CYP3A4 Inducers, Inhibitors, and Substrates Flashcards
1
Q
topiramate
A
Inducer
2
Q
erythromycin
A
Substrate and Inhibitor*
3
Q
phenobarbital
A
Inducer
4
Q
grapefruit
A
Inhibitor**
5
Q
prednisone
A
Inducer
6
Q
phenytoin
A
Inducer
7
Q
ziprasidone
A
Substrate
8
Q
ranolazine
A
Substrate and Inhibitor
9
Q
ketoconazole
A
Substrate and Inhibitor**
10
Q
hydrocodone
A
Substrate
11
Q
nifedipine
A
Substrate and Inhibitor
12
Q
pioglitazone
A
Inducer
13
Q
linagliptin
A
Substrate
14
Q
carbamazepine
A
Substrate and Inducer
15
Q
alprazolam
A
Substrate
16
Q
dexamethasone
A
Substrate and Inducer
17
Q
salmeterol
A
Substrate
18
Q
aripiprazole
A
Substrate
19
Q
tramadol
A
Substrate
20
Q
amitriptyline
A
Substrate
21
Q
lovastatin
A
Substrate
22
Q
verapamil
A
Substrate and Inhibitor*
23
Q
colchicine
A
Substrate
24
Q
fluoxetine
A
Inhibitor
25
fluvoxamine
Inhibitor
26
iloperidone
Substrate
27
cimetidine
Inhibitor
28
haloperidol
Substrate
29
amiodarone
Substrate and Inhibitor
30
venlafaxine
Substrate
31
felodipine
Substrate
32
voriconazole
Substrate and Inhibitor**
33
clozapine
Substrate
34
St. John’ s wort
Inducer
35
(R)-warfarin
Substrate
36
levonorgestrel
Substrate
37
buspirone
Substrate
38
modafinil
Inducer
39
methylprednisolone
Substrate
40
posaconazole
Inhibitor**
41
quetiapine
Substrate
42
repaglinide
Substrate
43
saxagliptin
Substrate
44
buprenorphine
Substrate
45
amlodipine
Substrate and Inhibitor
46
sertraline
Substrate
47
clarithromycin
Substrate and Inhibitor**
48
brexpiprazole
Substrate
49
citalopram
Substrate
50
isoniazid
Inhibitor
51
atorvastatin
Substrate
52
oral contraceptives
Substrate
53
fluconazole
Inhibitor*
54
Viekira Pak
Substrate
55
ritonavir
Substrate Inhibitor** and Inducer
56
trazodone
Substrate
57
eplerenone
Substrate
58
estrogens
Substrate
59
omeprazole
Substrate
60
etonogestrel
Substrate
61
diltiazem
Substrate and Inhibitor*
62
midazolam
Substrate
63
rifampin
Inducer
64
oxycodone
Substrate
65
fentanyl
Substrate
66
nefazodone
Substrate and Inhbitor**
67
dextromethorphan
Substrate
68
ciprofloxacin
Inhibitor*
69
itraconazole
Substrate and Inhibitor**
70
dronedarone
Inhibitor*
71
ethinyl estradiol
Substrate and Inhibitor
72
diazepam
Substrate
73
oxcarbazepine
Inducer
74
simvastatin
Substrate
75
lomitapide
Substrate
76
telithromycin
Substrate and Inhibitor**
77
esomeprazole
Substrate
78
triazolam
Substrate
79
lurasidone
Substrate
80
rivaroxaban
Substrate