Serpe Gen Flashcards

1
Q

Agonisti

A

Pieno
Parziale
Inverso - metoprorolo
Selettivo e allosterico

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2
Q

Teorie

A

Occupazione
Doppio stato

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3
Q

Antagonisti

A

Competitivo - Anti H2
Nono competitivo/allosterico

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4
Q

Antagonismo farmaceutico

A

Chimico
Farmacocinetico
Non competitivi
Fisiologico

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5
Q

Curve dose reisposta

A

EC50
ED50 e LD50

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6
Q

Modulazione recettoriale

A

Astinenza
Rimbalzo

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7
Q

Desensibilazione
Tolleranza
Refrattarietà
Farmacoresistenza

A

Tolleranza per esaurimento o fisiologico
Bypass tramite nuovi cloni

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8
Q

Potenza
Efficacia
Indice
Margine

A

Ricordateli

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