Drugs Flashcards
Bethancol
Direct muscarininc agonist
Carbachol
Directs acting muscarinic agonist
Methacholine
Direct acting muscarininc agonist
Pilocarpine
Direct acting muscarinic agonist
Physostigmine
Ach Esterase inhibitor
Pyridostigmine
Ach Esterase inhibitor
Neostigmine
Ach Esterase inhibitor
Galantamine
Ach Esterase inhibitor
Donepezil
Ach Esterase inhibitor
Rivastigmine
Ach Esterase inhibitor
Echothiophate
Ach esterase inhibitor
Malathion
Ach Esterase inhibitor
Sarin
Ach Esterase inhibitor
Pralidoxime
Antidote to AchE poisoning
Reactivates AchE
Atropine
Muscarinic antagonist
Glycopyrrolate
Muscarinic antagonist
Benztropine
Mus Antag
Darifenacin
Mus antag
Oxybutynin
Mus antag
Tolterodine
Mus Antag
Dicyclomine
Mus antag
Hyoscyamine
Mus antag
Ipratropium
Mus antag
Tiotropium
Mus antag
Tropicamide
Mus antag
Scopolamine
Mus antag
Mecamylamine
Ganglionic blocker
Varenicline
Nicotinic Partial agonist
Used to treat post op urinary retention or ileus
Bethanchol
Used to treat glaucoma and to induce miosis during surgery. Has some nicotinic activity in ganglia.
Carbachol
Used for Xerostomia and Sjogrens Syndrome
Pilocarpine
Challenge test for bronchial hyperactivity diagnosis
Methacholine
AchE inhibitor that crosses the BBB to get in to the CNS
Phy-sostigmine
AchE inhibitor used to treat myasthenia gravis
Neostigmine and Pyri-dostigmine
Irreversible drug used to treat glaucoma
Echothiophate
Used to treat Parkinson’s
Benzotropine
Used to treat overactive bladder
Darifenacin
Oxybutynin
Used as a GI spasmolytic (used to treat diarrhea)
Dicycloamine
Hyoscyamine
Used to treat asthma
Ipratropium Tiotropium
Mydriatic and Cycloplegia
Tropicamide
Motion sickness
Scopolamine