1 Flashcards
1
Q
olol
A
beta blocker
2
Q
muscarinic beta blockers can produce
A
xerostomia (see langley experiment)
3
Q
R*L/RL =
A
Kd = K-1/K1
4
Q
interaction of drugand receptor is based on law of
A
mass action - only use to describe drug binding, not action.
5
Q
Kd
A
concentration required for 1/2 maximal binding to receptor
6
Q
EC 50
A
dose of drug to get 1/2 max effect.
7
Q
EC 50 can be less than
A
Keq
8
Q
Efficacy
A
ability to do something
9
Q
Potency
A
Concentration where drug works. Efficacy and binding efficiency
10
Q
Drugs with no efficacy with high binding efficiency
A
antagonists
