1 Flashcards
albuterol
beta 2 agonist
timolol
non-selective beta blocker
betaxalol
selective beta 1 blocker
levobunolol
non selective beta blocker
carteolol
non selective beta blocker
metipranolol
non selective beta blocker
latanoprost
topical PG
travoprost
tropical PG
pralidoxime
cholinesterase reactivator
obidoxime
cholinesterase reactivator
homatropine
mydriatic atropine derivative
cyclopentolate
mydriatic atropine derivative
tropicamide
mydriatic atropine derivative
ipratropium
copd bronchial asthma atropine derivative
tiotropium
copd bronchial asthma atropine derivative
pirenzepine
atropine derivative used in peptic ulcer
telenzepine
atropine derivative used in peptic ulcer
clidinium
atropine derivative used in peptic ulcer
propanthelin
atropine derivative used in peptic ulcer
dicylomine
atropine derivative as antispasmodic
valthamate
atropine derivative as antispasmodic
flavoxate
atropine derivative as antispasmodic
oxybutinin
atropine derivative as antispasmodic
tolterodine
atropine derivative as antispasmodic
darifenacine
atropine derivative as antispasmodic
glycopyrrolate
preanesthetic atropine derivative
benztropine
atropine derivative in Parkinson
benzhexol
atropine derivative in Parkinson
buperidine
atropine derivative in Parkinson
procyclidine
atropine derivative in Parkinson
vesicoselective anticholinergic
oxybutinin (dry mouth), flavoxate (inflammation), tolterodine, darifenacun M3
drotavarine
pde inhibition
antispasmodic
uterine spasm relief/ intestinal, renal colic relief
glycopyrrolate
quaternary atropine
scopolamine
anticholinergic in motion sickness
anticholinergic side effects
antihistamines h1, TCA, phenothiazine-
postural hypotension
ganglionic blockade
Bupropion
inhibits NE DA uptake
varenicline
nicotinic partial agonist
trimethaphan iv
ganglionic blockade
trimethaphan iv
ganglionic blockade
trimethaphan iv
ganglionic blockade
trimethaphan iv
ganglionic blockade
trimethaphan iv
ganglionic blockade
trimethaphan iv
ganglionic blockade
baclofen
GABA B agonist (centrally acting sk ms relaxant)
diazepam
GABA A (centrally acting sk ms relaxant)
tizanidine
central alpha 2 agonist (centrally acting sk ms relaxant)
chlorzoxazone
spinal neurons (centrally acting sk ms relaxant)
methocarbamol
spinal neurons (centrally acting sk ms relaxant)(centrally acting sk ms relaxant)
riluzole
inhibits glutamate (centrally acting sk ms relaxant)(centrally acting sk ms relaxant)
thiocolchicoside
(centrally acting sk ms relaxant)(centrally acting sk ms relaxant)
succinyl Choline
depolarising blocker - two phase block
fasiculation
receptor configuration changes so Ach can’t bind
decamethonium
depolarising blocker - two phase
fasiculation
receptor configuration chnages - Ach can’t bind. cholinesterase partially reverse it
tubocurarine
non depolarising blocker, histamine releaser
pancuronium
non depolarising blocker - vagolytic
histamine releaser non depolarising blocker
tubocurarine, atracurium, mivacurium
doxacurium
non depolarising blocker
pipecuronium
non depolarising blocker, bradycardia, hypotension
vecuronium
most common non depolarising blocker
atracurium
non depolarising blocker (hoffman elimination+ pseudocholinesterase)
cisatracurium
non depolarising blocker - better than atracurium
rocurium
non depolarising blocker
mivacurium
short duration non depolarising blocker - pseudocholinesterase degradation
dobutamine
beta 1 agonist
salbuterol
beta 2 agonist
formeterol
beta 2 agonist
salbuterol
beta 2 agonist
terbutaline
beta 2 agonist
isoxsprine
beta 2 agonist
ritoderine
beta 2 agonist uterus
phenylephrine
alpha 1 agonist
methoximine
alpha 1 agonist
naphazoline
alpha 1 agonist
oxymetazoline
alpha 1 agonist
xylometazoline
alpha 1 agonist
clonidine
alpha 2 agonist
apraclonidine
alpha 2 agonist
alpha methyl dopa
alpha 2 agonist
brimodine
alpha 2 agonist
ephedrine
adrenergic agonist
increase NA
dopamine
alpha, beta1 , d1
indirect increase NA
mephentermine
increase NA
alpha 1 agonist
nasal decongestant
naphazoline, oxymetazoline, xylometazoline,
pseudoephedrine, phenylephrine antihistamines
tizanidine
alpha 2 agonist
d amphetamine
cns stimulation
l amphetamine
cvs stimulation
amphetamine
basic
poisoning- tx- sedatives, na nitroprusside
atomoxetine
SNRI
modafinil
cns stimulant
dopamine
low dose - d1 vasodilation
moderate dose - b1, d1
highdose - vc a1
fenoldopam
d1 agonist
mazindol
decrease NA reuptake
increase NA in brain
inhibit feeding centre
phentermine
inhibition of NA reuptake
feeding centre suppressed
sibutramine
inhibit NA, S reuptake
suppress appetite
orlistat
inhibit lipase
phentolamine
reversible non-selective alpha adrenergic blocker
tolazoline
reversible non-selective alpha adrenergic blocker
phenoxybenzamine
irreversible non-selective alpha adrenergic blocker
prazocin
alpha 1 blocker
terazocin
alpha 1 blocker
doxazocin
alpha 1 blocker