CYP1A2 Flashcards
1
Q
Montelukast
A
CYP1A2 Inducer
2
Q
Mirtazapine
A
CYP1A2 Substrate
3
Q
Phenobarbital
A
CYP1A2 Inducer
4
Q
Carbamazepine
A
CYP1A2 Inducer
5
Q
Zafirlukast
A
CYP1A2 Inhibitor
6
Q
Roflumilast
A
CYP1A2 Substrate
7
Q
R-warfarin
A
CYP1A2 Substrate
8
Q
Smoking
A
CYP1A2 Inducer
9
Q
Caffeine
A
CYP1A2 Substrate and Inhibitor
10
Q
Ramelteon
A
CYP1A2 Substrate
11
Q
Fluvoxamine**
A
CYP1A2 Inhibitor
12
Q
Oral contraceptives*
A
CYP1A2 Inhibitor
13
Q
Duloxetine
A
CYP1A2 Substrate
14
Q
Ethinyl estradiol*
A
CYP1A2 Inhibitor
15
Q
Rifampin
A
CYP1A2 Inducer
16
Q
Olanzapine
A
CYP1A2 Substrate
17
Q
Melatonin
A
CYP1A2 Substrate
18
Q
Allopurinol
A
CYP1A2 Inhibitor
19
Q
Phenytoin
A
CYP1A2 Inducer
20
Q
Propranolol
A
CYP1A2 Substrate and Inhibitor
21
Q
Clozapine
A
CYP1A2 Substrate
22
Q
Theophylline
A
CYP1A2 Substrate
23
Q
Verapamil
A
CYP1A2 Inhibitor
24
Q
Ritonavir
A
CYP1A2 Inducer
25
Zileuton\*
CYP1A2 Inhibitor
26
Amiodarone
CYP1A2 Inhibitor
27
Omeprazole
CYP1A2 Inducer
28
Methadone
CYP1A2 Substrate
29
Ciprofloxacin\*\*
CYP1A2 Inhibitor
30
Isoniazid
CYP1A2 Inhibitor
31
Acyclovir
CYP1A2 Inhibitor
32
Zolmitriptan
CYP1A2 Substrate
33
Cimetidine
CYP1A2 Inhibitor
34
Famotidine
CYP1A2 Inhibitor