproheptadine
Serotonin antagonist
- Serotonin syndrome
Pseudoephedrine & Phenylpropanolamine
Cheese Reaction
- OTC cold preparations contraindicated in pts. taking MAOI
Phentolamine & Prazosin
Manage Tyramine-induced hypertension
Amitriptyline
TCA (AD)
Clomipramine
TCA (AD)
Desipramine
TCA (AD)
Imipramine
TCA (AD)
Nortriptyline
TCA (AD)
Sodium Bicarbonate
Reverses Conduction block caused by TCA overdose
Citalopram
SSRI (AD)
Escitalopram
SSRI (AD)
Fluoxetine
SSRI (AD)
Paroxetine
SSRI (AD)
Sertraline
SSRI (AD)
Fluvoxamine
SSRI (AD)
Nefazodone
SARI (AD)
Trazodone
SARI (AD)
Venlafaxine
SNRI (AD)
Duloxetine
SNRI (AD)
Buproprion
NDRI (AD)
Mirtazapine
NaSSA (AD)
Lithium
Bipolar DOC
Amiloride
Treat nephrogenic DI caused by Lithium
Valproate & Carbamazepine & Lamotrigine
Antiepileptic - Alternatives to Lithium
+ Atypical antipsychotics
Phenytoin
Voltage-gated Na+ channel blockers (AE)
Carbamazepine
Voltage-gated Na+ channel blockers (AE)
Lamotrigine
Voltage-gated Na+ channel blockers (AE)
Zonisamide
Voltage-gated Na+ channel blockers (AE)
Phenobarbital
Effects may be contributed by Voltage-gated Na+ channel blockers (AE)
Valproate
Effects may be contributed by Voltage-gated Na+ channel blockers (AE
Topiramate
Effects may be contributed by Voltage-gated Na+ channel blockers (AE
Ethosuximide
T-type Ca2+ channel blockers
Valproate
T-type Ca2+ channel blockers
Tiagabine
GABA reuptake inhibitor
Vigabatrin
GABA aminotransferase (degradation) inhibitor
Phenobarbital
Topiramate
Gabapentin
Presynaptic voltage-gated Ca2+ channel blockers (AE)
Pregabalin
Presynaptic voltage-gated Ca2+ channel blockers (AE)
Levetiracetam
Chlopromazine
Classical AP
Fluphenazine
Classical AP
Haloperidol
Classical AP
Thioridazine
Classical AP
Clozapine
Atypical Ap
Risperidone
Atypical AP
Olanzapine
Atypical AP
Quetiapine
Atypical AP
Aripiprazole
Atypical AP
Pimavanserin
Atypical AP
Levodopa
Dopamine Precursor- Restore dopamine actions
Carbidopa
Dopa Decarboxylase inhibitor
Sinemet
Levodopa + Carbidopa formula
Apomorphine
Non-selective dopamine agonists - used to treat On-Off phenomenon of Levodopa
Bromocriptine
Ergot Dopamine Agonist
Dopamine Receptor Agonists- Restore dopamine actions
Pramipexole
Non-Ergot Dopamine Agonist
Dopamine Receptor Agonists- Restore dopamine actions
Ropinirole
Ergot Dopamine Agonist
Dopamine Receptor Agonists- Restore dopamine actions
Rotigotine
Ergot Dopamine Agonist
Dopamine Receptor Agonists- Restore dopamine actions
Apomorphine
Non-Ergot Dopamine Agonist
Dopamine Receptor Agonists- Restore dopamine actions
Trimethobenzamide
Antiemetic used as pretreatment for Apomorphine use
Rasagiline
MAOI (Inhibitor of Dopamine metabolism for Parkinson treatment)
Selegiline
MAOI (Inhibitor of Dopamine metabolism for Parkinson treatment)
Tolcapone
COMT Inhibitor (Inhibitor of Dopamine metabolism for Parkinson treatment)
Entacapone
COMT Inhibitor (Inhibitor of Dopamine metabolism for treatment)
Amantadine
NMDA receptor antagonist
Antiviral drug used for Anti-Parkinson actions
Benztropine
Antimuscarinic used as adjunct therapy for Parkinson