Anti Malarial Flashcards
Blood
Chloroquine Amodiaquine Quinine Pyrimethamine Lumefantrine Artemisinin
Tissue
Primaquine
Pre erythrocytic
Pyrimethamine
Primaquine
Proguanil
Gameocidal
Vivax: quinine
Falciparum: primaquine
Sporontocoides
Primaquine
Choroguanide
8-aminoquinolone
Primaquine
Gametocyte for all four plasmodia
Primaquine
AE of primaquine
Hemolytic anemia for G6PD Deficiency
Abdominak pain with chloroquine
Methhemoglobinemia
CI Pregnancy
4 aminoquinolone
Chloroquine
Mainstay of antimalarial therapy
Chloroquine
Also used for Amoebiasis
Chloroquine
AE of chloroquine
Rash
Headache
Blurred vision
Multidrug resistant falciparum
Mefloquine
AE of Mefloquine
Dizziness Confusions Hallucinations Depression ECG abnormality with quinine
Interfere with heme polymerization
Quinine and Quinidine
Cinchonism
Quinine and Quinidine
Vomitting, vertigo, tittinus
Severe multidrug resistant malria
Artemisinin
High doses of artemisinin
Neurotoxicity and QT prolongation
Dihyrdofolate reductase inhibitor (reduces tetrahydrofolate)
Pyrimethamine
Prophylaxis for pregnant women
Sulfadoxine
Pyrimethamine
Prevention in chloroquine resitsbt malaria
Doxycycline
Mefloquine
Malarone (atovaquone+proguanil)