2C19 Flashcards
Apalutamide
Strong inducer
Efavirenz
Moderate Inducer, Inhibitor
Enzalutamide
Moderate inducer
Rifampicin
Strong inducer
Ritonavir
Strong inducer
St john’s wort
Inducer
Clarithromucin
inhibitor
Esomeprazole
Inhibitor
Etravirine
Inhibitor, Substrate
Fluconazole
Strong inhibitor
Fluoxetine
Strong inhibitor
Fluvoxamine
Strong inhibitor
Ketoconazole
inhibitor
Omeprazole
Inhibitor, Substrate
Oxcarbazepine
Inhibitor
Stiripentol
Inhibitor, Substrate
Topiramate
Inhibitor
Voriconazole
Moderate inhibitor, Substrate
Amitriptyline
Substrate
Axitinib
Substrate
Bortezomib
Substrate
Brivaracetam
Substrate
Cannabidol
Substrate
Citalopram
Substrate
Clopidogrel
Substrate
Cyclophosphamide
Substrate
Diazepam
Substrate
Escitalopram
Substrate
Imipramine
Substrate
Lansoprazole
Substrate
Mavacamtem
Substrate
Pantoprazole
Substrate
Phenobarbital
Substrate
Phenytoin
Substrate
Propranolol
Substrate
Warfarin (R-isomer)
Substrate