CYP anti-épileptiques Flashcards

1
Q

Phénytoïne

A

Induction : 2C, 3A
Inhibition :
Substrat : 2C9, 2C19

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2
Q

CBZ

A

Induction : 2C9, 3A
Inhibition :
Substrat : 1A2, 2C8, 2C9, 3A4

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3
Q

Zarontin

A

Induction :
Inhibition :
Substrat : 3A4

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4
Q

Phénobarbital

A

Induction : 2C, 3A
Inhibition :
Substrat : 2C9, 2C19

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5
Q

Valproate

A

Induction :
Inhibition : UGT, 2B7, 2C9
Substrat : 2C9, 2C19, UGT

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6
Q

Lamotrigine

A

Induction :
Inhibition :
Substrat : UGT

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7
Q

Oxcarbamazépine

A

Induction : 3A4
Inhibition : 2C19
Substrat : UGT

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8
Q

Zonisamide

A

Induction :
Inhibition :
Substrat : 3A4

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9
Q

Tiagabine

A

Induction :
Inhibition :
Substrat : 3A4

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10
Q

Topiramate

A

Induction : 3A4
Inhibition : 2C19
Substrat : 3A4, UGT

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11
Q

Lacosamide

A

Induction :
Inhibition :
Substrat : 2C19

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12
Q

Perampanel

A

Induction :
Inhibition :
Substrat : 3A4

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13
Q

Eslicarbamazépinde

A

Induction : 2C9
Inhibition :
Substrat : UGT

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14
Q

Ezogabine

A

Induction :
Inhibition :
Substrat : +++

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