Wirkstoff-Stichwörter Flashcards

1
Q

Acetylsalicylsäure

A

COX-Hemmstoff

NSAID, NSAR

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2
Q

Adrenalin

A

Neurotransmitter

Sympathikus

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3
Q

Aflatoxin

A

Metabolismus und toxischer Mechanismus

Toxikologie

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4
Q

Amphetamin

A

Transmitter-Freisetzung

Sympathikus

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5
Q

Atenolol

A

β1-Rezeptorblocker

Sympathikus

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6
Q

Atracurium

A

nAChR-Antagonist

Parasympathikus

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7
Q

Atropin

A

mAChR-Antagonist

Parasympathikus

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8
Q

Biperiden

A

mAChR-Antagonist

Parasympathikus

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9
Q

Botulinustoxin

A

Parasympatholytikum

Parasympathikus

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10
Q

Butylscopolamin

A

mAChR-Antagonist

Parasympathikus

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11
Q

Clonidin

A

α2-Agonist

Sympathikus

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12
Q

Cocain

A

Wiederaufnahmehemmer

Sympathikus

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13
Q

Dantrolen

A

Ryanodin-Rez. Antagonist

Calcium

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14
Q

Doxazosin

A

α1−Antagonist

Sympathikus

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15
Q

Entacapon

A

COMT-Hemmstoff

Sympathikus

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16
Q

Glyceroltrinitrat

A

Aktivierung Guanylatzyklase

Glatter Muskel

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17
Q

Isoprenalin

A

β-Agonist

Sympathikus

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18
Q

Methanol

A

Prodrug für Ameisensäure

Toxikologie

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19
Q

Methylphenidat

A

Transmitter-Freisetzung

Sympathikus

20
Q

MPTP

A

Neurotoxin

Toxikologie

21
Q

Neostigmin

A

AChE-Hemmstoff

Parasympathikus

22
Q

Organophosphate

A

AChE-Hemmstoff

Parasympathikus

23
Q

Oxymetazolin

A

α1-Agonist

Sympathikus

24
Q

Pancuronium

A

nAChR-Antagonist

Parasympathikus

25
Paracetamol
Giftung durch CYP | Toxikologie
26
Physostigmin
AChE-Hemmstoff | Parasympathikus
27
Pilocarpin
mAChR-Agonist | Parasympathikus
28
Prazosin
α-Blocker | Sympathikus
29
Propranolol
β-Blocker | Sympathikus
30
Scopolamin
mAChR-Antagonist | Parasympathikus
31
Selegilin
MAO-B-Hemmstoff | Sympathikus
32
Sildenafil
PDE-5-Hemmstoff | Glatter Muskel
33
Suxamethonium
AChR-Agonist | Parasympathikus
34
Terbutalin
β2-Agonist | Sympathikus
35
Trospiumchlorid
mAChR-Antagonist | Parasympathikus
36
Venlafaxin
Wiederaufnahmehemmer | Sympathikus
37
Xylometazolin
α1-Agonist | Sympathikus
38
β-Lactame
Penicilline (z.B. Amoxicillin), Carbapeneme (z.B. Imipenem), Cephalosporine (z.B. Cefuroxim), Clavulansäure
39
Glykopeptidantibiotika
Vancomycin
40
Sulfonamide
Cotrimoxazol (Trimethoprim)
41
Makrolide
Clarithromycin
42
Tetracycline
Doxycyclin
43
Fluorchinolone
(GyrasehCeimprmofelorx)acin
44
CYP3A4-Inhibitoren und Induktoren
* Ketoconazole * Itraconazole * Fluconazole * Cimetidine * Clarithromycin * Erythromycin * Troleandomycin * Grapefruit juice
45
Type I Prodrugs
anti-viral nucleoside analogs | lipid-lowering statins
46
Type II Prodrugs
salicin, | enzymes