Adrenergic Drugs Flashcards

1
Q

Direct Adrenergic Agonists

A
Alpha:
  Phenylephrine
  Clonidine
Mixed alpha and beta:
  NE
  Epi
Beta:
  Dobutamine
  Isoproterenol
  Albuterol
Dopamine
  Fenoldopam
How well did you know this?
1
Not at all
2
3
4
5
Perfectly
2
Q

Phenylephrine

A

a1>a2 agonist

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
3
Q

Clonidine

A

a2>a1 agonist

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
4
Q

Norepinephrine

A

a1, a2, B1 agonist

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
5
Q

Epinephrine

A

a1, a2, B1, B2 agonist

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
6
Q

Dobutamine

A

B1>B2 agonist

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
7
Q

Isoproterenol

A

B1, B2 agonist

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
8
Q

Albuterol

A

B2»B1 agonist

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
9
Q

Dopamine

A

D1, D2 agonist
D1: vasodilation of Renal, Cerebral, Mesenteric, and Coronary arteries. Fenoldopam.
D2: inhibits NE release

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
10
Q

Indirect Adrenergic Agonists

A
Cocaine
Phenelzine
Selegiline
Amphetamine
Methylphenidate
Ephedrine
Tyramine
How well did you know this?
1
Not at all
2
3
4
5
Perfectly
11
Q

Cocaine

A

DA/NE reuptake inhibitor

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
12
Q

Phenelzine

A

MAO inhibitor
Incr. NE in CNS
Antidepressant

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
13
Q

Amphetamine

A

DA/NE reuptake inhibitor
Increases release of DA & NE
ADHD

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
14
Q

Selegiline

A

MAO inhibitor
Incr. NE in CNS
Antidepressant

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
15
Q

Methylphenidate

A

DA/NE reuptake inhibitor
Increases release of DA & NE
ADHD

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
16
Q

Ephedrine

A

Indirect general agonist, releases stored NE/DA

17
Q

Tyramine

A

Release of stored NE.

Risk of incr BP with MAOIs

18
Q

Adrenergic Antagonists

A
Alpha nonselective:
  Phentolamine
  Phenoxybenzamine
Alpha 1: 
  -osin
Mixed: a1, B1, B2
  Labet-alol
  Carved-ilol
Beta:  -olol
  B1 selective = A to M
  Nonselective = N to Z
19
Q
Acebutolol
Atenolol
Betaxolol
Bisoprolol
Esmolol
Metoprolol
A

B1 antagonist

20
Q

Nadolol
Pindolol
Propranolol
Timolol

A

B1, B2 antagonist

21
Q

Beta Blocker Antagonists

A
ANtagonistic PeanutButter
Atenolol
Nadolol
Propranolol
Betaxolol
22
Q

Beta Blocker Partial Agonists

A

PArtiaL
Pindolol
Acebutolol
Labetalol

23
Q

Beta Blocker Inverse Agonists

A

CM
Carvedilol
Metoprolol