W4/L3 Flashcards

1
Q

What drugs are allosteric modulators of the GABA-A receptor?

A

Benzodiazepines

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
2
Q

What an advantage of allosteric antagonism?

A

More selectivity between subtypes

Incomplete antagonism possible

How well did you know this?
1
Not at all
2
3
4
5
Perfectly
3
Q

What type of antagonism is usually surmountable?

A

Competitive reversible

How well did you know this?
1
Not at all
2
3
4
5
Perfectly