Anticholinergic Agents Flashcards
Atropine
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Scopolamine
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Homatropine (generic, Isopto Homatropine)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Pirenzepine
Anticholinergic Agent
Muscarinic antagonist
- Tertiary amine (CNS accessible)
- M-3 SELECTIVE
Tropicamide (generic, Mydriacyl Opthalmic, etc.)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Tolterodine (Detrol)
Anticholinergic Agent
Muscarinic antagonist
- Tertiary amine (CNS accessible)
- M-3 SELECTIVE
Dicyclomine (Bentyl)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Fesoteridine (Toviaz)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Mepenzolate (Cantil)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Solifenacin (Vesicare)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Oxybutynin (Ditropan, Oxytrol)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Darifenacin (Emablex)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Trospium (Spasmex)
Anticholinergic Agent
Muscarinic antagonist
-Tertiary amine (CNS accessible)
Atropine methyl nitrate
Anticholinergic Agent
Muscarinic antagonist
-Quaternary amine (not able to cross blood-brain barrier)
Methscopolamine (generic, Pamine)
Anticholinergic Agent
Muscarinic antagonist
-Quaternary amine (not able to cross blood-brain barrier)
Ipratropium (generic, Atrovent)
Anticholinergic Agent
Muscarinic antagonist
-Quaternary amine (not able to cross blood-brain barrier)
Propantheline (generic, Pro-Banthine, others)
Anticholinergic Agent
Muscarinic antagonist
-Quaternary amine (not able to cross blood-brain barrier)
Glycopyrrolate (generic, Robinul)
Anticholinergic Agent
Muscarinic antagonist
-Quaternary amine (not able to cross blood-brain barrier)
Hexamethonium
Anticholinergic Agent
Ganglionic blocker
Trimethaphan (Arfonad)
Anticholinergic Agent
Ganglionic blocker
*lacks CNS effects
Mecamylamine (Inversine)
Anticholinergic Agents
Ganglionic blocker
Pralidoxime (2-PAM) (general, Protopam)
Anticholinergic Agent
Cholinesterase regenerator